| Article ID | Journal | Published Year | Pages | File Type |
|---|---|---|---|---|
| 1254905 | Chinese Chemical Letters | 2013 | 4 Pages |
Abstract
An efficient method for mono-phosphorylation of 2 (KRP203) using cbz-protection, dibenzylphosphoryl chloride and TMSI affording 2-P (KRP203-P) was developed. We applied the present method to the synthesis of KRP203 phosphate analogs which were difficult to produce through tradition procedures.
Graphical abstractA three-step procedure for the preparation of mono-phosphorylation of KRP203 to 2-P has been developed. This method was considered as an effective route to synthesize various analogs of 2-P.Figure optionsDownload full-size imageDownload as PowerPoint slide
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Physical Sciences and Engineering
Chemistry
Chemistry (General)
Authors
Xiao-Jian Wang, Jian-Guo Qi, Gang Li, Yu-Lin Tian, Da-Li Yin,