| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1374349 | Bioorganic & Medicinal Chemistry Letters | 2011 | 4 Pages |
Abstract
Amino-anthranilic acid derivatives have been identified as a new class of low serum shifted, high affinity full agonists of the human orphan G-protein-coupled receptor GPR109a with improved ADME properties.
Graphical abstractAmino-anthranilic acid derivatives have been identified as a new class of low serum shifted, high affinity full agonists of the human orphan G-protein-coupled receptor GPR109a with improved ADME properties.Figure optionsDownload full-size imageDownload as PowerPoint slide
Related Topics
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Authors
Jason E. Imbriglio, Daniel DiRocco, Rena Bodner, Subharekha Raghavan, Weichun Chen, Daria Marley, Craig Esser, Tom G. Holt, Michael S. Wolff, Andrew K.P. Taggart, M. Gerard Waters, James R. Tata, Steven L. Colletti,