Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
10596973 | Bioorganic & Medicinal Chemistry Letters | 2005 | 4 Pages |
Abstract
A series of 1,2,4-benzothiadiazine derivatives were synthesized and tested as selective ligands at α1-adrenergic and 5-HT1A receptor systems. Compound 1 has been characterized as a α1D-antagonist, while 6 as a 5-HT1A partial agonist.
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Authors
Annalisa Tait, Amedeo Luppi, Silvia Franchini, Elisa Preziosi, Carlo Parenti, Michela Buccioni, Gabriella Marucci, Amedeo Leonardi, Elena Poggesi, Livio Brasili,