| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1373157 | Bioorganic & Medicinal Chemistry Letters | 2011 | 4 Pages |
Abstract
SAR studies of pyrrolo[1,2-f]triazines as JAK2 inhibitors is presented. Achieving JAK2 inhibition selectively over JAK3 is discussed.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
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Authors
Lalgudi S. Harikrishnan, Muthoni G. Kamau, Honghe Wan, Jennifer A. Inghrim, Kurt Zimmermann, Xiaopeng Sang, Harold A. Mastalerz, Walter L. Johnson, Guifen Zhang, Louis J. Lombardo, Michael A. Poss, George L. Trainor, John S. Tokarski, Matthew V. Lorenzi,