Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1365377 | Bioorganic & Medicinal Chemistry Letters | 2008 | 6 Pages |
Abstract
A series of imidazole derivatives have been designed and optimized for CXCR3 antagonism, pharmacokinetic properties, and reduced formation of glutathione conjugates.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Xiaohui Du, Xiaoqi Chen, Jeffrey T. Mihalic, Jeffrey Deignan, Jason Duquette, An-Rong Li, Bryan Lemon, Ji Ma, Shichang Miao, Karen Ebsworth, Timothy J. Sullivan, George Tonn, Tassie L. Collins, Julio C. Medina,