| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1373880 | Bioorganic & Medicinal Chemistry Letters | 2009 | 5 Pages |
Abstract
Two series of amino acid-derived heterocyclic progesterone receptor (PR) ligands are reported. Tetrazole-containing ligands behaved as potent PR partial agonists, while 1,2,4-triazole-containing ligands tended to act as PR full agonists in vitro.
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Authors
Marlys Hammond, Jaclyn R. Patterson, Sharada Manns, Tram H. Hoang, David G. Washburn, Walter Trizna, Lindsay Glace, Eugene T. Grygielko, Rakesh Nagilla, Melanie Nord, Harvey E. Fries, Douglas J. Minick, Nicholas J. Laping, Jeffrey D. Bray,