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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Benzoic Acid and Chlorobenzoic Acids: Thermodynamic Study of the Pure Compounds and Binary Mixtures With Water
Fulltext Access 9 Pages 2016
Graphical contents list
Fulltext Access 9 Pages 2016
Design, synthesis and antiproliferative activity of novel 5-nitropyrimidine-2,4-diamine derivatives bearing alkyl acetate moiety
Fulltext Access 9 Pages 2016
Synthesis, characterization and in vitro evaluation of amphiphilic ion pairs of erythromycin and kanamycin antibiotics with liposaccharides
Fulltext Access 9 Pages 2016
Tyrosol and hydroxytyrosol derivatives as antitrypanosomal and antileishmanial agents
Fulltext Access 9 Pages 2016
Graphical contents list
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Polyvalent effect enhances diglycosidic antiplasmodial activity
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The Ikaros family of zinc-finger proteins
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Isoniazid metabolism and hepatotoxicity
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Impact of feed counterion addition and cyclone type on aerodynamic behavior of alginic-atenolol microparticles produced by spray drying
Fulltext Access 9 Pages 2016
Synthetic biology platform technologies for antimicrobial applications
Fulltext Access 9 Pages 2016
Prediction of the Adsorption of Diazepam by Activated Carbon in Aqueous Media
Fulltext Access 9 Pages 2016
Development of Suberin Fatty Acids and Chloramphenicol-Loaded Antimicrobial Electrospun Nanofibrous Mats Intended for Wound Therapy
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Design, synthesis, and structure-activity relationship study of glycyrrhetinic acid derivatives as potent and selective inhibitors against human carboxylesterase 2
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Population Pharmacokinetic-Toxicodynamic Modeling and Simulation of Cisplatin-Induced Acute Renal Injury in Rats: Effect of Dosing Rate on Nephrotoxicity
Fulltext Access 9 Pages 2016
Synergistic Skin Penetration Enhancer and Nanoemulsion Formulations Promote the Human Epidermal Permeation of Caffeine and Naproxen
Fulltext Access 9 Pages 2016
Intra-articular Administration of Chitosan Thermosensitive In Situ Hydrogels Combined With Diclofenac Sodium-Loaded Alginate Microspheres
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Spectroscopic-Based Chemometric Models for Quantifying Low Levels of Solid-State Transitions in Extended Release Theophylline Formulations
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Process and Formulation Effects on Protein Structure in Lyophilized Solids Using Mass Spectrometric Methods
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Quality by Design Approaches to Formulation Robustness-An Antibody Case Study
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Implications of In-Use Photostability: Proposed Guidance for Photostability Testing and Labeling to Support the Administration of Photosensitive Pharmaceutical Products, Part 3. Oral Drug Products
Fulltext Access 9 Pages 2016
Mouse Models for Assessing Protein Immunogenicity: Lessons and Challenges
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Protolytic Equilibria of Sartans in Micellar Solutions of Differently Charged Surfactants
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A Simplified Model of Moisture Transport in Hydrophilic Porous Media With Applications to Pharmaceutical Tablets
Fulltext Access 9 Pages 2016
A Micro-Polyethylene Glycol Precipitation Assay as a Relative Solubility Screening Tool for Monoclonal Antibody Design and Formulation Development
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Rapid Conformational Analysis of Protein Drugs in Formulation by Hydrogen/Deuterium Exchange Mass Spectrometry
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Epilepsy coexisting with depression
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Synthesis and bioactivity of novel triazole incorporated benzothiazinone derivatives as antitubercular and antioxidant agent
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Synthesis, biological evaluation and structure-activity relationship of 2-styrylquinazolones as anti-tubercular agents
Fulltext Access 9 Pages 2016
Design, synthesis and biological evaluation of pyrazolylaminoquinazoline derivatives as highly potent pan-fibroblast growth factor receptor inhibitors
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Isolation, analytical measurements, and cell line studies of the iron-bryostatin-1 complex
Fulltext Access 9 Pages 2016
Strigolactone derivatives for potential crop enhancement applications
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Solution and Solid State Nuclear Magnetic Resonance Spectroscopic Characterization of Efavirenz
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Physiologically Based Pharmacokinetic Modeling for Substitutability Analysis of Venlafaxine Hydrochloride Extended-Release Formulations Using Different Release Mechanisms: Osmotic Pump Versus Openable Matrix
Fulltext Access 9 Pages 2016
The Use of Binary Polymeric Networks in Stabilizing Polyethylene Oxide Solid Dispersions
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Novel Displacement Agents for Aqueous 2-Phase Extraction Can Be Estimated Based on Hybrid Shortcut Calculations
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Studying the Propensity of Compounds to Supersaturate: A Practical and Broadly Applicable Approach
Fulltext Access 9 Pages 2016
Non-Ablative Fractional Laser to Facilitate Transdermal Delivery
Fulltext Access 9 Pages 2016
Characterizing Reversible Protein Association at Moderately High Concentration Via Composition-Gradient Static Light Scattering
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A Nanoscale Polymeric Penetration Enhancer Based on Polylysine for Topical Delivery of Proteins and Peptides
Fulltext Access 9 Pages 2016
The Crystal Structure and Behavior of Fenamic Acid-Acridine Complex Under High Pressure
Fulltext Access 9 Pages 2016
Simple spectrophotometric methods for the simultaneous determination of antipyrine and benzocaine
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Cryptic prophages as targets for drug development
Fulltext Access 9 Pages 2016
Investigating how the attributes of self-associated drug complexes influence the passive transport of molecules through biological membranes
Fulltext Access 9 Pages 2016
Synthesis and evaluation of novel lipopeptide as a vehicle for efficient gene delivery and gene silencing
Fulltext Access 9 Pages 2016
Hydrogel-forming microneedle arrays: Potential for use in minimally-invasive lithium monitoring
Fulltext Access 9 Pages 2016
Lidocaine self-sacrificially improves the skin permeation of the acidic and poorly water-soluble drug etodolac via its transformation into an ionic liquid
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Application of Hansen Solubility Parameters to predict drug-nail interactions, which can assist the design of nail medicines
Fulltext Access 9 Pages 2016
Development and characterization of novel 1-(1-Naphthyl)piperazine-loaded lipid vesicles for prevention of UV-induced skin inflammation
Fulltext Access 9 Pages 2016
The solubility-permeability interplay and oral drug formulation design: Two heads are better than one
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Tumor microenvironment for cancer stem cells
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Protective effect of mesoporous silica particles on encapsulated folates
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Investigating the effect of processing parameters on pharmaceutical tablet disintegration using a real-time particle imaging approach
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Estimation of design space for an extrusion–spheronization process using response surface methodology and artificial neural network modelling
Fulltext Access 9 Pages 2016
The combined effect of wet granulation process parameters and dried granule moisture content on tablet quality attributes
Fulltext Access 9 Pages 2016
Asymmetric distribution in twin screw granulation
Fulltext Access 9 Pages 2016
Development of a pharmaceutical cocrystal with solution crystallization technology: Preparation, characterization, and evaluation of myricetin-proline cocrystals
Fulltext Access 9 Pages 2016
A novel solubilization technique for poorly soluble drugs through the integration of nanocrystal and cocrystal technologies
Fulltext Access 9 Pages 2016
Unsaturated fatty acids lactose esters: cytotoxicity, permeability enhancement and antimicrobial activity
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Spheronization mechanism of pharmaceutical material crystals processed by extremely high shearing force using a mechanical powder processor
Fulltext Access 9 Pages 2016
Tissue engineering the cardiac microenvironment: Multicellular microphysiological systems for drug screening
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Hydrogels for therapeutic cardiovascular angiogenesis
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Bioengineering Hematopoietic Stem Cell Niche toward Regenerative Medicine
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Properties and mechanisms of drug release from matrix tablets containing poly(ethylene oxide) and poly(acrylic acid) as release retardants
Fulltext Access 9 Pages 2016
Treatment with high dose of atorvastatin reduces vascular injury in diabetic rats
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Cytoprotective mechanism of action of curcumin against cataract
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Method of hyperthermia and tumor size influence effectiveness of doxorubicin release from thermosensitive liposomes in experimental tumors
Fulltext Access 9 Pages 2016
Doxorubicin/gold-loaded core/shell nanoparticles for combination therapy to treat cancer through the enhanced tumor targeting
Fulltext Access 9 Pages 2016
Glucose and magnetic-responsive approach toward in situ nitric oxide bubbles controlled generation for hyperglycemia theranostics
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Synthesis and biological evaluation of salicylic acid conjugated isoxazoline analogues on immune cell proliferation and angiogenesis
Fulltext Access 9 Pages 2016
Protective effects of kaempferol against reactive oxygen species-induced hemolysis and its antiproliferative activity on human cancer cells
Fulltext Access 9 Pages 2016
Graphical contents list
Fulltext Access 9 Pages 2016
Synthesis and antimicrobial activity of styryl/pyrrolyl/pyrazolyl sulfonylmethyl-1,3,4-oxadiazolyl amines and styryl/pyrrolyl/pyrazolyl sulfonylmethyl-1,3,4-thiadiazolyl amines
Fulltext Access 9 Pages 2016
Synthesis, anti-cancer evaluation of benzenesulfonamide derivatives as potent tubulin-targeting agents
Fulltext Access 9 Pages 2016
Synthesis and biological evaluation of new naphthalene substituted thiosemicarbazone derivatives as potent antifungal and anticancer agents
Fulltext Access 9 Pages 2016
Effects of ramp-up of inspired airflow on in vitro aerosol dose delivery performance for certain dry powder inhalers
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Hepatic Clearance Prediction of Nine Human Immunodeficiency Virus Protease Inhibitors in Rat
Fulltext Access 9 Pages 2016
Development of a Novel Lung Slice Methodology for Profiling of Inhaled Compounds
Fulltext Access 9 Pages 2016
Mechanism of Decarboxylation of Pyruvic Acid in the Presence of Hydrogen Peroxide
Fulltext Access 9 Pages 2016
The Effect of Capsaicin Derivatives on Tight-Junction Integrity and Permeability of Madin-Darby Canine Kidney Cells
Fulltext Access 9 Pages 2016
Quality and Batch-to-Batch Consistency of Original and Biosimilar Epoetin Products
Fulltext Access 9 Pages 2016
Development of a Support Vector Machine-Based System to Predict Whether a Compound Is a Substrate of a Given Drug Transporter Using Its Chemical Structure
Fulltext Access 9 Pages 2016
Pharmacokinetic Modeling to Simulate the Concentration-Time Profiles After Dermal Application of Rivastigmine Patch
Fulltext Access 9 Pages 2016
Three-Dimensional Printing of Carbamazepine Sustained-Release Scaffold
Fulltext Access 9 Pages 2016
Co-administration of morphine and gabapentin leads to dose dependent synergistic effects in a rat model of postoperative pain
Fulltext Access 9 Pages 2016
Nanonized itraconazole powders for extemporary oral suspensions: Role of formulation components studied by a mixture design
Fulltext Access 9 Pages 2016
Effect of pirfenidone delivered using layer-by-layer thin film on excisional wound healing
Fulltext Access 9 Pages 2016
Fundamental understanding of drug absorption from a parenteral oil depot
Fulltext Access 9 Pages 2016
Synthesis, characterization and biological evaluation of benzothiazoles and tetrahydrobenzothiazoles bearing urea or thiourea moieties as vasorelaxants and inhibitors of the insulin releasing process
Fulltext Access 9 Pages 2016
Chitosan-pectin hybrid nanoparticles prepared by coating and blending techniques
Fulltext Access 9 Pages 2016
Synthesis and characterization of a novel radioiodinated phenylacetamide and its homolog as theranostic agents for malignant melanoma
Fulltext Access 9 Pages 2016
Olanzapine modulation of hepatic oxidative stress and inflammation in socially isolated rats
Fulltext Access 9 Pages 2016
The molecular assembly of the ionic liquid/aliphatic carboxylic acid/aliphatic amine as effective and safety transdermal permeation enhancers
Fulltext Access 9 Pages 2016
Uptake of free, calcium-bound and liposomal encapsulated nitrogen containing bisphosphonates by breast cancer cells
Fulltext Access 9 Pages 2016
Co-spray dried resveratrol and budesonide inhalation formulation for reducing inflammation and oxidative stress in rat alveolar macrophages
Fulltext Access 9 Pages 2016
A supersaturating delivery system of silibinin exhibiting high payload achieved by amorphous nano-complexation with chitosan
Fulltext Access 9 Pages 2016
Real-time monitoring of cocrystallization processes by solvent evaporation: A near infrared study
Fulltext Access 9 Pages 2016
Black seed oil ameliorated scopolamine-induced memory dysfunction and cortico-hippocampal neural alterations in male Wistar rats
Fulltext Access 9 Pages 2016
Visualization of drug translocation in the nasal cavity and pharmacokinetic analysis on nasal drug absorption using positron emission tomography in the rat
Fulltext Access 9 Pages 2016
Prolonged anti-bacterial activity of ion-complexed doxycycline for the treatment of osteomyelitis
Fulltext Access 9 Pages 2016
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