| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1374390 | Bioorganic & Medicinal Chemistry Letters | 2006 | 4 Pages |
Abstract
A new class of high affinity hNK1R antagonists based on seven-membered ring cores has been identified. This series, with relatively simple, compact structures, includes compounds with high affinity, good selectivity, and promising in vivo properties.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Jason M. Elliott, Emma J. Carlson, Gary G. Chicchi, Olivier Dirat, Maria Dominguez, Ute Gerhard, Richard Jelley, A. Brian Jones, Marc M. Kurtz, Kwei lan Tsao, Alan Wheeldon,