| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1377577 | Bioorganic & Medicinal Chemistry Letters | 2007 | 4 Pages |
Abstract
The synthesis and structure–activity relationships against the C3a receptor of a series of substituted aminopiperidine derivatives are reported. DMPK properties and functional activities of selected compounds are described. The compounds obtained are the first non-arginine ligands of C3aR.
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Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Frédéric Denonne, Sophie Binet, Maggi Burton, Philippe Collart, Sabine Defays, Alan Dipesa, Maria Eckert, Alexander Giannaras, Seema Kumar, Beth Levine, Jean-Marie Nicolas, Patrick Pasau, Cécile Pégurier, Dorin Preda, Nathalie Van houtvin,