Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1375479 | Bioorganic & Medicinal Chemistry Letters | 2005 | 5 Pages |
Abstract
A series of ligands with varying heterocyclic cores and substituents that display a range of selectivity’s (up to >100x) for ER-β over ER-α are reported.
Graphical abstractA series of ligands with varying heterocyclic cores and substituents that display a range of selectivities (up to >100×) for ER-β over ER-α are reported.Figure optionsDownload full-size imageDownload as PowerPoint slide
Keywords
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Richard Chesworth, Matthew D. Wessel, Lisa Heyden, F. Michael Mangano, Michael Zawistoski, Laura Gegnas, David Galluzzo, Bruce Lefker, Kimberly O. Cameron, Jeanne Tickner, Bihong Lu, Tessa A. Castleberry, Donna N. Petersen, Amy Brault, Pia Perry,