| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1369589 | Bioorganic & Medicinal Chemistry Letters | 2012 | 4 Pages |
Abstract
Four hinge-binding scaffolds have been explored for novel selective Aurora kinase inhibitors. The structure activity relationship, selectivity and pharmacokinetic profiles have been evaluated.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Zhiqin Ji, Yujia Dai, Cele Abad-Zapatero, Daniel H. Albert, Jennifer J. Bouska, Keith B. Glaser, Patrick A. Marcotte, Nirupama B. Soni, Terry J. Magoc, Kent D. Stewart, Ru-Qi Wei, Steve K. Davidsen, Michael R. Michaelides,