| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1377831 | Bioorganic & Medicinal Chemistry Letters | 2006 | 4 Pages |
Abstract
We report the synthesis of kinase targeted libraries based on the thienopyrazole scaffold. Several thienopyrazole analogs have been identified as submicromolar inhibitors of KDR.
Graphical abstractWe report the synthesis of kinase targeted libraries based on the thienopyrazole scaffold. Several thienopyrazole analogs have been identified as submicromolar inhibitors of KDR.Figure optionsDownload full-size imageDownload as PowerPoint slide
Keywords
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Irini Akritopoulou-Zanze, Daria Darczak, Kathy Sarris, Kathleen M. Phelan, Jeffrey R. Huth, Danying Song, Eric F. Johnson, Yong Jia, Stevan W. Djuric,