| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 10596355 | Bioorganic & Medicinal Chemistry Letters | 2009 | 5 Pages |
Abstract
Synthesis and SAR studies of a novel series of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one derivatives as potent class of PARP-1 inhibitors are reported.
Keywords
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Federica Orvieto, Danila Branca, Claudia Giomini, Philip Jones, Uwe Koch, Jesus M. Ontoria, Maria Cecilia Palumbi, Michael Rowley, Carlo Toniatti, Ester Muraglia,
![First Page Preview: Identification of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one as potent poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors Identification of substituted pyrazolo[1,5-a]quinazolin-5(4H)-one as potent poly(ADP-ribose)polymerase-1 (PARP-1) inhibitors](/preview/png/10596355.png)