Article ID | Journal | Published Year | Pages | File Type |
---|---|---|---|---|
1376128 | Bioorganic & Medicinal Chemistry Letters | 2008 | 5 Pages |
Abstract
A novel series of potent zwitterionic uracil GnRH antagonists were discovered that showed reduced liability for CYP3A4 enzyme inhibition.
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Related Topics
Physical Sciences and Engineering
Chemistry
Organic Chemistry
Authors
Colin F. Regan, Zhiqiang Guo, Yongsheng Chen, Charles Q. Huang, Mi Chen, Wanlong Jiang, Jaimie K. Rueter, Timothy Coon, Chen Chen, John Saunders, Michael S. Brown, Steve F. Betz, R. Scott Struthers, Chun Yang, Jenny Wen, Ajay Madan, Yun-Fei Zhu,