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Daneshyari Pharmacology Journas Latest Articles

Pharmacology Research Articles

Pharmacokinetics of Oltipraz in Mutant Nagase Analbuminemic Rats
Fulltext Access 8 Pages 2006
Serotonin 2A receptor antagonist treatment reduces dopamine D1 receptor-mediated rotational behavior but not l-DOPA-induced abnormal involuntary movements in the unilateral dopamine-depleted rat
Fulltext Access 8 Pages 2006
meso-Dihydroguaiaretic acid attenuates the neurotoxic effect of staurosporine in primary rat cortical cultures
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Enhancement of the analgesic activity of paracetamol and nitroparacetamol by the oral administration of all-trans retinoic acid
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Retigabine-induced population primary afferent hyperpolarisation in vitro
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Identification of residues critical for Cu2+-mediated inhibition of glycine α1 receptors
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Cyclosporin A inhibits apolipoprotein A-I-induced early events in cellular cholesterol homeostasis in rat astrocytes
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Molecular mechanisms mediating gastrin-releasing peptide receptor modulation of memory consolidation in the hippocampus
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The enantiomer of progesterone acts as a molecular neuroprotectant after traumatic brain injury
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Presynaptic inhibition by kainate receptors converges mechanistically with presynaptic inhibition by adenosine and GABAB receptors
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Distinct endocrine effects of chronic haloperidol or risperidone administration in male rats
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Preliminary Evaluation of Polymer-Based Drug Composite Microparticle Production by Coacervate Desolvation with Supercritical Carbon Dioxide
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2-Aminoethoxydiphenyl borate (2-APB) stimulates a conformationally coupled calcium release pathway in the NG115-401L neuronal cell line
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Biowaiver Monographs for Immediate Release Solid Oral Dosage Forms: Amitriptyline Hydrochloride*
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Therapeutic utility of a novel tight junction modulating peptide for enhancing intranasal drug delivery
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In Vivo use of the P450 inactivator 1-aminobenzotriazole in the rat: Varied dosing route to elucidate gut and liver contributions to first-pass and systemic clearance
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Investigation of the absorption mechanisms of baicalin and baicalein in rats
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Transport of levovirin prodrugs in the human intestinal Caco-2 cell line
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Bioavailability and in Vivo Release Behavior of Controlled-Release Multiple-Unit Theophylline Dosage Forms in Beagle Dogs, Cynomolgus Monkeys, and Göttingen Minipigs
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Thermodynamic modeling of activity coefficient and prediction of solubility: Part 1 predictive models
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Towards characterization and identification of solid state pharmaceutical mixtures through second harmonic generation
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A process analytical technology approach based on near infrared spectroscopy: Tablet hardness, content uniformity, and dissolution test measurements of intact tablets
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High throughput solubility measurement with automated polarized light microscopy analysis
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Effects of Deaeration Methods on Dissolution Testing in Aqueous Media: A Study Using a Total Dissolved Gas Pressure Meter*
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Endocannabinoids at the spinal level regulate, but do not mediate, nonopioid stress-induced analgesia
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Accessibility to residues in transmembrane segment four of the glycine receptor
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Enhanced nicotinic acetylcholine receptor-mediated [3H]norepinephrine release from neonatal rat hypothalamus
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The locus coeruleus nucleus as a site of action of the antinociceptive and behavioral effects of the nicotinic receptor agonist, epibatidine
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Injection of l-glutamate into medial prefrontal cortex induces cardiovascular responses through NMDA receptor – nitric oxide in rat
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In vivo effect of tramadol on locus coeruleus neurons is mediated by α2-adrenoceptors and modulated by serotonin
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Selective changes in thalamic and cortical GABAA receptor subunits in a model of acquired absence epilepsy in the rat
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3-Hydroxypyridazine 1-oxides as carboxylate bioisosteres: A new series of subtype-selective AMPA receptor agonists
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Effects of chronic nicotine administration and its withdrawal on striatal FosB/ΔFosB and c-Fos expression in rats and mice
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Mu opioid receptor-dependent and independent components in effects of tramadol
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Analgesic effects of mGlu1 and mGlu5 receptor antagonists in the rat formalin test
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Orexin A affects ascending contraction depending on downstream cholinergic neurons and descending relaxation through independent pathways in mouse jejunum
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Enhancing exposure of protein therapeutics
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The N-terminus of the norepinephrine transporter regulates the magnitude and selectivity of the transporter-associated leak current
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Blockade of intracellular calcium release induces an antidepressant-like effect in the mouse forced swimming test
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In vitro and ex vivo distribution of [3H]harmane, an endogenous β-carboline, in rat brain
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An NMDA receptor-dependent hydroxyl radical pathway in the rabbit hypothalamus may mediate lipopolysaccharide fever
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Effects of histamine H3 antagonists and donepezil on learning and mnemonic deficits induced by pentylenetetrazol kindling in weanling mice
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Adenylyl cyclase type II activity is regulated by two different mechanisms: Implications for acute and chronic opioid exposure
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l-3,4-Dihydroxyphenylalanine-induced c-Fos expression in the CNS under inhibition of central aromatic l-amino acid decarboxylase
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The GABAB receptor allosteric modulator CGP7930, like baclofen, reduces operant self-administration of ethanol in alcohol-preferring rats
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The acetylcholinesterase inhibitor, Donepezil, regulates a Th2 bias in Alzheimer's disease patients
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Regional and cellular distribution of CYP2E1 in monkey brain and its induction by chronic nicotine
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Anti-inflammatory properties of cholinergic up-regulation: A new role for acetylcholinesterase inhibitors
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Chemokines and chemokine receptors: Large and small therapeutic strategies for inflammatory diseases
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Injectable formulation of disodium 1-[2-(carboxylato)pyrrolidin-1-yl]diazen-1-ium-1,2-diolate (PROLI/NO), an ultrafast nitric oxide donor prodrug
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A rabbit model for sublingual drug delivery: Comparison with human pharmacokinetic studies of propranolol, verapamil and captopril
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Different effects of ATP on the contractile activity of mice diaphragmatic and skeletal muscles
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Differential activation of protein kinase C isoforms following chemical ischemia in rat cerebral cortex slices
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Hypobaric hypoxia induces oxidative stress in rat brain
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Epigenetic modulation of the developing serotonergic neurotransmission in the semi-precocial rodent Octodon degus
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Antimicrobial peptides in skin disease
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Why do we not have a vaccine against congenital cytomegalovirus (CMV) infection?
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Can efflux inhibitors really counter resistance?
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Tigecycline: First class glycylcycline: a new choice for empiric therapy
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Meningococcal diseases: From genomes to vaccines
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Anti-inflammatory strategies for the treatment of multiple sclerosis – tryptophan catabolites may hold the key
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Quantitative determination of amorphous cyclosporine in crystalline cyclosporine samples by Fourier transform infrared spectroscopy
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Antibody treatment of ulcerative colitis
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Employment of microRNA profiles and RNA interference and antagomirs for the characterization and treatment of respiratory disease
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Toll-like receptors and airway disease
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Tumour necrosis factor-α as a therapeutic target in asthma
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Interactions between long-acting β2-agonists and glucocorticoids
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Emerging pharmacotherapeutic strategies for the treatment of ischemic stroke
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Targeting melanocortin receptors for the treatment of obesity
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Benzodiazepine receptor agonists and insomnia: Is subtype selectivity lost in translation?
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Enhancing AMPA to NMDA throughput as a convergent mechanism for antidepressant action
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Development of functionally selective agonists as novel therapeutic agents
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Novel biomarker platforms in toxicology
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Miniaturization: Chip-based liquid chromatography and proteomics
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Target ability and therapy efficacy of immunoliposomes using a humanized antihepatoma disulfide-stabilized Fv fragment on tumor cells
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In Situ Measurement of Solvent-Mediated Phase Transformations During Dissolution Testing
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Effects of Cyclodextrins on Chemically and Thermally Induced Unfolding and Aggregation of Lysozyme and Basic Fibroblast Growth Factor
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Degradation Rate of Lyophilized Insulin, Exhibiting an Apparent Arrhenius Behavior around Glass Transition Temperature Regardless of Significant Contribution of Molecular Mobility
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Contribution of lysosomes to concentrative uptake of DX-9065a into rat liver
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Permeation of 4-Cyanophenol and Methyl Paraben from Powder and Saturated Aqueous Solution through Silicone Rubber Membranes and Human Skin
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Pharmacokinetics and Hepatic Extraction of Recombinant Human Parathyroid Hormone, hPTH (1-34), in Rat, Dog, and Monkey
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Gastrointestinal transit and mucoadhesive characteristics of complexation hydrogels in rats
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Acid decomposition of omeprazole in the absence of thiol: A differential pulse polarographic study at the static mercury drop electrode (SMDE)
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Molecular mobility of nifedipine−PVP and phenobarbital−PVP solid dispersions as measured by 13C-NMR spin-lattice relaxation time
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Biorelevant dissolution media: Aggregation of amphiphiles and solubility of estradiol
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The Effects of Surface Lactone Hydrolysis and Temperature on the Specific and Nonspecific Interactions Between Phenobarbital and Activated Carbon Surfaces
Fulltext Access 9 Pages 2006
Investigation of Solid-State NMR Line Widths of Ibuprofen in Drug Formulations
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Prediction of Tablet Hardness Based on Near Infrared Spectra of Raw Mixed Powders by Chemometrics
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Deep Percutaneous Penetration into Muscles and Joints
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Bile Acid Salt Binding with Colesevelam HCl is Not Affected by Suspension in Common Beverages
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Transcellular route of diffusion through stratum corneum: Results from finite element models
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Tetrazole compounds: The effect of structure and pH on Caco-2 cell permeability
Fulltext Access 9 Pages 2006
Bioadhesive monolayer film for the in vitro transdermal delivery of sumatriptan
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Primary Microparticles and Agglomerates of Morphine for Nasal Insufflation
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Thiol exchange: An in vitro assay that predicts the efficacy of novel homocysteine lowering therapies
Fulltext Access 9 Pages 2006
Labetalol absorption kinetics: Rat small intestine and colon studies
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Static light scattering and small-angle neutron scattering study on aggregated recombinant gelatin in aqueous solution
Fulltext Access 9 Pages 2006
An efficient approach for the rapid assessment of oral rat exposures for new chemical entities in drug discovery
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Release-Controlling Absorption Enhancement of Enterally Administered Ophiopogon Japonicus Polysaccharide by Sodium Caprate in Rats
Fulltext Access 9 Pages 2006
Metabolism of Dopamine by the Nasal Mucosa
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