| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1375287 | Bioorganic & Medicinal Chemistry Letters | 2009 | 5 Pages |
Abstract
A new class of inhibitors of HIV-1 integrase has been optimized to provide selective and highly efficient strand transfer inhibition.
Graphical abstractThe synthesis and SAR of a new class of HIV-1 integrase inhibitors is reported.Figure optionsDownload full-size imageDownload as PowerPoint slide
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
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Authors
Monica Donghi, Olaf D. Kinzel, Vincenzo Summa,