Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10595357 | Bioorganic & Medicinal Chemistry Letters | 2012 | 7 Pages |
Abstract
A series of novel, non-steroidal AR antagonists were discovered through HTS. ADME profile was also improved by designing more ligand-efficient molecules.
Keywords
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Chuangxing Guo, Susan Kephart, Martha Ornelas, Javier Gonzalez, Angelica Linton, Mason Pairish, Asako Nagata, Samantha Greasley, Jeff Elleraas, Natilie Hosea, Jon Engebretsen, Andrea N. Fanjul,