Article ID Journal Published Year Pages File Type
10596450 Bioorganic & Medicinal Chemistry Letters 2009 5 Pages PDF
Abstract
Modification of the benzo rings of 3-(1,1-dioxo-2H-(1,2,4)-benzothiadiazin-3-yl)-4-hydroxy-2(1H)-quinolinones into heteroaromatic systems was investigated to enhance physicochemical properties and potency profile of this class of inhibitors. The synthesis and biological activity of the derived compounds is discussed.
Related Topics
Physical Sciences and Engineering Chemistry Organic Chemistry
Authors
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