Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1376981 | Bioorganic & Medicinal Chemistry Letters | 2006 | 6 Pages |
Abstract
3-Hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles were discovered as potent in vitro MEK1 inhibitors.
Graphical abstract3-Hydroxy-4-carboxyalkylamidino-5-arylamino-isothiazoles were discovered as potent in vitro MEK InhibitorsFigure optionsDownload full-size imageDownload as PowerPoint slide
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Chamakura V.N.S. Varaprasad, Dinesh Barawkar, Hassan El Abdellaoui, Subrata Chakravarty, Matthew Allan, Huanming Chen, Weijian Zhang, Jim Z. Wu, Robert Tam, Robert Hamatake, Stanley Lang, Zhi Hong,