Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1376482 | Bioorganic & Medicinal Chemistry Letters | 2006 | 5 Pages |
Abstract
Binding affinities for a range of epibatidine isomers and analogues at the α4β2 and α3β4 nAChR subtypes are reported; compounds having similar N–N distances to epibatidine show similar, high potencies.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Richard White, John R. Malpass, Sandeep Handa, S. Richard Baker, Lisa M. Broad, Liz Folly, Adrian Mogg,