| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1374105 | Bioorganic & Medicinal Chemistry Letters | 2006 | 6 Pages |
Abstract
A group of tri and tetrasubstituted urea derivatives have been found to be hH3-antagonists. The most potent compounds were found in the class of (piperazine-1-yl)-(piperidine-1-yl)-methanones which in addition showed negligible hERG inhibition.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jesper F. Lau, Claus Bekker Jeppesen, Karin Rimvall, Rolf Hohlweg,