| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1377312 | Bioorganic & Medicinal Chemistry Letters | 2008 | 5 Pages |
Abstract
The synthesis and the SAR of a new series of potent and selective dopamine D3 receptor antagonists is reported. The new scaffolds of the [g]-fused and the hetero-fused tricyclic benzazepine are here reported together with their pharmacokinetic profile.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
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Authors
Fabrizio Micheli, Giorgio Bonanomi, Simone Braggio, Anna Maria Capelli, Federica Damiani, Romano Di Fabio, Daniele Donati, Gabriella Gentile, Dieter Hamprecht, Ornella Perini, Marcella Petrone, Giovanna Tedesco, Silvia Terreni, Angela Worby,