[186Re]Liposomal doxorubicin (Doxil): in vitro stability, pharmacokinetics, imaging and biodistribution in a head and neck squamous cell carcinoma xenograft model Fulltext Access 10 Pages 2009
The remodeling of connexin in the hypertrophied right ventricular in pulmonary arterial hypertension and the effect of a dual ET receptor antagonist (bosentan) Fulltext Access 10 Pages 2009
Histological expression of angiogenic factors: VEGF, PDGFRα, and HIF-1α in Hodgkin lymphoma Fulltext Access 10 Pages 2009
The challenge of apocrine proliferations of the breast: A morphologic approach Fulltext Access 10 Pages 2009
Biopsies of colorectal clinical polyps – emergence of diagnostic information on deeper levels Fulltext Access 10 Pages 2009
Hepatocyte growth factor suppresses tumor cell apoptosis in nasopharyngeal carcinoma by upregulating Bcl-2 protein expression Fulltext Access 10 Pages 2009
Expression of xenobiotic and steroid hormone metabolizing enzymes in hepatocellular tumors of the non-cirrhotic liver Fulltext Access 10 Pages 2009
[18F]Fallypride dopamine D2 receptor studies using delayed microPET scans and a modified Logan plot Fulltext Access 10 Pages 2009
Tumor targeting and SPECT imaging properties of an 111In-labeled galectin-3 binding peptide in prostate carcinoma Fulltext Access 10 Pages 2009
18F-Labeled benzylideneaniline derivatives as new ligands for β-amyloid plaque imaging in Alzheimer's disease Fulltext Access 10 Pages 2009
Vitamin C enters mouse T cells as dehydroascorbic acid in vitro and does not recapitulate in vivo vitamin C effects Fulltext Access 10 Pages 2009
Cu(II) bis(thiosemicarbazone) radiopharmaceutical binding to serum albumin: further definition of species dependence and associated substituent effects Fulltext Access 10 Pages 2009
Evaluation of an anti-p185HER2 (scFv-CH2-CH3)2 fragment following radioiodination using two different residualizing labels: SGMIB and IB-Mal-d-GEEEK Fulltext Access 10 Pages 2009
Synthesis, radiolabeling, in vitro and in vivo evaluation of [18F]-FPECMO as a positron emission tomography radioligand for imaging the metabotropic glutamate receptor subtype 5 Fulltext Access 10 Pages 2009
Radiolabeled annexin V for imaging apoptosis in radiated human follicular thyroid carcinomas — is an individualized protocol necessary? Fulltext Access 10 Pages 2009
Mono and bis-6-arylbenzimidazo[1,2-c]quinazolines: A new class of antimicrobial agents Fulltext Access 10 Pages 2009
Total synthesis and anticancer activity of highly potent novel glycolipid derivatives Fulltext Access 10 Pages 2009
Conformationally constrained analogues of N′-(4-tert-butylbenzyl)-N-(4-methylsulfonylaminobenzyl)thiourea as TRPV1 antagonists Fulltext Access 10 Pages 2009
Molecular modeling and inhibition of phospholipase A2 by polyhydroxy phenolic compounds Fulltext Access 10 Pages 2009
Quantitative structure–activity relationship (QSAR) of aryl alkenyl amides/imines for bacterial efflux pump inhibitors Fulltext Access 10 Pages 2009
Prediction of CCR5 receptor binding affinity of substituted 1-(3,3-diphenylpropyl)-piperidinyl amides and ureas based on the heuristic method, support vector machine and projection pursuit regression Fulltext Access 10 Pages 2009
Ablation of Stat3 by siRNA Alters Gene Expression Profiles in JEG-3 Cells: A Systems Biology Approach Fulltext Access 10 Pages 2009
Cutaneous distribution of plasmacytoid dendritic cells in lupus erythematosus. Selective tropism at the site of epithelial apoptotic damage Fulltext Access 10 Pages 2009
Rheological and Physiological Consequences of Conversion of the Maternal Spiral Arteries for Uteroplacental Blood Flow during Human Pregnancy Fulltext Access 10 Pages 2009
IGF-dependent and IGF-independent actions of IGF-binding protein-1 and -2: implications for metabolic homeostasis Fulltext Access 10 Pages 2009
Leptin Acts via Leptin Receptor-Expressing Lateral Hypothalamic Neurons to Modulate the Mesolimbic Dopamine System and Suppress Feeding Fulltext Access 10 Pages 2009
Ablation of Neutral Cholesterol Ester Hydrolase 1 Accelerates Atherosclerosis Fulltext Access 10 Pages 2009
Novel Soluble Flt-1 Isoforms in Plasma and Cultured Placental Explants from Normotensive Pregnant and Preeclamptic Women Fulltext Access 10 Pages 2009
Altered Global Gene Expression in First Trimester Placentas of Women Destined to Develop Preeclampsia Fulltext Access 10 Pages 2009
Differential Placental Hormone Gene Expression during Pregnancy in a Transgenic Mouse Containing the Human Growth Hormone/Chorionic Somatomammotropin Locus Fulltext Access 10 Pages 2009
Regioselective synthesis of dispiro[1H-indene-2,3′-pyrrolidine-2′,3″-[3H]indole]-1,2″(1″H)-diones of potential anti-tumor properties Fulltext Access 10 Pages 2009
The Isolation and Characterization of a Novel Telomerase Immortalized First Trimester Trophoblast Cell Line, Swan 71 Fulltext Access 10 Pages 2009
The proprotein convertase furin in human trophoblast: Possible role in promoting trophoblast cell migration and invasion Fulltext Access 10 Pages 2009
Identification of critical antibody-binding sites in the HIV-1 gp41 six-helix bundle core as potential targets for HIV-1 fusion inhibitors Fulltext Access 10 Pages 2009
The pharmacodynamic effect of sirolimus: Individual variation of cytokine mRNA expression profiles in human whole blood samples Fulltext Access 10 Pages 2009
The variation in cytoplasmic distribution of mouse peritoneal macrophage during phagocytosis modulated by mangiferin, an immunomodulator Fulltext Access 10 Pages 2009
Antitumor efficacy induced by human ovarian cancer cells secreting IL-21 alone or combination with GM-CSF cytokines in nude mice model Fulltext Access 10 Pages 2009
Free intracellular Ca2+ regulates bacterial lipopolysaccharide induction of iNOS in human macrophages Fulltext Access 10 Pages 2009
Delayed recruitment of lymphocytes into the lungs of CD30-deficient mice during aerogenic Mycobacterium avium infections Fulltext Access 10 Pages 2009
Zymosan treatment of mouse mast cells enhances dectin-1 expression and induces dectin-1-dependent reactive oxygen species (ROS) generation Fulltext Access 10 Pages 2009
Synthesis and in vitro trichomonicidal, giardicidal and amebicidal activity of N-acetamide(sulfonamide)-2-methyl-4-nitro-1H-imidazoles Fulltext Access 10 Pages 2009
Cyclocondensation reaction of heterocyclic carbonyl compounds, Part XIII: Synthesis and cytotoxic activity of some 3,7-diaryl-5-(3,4,5-trimethoxyphenyl)pyrazolo[4,3-e][1,2,4]triazines Fulltext Access 10 Pages 2009
Design, synthesis and pharmacological evaluation of new 1-[3-(4-arylpiperazin-1-yl)-2-hydroxy-propyl]-3,3-diphenylpyrrolidin-2-one derivatives with antiarrhythmic, antihypertensive, and α-adrenolytic activity Fulltext Access 10 Pages 2009
Facile synthesis and in vitro properties of 1-alkyl- and 1-alkyl-N-propargyl-1,2,3,4-tetrahydroisoquinoline derivatives on PC12 cells Fulltext Access 10 Pages 2009
Preparation and antitubercular activities in vitro and in vivo of novel Schiff bases of isoniazid Fulltext Access 10 Pages 2009
S- and C-nucleosidoquinazoline as new nucleoside analogs with potential analgesic and anti-inflammatory activity Fulltext Access 10 Pages 2009
Physicochemical properties and membrane interactions of anti-apoptotic derivatives 2-(4-fluorophenyl)-3-(pyridin-4-yl)imidazo[1,2-a]pyridine depending on the hydroxyalkylamino side chain length and conformation: An NMR and ESR study Fulltext Access 10 Pages 2009
Discovering a new analogue of thalidomide which may be used as a potent modulator of TNF-α production Fulltext Access 10 Pages 2009
Synthesis and anticonvulsant activity of new N-[(4-arylpiperazin-1-yl)-alkyl] derivatives of 3-phenyl-pyrrolidine-2,5-dione Fulltext Access 10 Pages 2009
Synthesis of glycose carbamides and evaluation of the induction of erythroid differentiation of human erythroleukemic K562 cells Fulltext Access 10 Pages 2009
Synthesis and in vitro anticancer activity of 2,4-azolidinedione-acetic acids derivatives Fulltext Access 10 Pages 2009
Synthesis and antitumor activity of novel dithiocarbamate substituted chromones Fulltext Access 10 Pages 2009
Discovery of a new family of bis-8-hydroxyquinoline substituted benzylamines with pro-apoptotic activity in cancer cells: Synthesis, structure–activity relationship, and action mechanism studies Fulltext Access 10 Pages 2009
Comparative chemometric modeling of cytochrome 3A4 inhibitory activity of structurally diverse compounds using stepwise MLR, FA-MLR, PLS, GFA, G/PLS and ANN techniques Fulltext Access 10 Pages 2009
Novel derivatives of 6-mercaptopurine: Synthesis, characterization and antiproliferative activities of S-allylthio-mercaptopurines Fulltext Access 10 Pages 2009
Synthesis and anticancer activity of N-bis(trifluoromethyl)alkyl-N′-thiazolyl and N-bis(trifluoromethyl)alkyl-N′-benzothiazolyl ureas Fulltext Access 10 Pages 2009
Design, cytotoxic and fluorescent properties of novel N-phosphorylalkyl substituted E,E-3,5-bis(arylidene)piperid-4-ones Fulltext Access 10 Pages 2009
Synthesis, biological evaluation and molecular modeling of oxoisoaporphine and oxoaporphine derivatives as new dual inhibitors of acetylcholinesterase/butyrylcholinesterase Fulltext Access 10 Pages 2009
Large ring 1,3-bridged 2-azetidinones: Experimental and theoretical studies Fulltext Access 10 Pages 2009
Studies on chemical structure modification and biology of a natural product, Gambogic acid (I): Synthesis and biological evaluation of oxidized analogues of gambogic acid Fulltext Access 10 Pages 2009
New acyclic nucleosides analogues as potential analgesic, anti-inflammatory, anti-oxidant and anti-microbial derived from pyrimido[4,5-b]quinolines Fulltext Access 10 Pages 2009
Modeling the activity of furin inhibitors using artificial neural network Fulltext Access 10 Pages 2009
Crystal structures, antioxidation and DNA binding properties of Dy(III) complexes with Schiff-base ligands derived from 8-hydroxyquinoline-2-carboxaldehyde and four aroylhydrazines Fulltext Access 10 Pages 2009
Design, synthesis and biological evaluation of novel fluorinated docetaxel analogues Fulltext Access 10 Pages 2009
Synthesis, biological evaluation and 2D-QSAR analysis of benzoxazoles as antimicrobial agents Fulltext Access 10 Pages 2009
Application of desirability-based multi(bi)-objective optimization in the design of selective arylpiperazine derivates for the 5-HT1A serotonin receptor Fulltext Access 10 Pages 2009
Synthesis, pharmacological and antiviral activity of 1,3-thiazepine derivatives Fulltext Access 10 Pages 2009
Synthesis and in vitro antitumor activities of novel 4-anilinoquinazoline derivatives Fulltext Access 10 Pages 2009
Synthesis, antiarrhythmic and anticoagulant activities of novel thiazolo derivatives from methyl 2-(thiazol-2-ylcarbamoyl)acetate Fulltext Access 11 Pages 2009
Design, synthesis and evaluation of novel uracil acetamide derivatives as potential inhibitors of Plasmodium falciparum dUTP nucleotidohydrolase Fulltext Access 11 Pages 2009
Synthesis of 2-styrylchromones as a novel class of antiproliferative agents targeting carcinoma cells Fulltext Access 11 Pages 2009
Discovery of novel acetanilide derivatives as potent and selective β3-adrenergic receptor agonists Fulltext Access 11 Pages 2009
Synthesis and characterization of dinuclear macrocyclic cobalt(II), copper(II) and zinc(II) complexes derived from 2,2,2′,2′-S,S[bis(bis-N,N-2-thiobenzimidazolyloxalato-1,2-ethane)]: DNA binding and cleavage studies Fulltext Access 11 Pages 2009
Phenethyl pyridines with non-polar internal substitutents as selective ligands for estrogen receptor beta Fulltext Access 11 Pages 2009
Primaquine dipeptide derivatives bearing an imidazolidin-4-one moiety at the N-terminus as potential antimalarial prodrugs Fulltext Access 11 Pages 2009
Synthesis and evaluation of some novel isochroman carboxylic acid derivatives as potential anti-diabetic agents Fulltext Access 11 Pages 2009
Design, synthesis and AChE inhibitory activity of indanone and aurone derivatives Fulltext Access 11 Pages 2009
Fragment and knowledge-based design of selective GSK-3β inhibitors using virtual screening models Fulltext Access 11 Pages 2009
Synthesis and activity of fibrillogenesis peptide inhibitors related to the 17–21 β-amyloid sequence Fulltext Access 11 Pages 2009
Substituted quinolinyl chalcones and quinolinyl pyrimidines as a new class of anti-infective agents Fulltext Access 11 Pages 2009
Hansch analysis of substituted benzoic acid benzylidene/furan-2-yl-methylene hydrazides as antimicrobial agents Fulltext Access 11 Pages 2009
Synthesis, HIV-RT inhibitory activity and SAR of 1-benzyl-1H-1,2,3-triazole derivatives of carbohydrates Fulltext Access 11 Pages 2009
Tetrahydronaphthyl azole oxime ethers: The conformationally rigid analogues of oxiconazole as antibacterials Fulltext Access 11 Pages 2009
Anti-trypanosomatid benzofuroxans and deoxygenated analogues: Synthesis using polymer-supported triphenylphosphine, biological evaluation and mechanism of action studies Fulltext Access 11 Pages 2009
New derivatives of 3,5-substituted-1,4,2-dioxazoles: Synthesis and activity against Entamoeba histolytica Fulltext Access 11 Pages 2009
Design and in silico screening of combinatorial library of antimalarial analogs of triclosan inhibiting Plasmodium falciparum enoyl-acyl carrier protein reductase Fulltext Access 11 Pages 2009
Synthesis and evaluation of pyrido[1,2-a]pyrimidines as inhibitors of nitric oxide synthases Fulltext Access 11 Pages 2009
Synthesis and evaluation of a novel series of heterocyclic oleanolic acid derivatives with anti-osteoclast formation activity Fulltext Access 11 Pages 2009
Novel CYP17 inhibitors: Synthesis, biological evaluation, structure–activity relationships and modelling of methoxy- and hydroxy-substituted methyleneimidazolyl biphenyls Fulltext Access 11 Pages 2009
Identification of putative steroid-binding sites in human ABCB1 and ABCG2 Fulltext Access 11 Pages 2009
Synthesis and antibacterial activity of novel 15-membered macrolide derivatives: 4â³-Carbamate, 11,12-cyclic carbonate-4â³-carbamate and 11,4â³-di-O-arylcarbamoyl analogs of azithromycin Fulltext Access 11 Pages 2009
Novel modified steroid derivatives of androstanolone as chemotherapeutic anti-cancer agents Fulltext Access 11 Pages 2009