Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
5156230 | Bioorganic & Medicinal Chemistry Letters | 2017 | 7 Pages |
Keywords
CREBqPCRCSPsCBPATAD2BRPF1EP300cyclic-AMP response element binding proteinSTDDSFnuclear magnetic resonanceDMSOAlphaEpigeneticsHACX-ray crystallographyNMRSaturation transfer differenceDockingDimethyl sulfoxideNMR spectroscopyVirtual screeningDifferential scanning fluorimetryBromodomain inhibitorsCREB-binding proteinLigand efficiencyKac
Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Dimitrios Spiliotopoulos, Jian Zhu, Eike-Christian Wamhoff, Nicholas Deerain, Jean-Rémy Marchand, Jonas Aretz, Christoph Rademacher, Amedeo Caflisch,