Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10596883 | Bioorganic & Medicinal Chemistry Letters | 2005 | 5 Pages |
Abstract
Considering importance of developing selective estrogen receptor modulators (SERMs), the present paper explores selectivity requirements of tetrahydroisoquinoline derivatives for binding with ERα versus ERβ receptors using E-state index and physicochemical parameters.
Keywords
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Subhendu Mukherjee, Achintya Saha, Kunal Roy,