Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1377342 | Bioorganic & Medicinal Chemistry Letters | 2008 | 5 Pages |
Abstract
To improve poor pharmacokinetic characters of the preceding VLA-4 inhibitors, novel piperazinylphenylalanine derivatives were designed and optimized for oral bioavailability.
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Osamu Saku, Kiminori Ohta, Eri Arai, Yuji Nomoto, Hiroko Miura, Hiroaki Nakamura, Eiichi Fuse, Yoshisuke Nakasato,