| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1377478 | Bioorganic & Medicinal Chemistry Letters | 2006 | 5 Pages |
Abstract
A novel series of tetracyclic indoles have been designed, synthesized and evaluated as androgen receptor (AR) ligands. Studies of structure–activity relationships (SARs) were investigated, which led to some compounds in this series as strong binders to androgen receptors.
Graphical abstractA novel series of tetracyclic indoles (I) have been designed, synthesized and evaluated as androgen receptor (AR) ligands. Studies of structure–activity relationships (SARs) were investigated, which led to some compounds in this series as strong binders to androgen receptors.Figure optionsDownload full-size imageDownload as PowerPoint slide
Related Topics
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Authors
Xuqing Zhang, Xiaojie Li, George F. Allan, Amy Musto, Scott G. Lundeen, Zhihua Sui,