| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1361980 | Bioorganic & Medicinal Chemistry Letters | 2011 | 5 Pages |
Abstract
The discovery of a novel series of 8-azabicyclo[3.2.1]octan-3-yl)-3-(4-chlorophenyl) propanamide antagonists of the vasopressin V1A receptor is disclosed. Compounds 47 and 48 were found to be high affinity, selective vasopressin V1A antagonists.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
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Authors
Susan Napier, Grant Wishart, William Arbuckle, James Baker, David Barn, Matilda Bingham, Angus Brown, Alan Byford, Chris Claxton, Mark Craighead, Kirsteen Buchanan, Lee Fielding, Lindsay Gibson, Richard Goodwin, Susan Goutcher, Nicholas Irving,