Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10596850 | Bioorganic & Medicinal Chemistry Letters | 2010 | 5 Pages |
Abstract
A new structural class of potent antagonists of the Neuropeptide S Receptor (NPSR) is reported. NPSR-PI1 demonstrates potent in vitro NPSR antagonism and central exposure in vivo.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
B. Wesley Trotter, Kausik K. Nanda, Peter J. Manley, Victor N. Uebele, Cindra L. Condra, Anthony L. Gotter, Karsten Menzel, Martin Henault, Rino Stocco, John J. Renger, George D. Hartman, Mark T. Bilodeau,