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Daneshyari Pharmaceutical Science Journas Latest Articles

Pharmaceutical Science Research Articles

Synthesis and biological evaluation of selective tubulin inhibitors as anti-trypanosomal agents
Fulltext Access 26 Pages 2017
Development of gallic acid formazans as novel enoyl acyl carrier protein reductase inhibitors for the treatment of tuberculosis
Fulltext Access 26 Pages 2017
Rapid discrimination and determination of antibiotics drugs in plastic syringes using near infrared spectroscopy with chemometric analysis: Application to amoxicillin and penicillin
Fulltext Access 26 Pages 2017
Design, synthesis, and biological evaluation of a highly water-soluble psoralen-based photosensitizer
Fulltext Access 26 Pages 2017
Enhancement in recovery of drugs with high protein binding efficiency from human plasma using magnetic nanoparticles
Fulltext Access 26 Pages 2017
Rapid screening of non-steroidal anti-inflammatory drugs illegally added in anti-rheumatic herbal supplements and herbal remedies by portable ion mobility spectrometry
Fulltext Access 26 Pages 2017
Reliability of point-of-collection testing devices for drugs of abuse in oral fluid: A systematic review and meta-analysis
Fulltext Access 26 Pages 2017
Recent synthetic and medicinal perspectives of dihydropyrimidinones: A review
Fulltext Access 27 Pages 2017
Design, synthesis and structure-bactericidal activity relationships of novel 9-oxime ketolides and reductive epimers of acylides
Fulltext Access 27 Pages 2017
Impact of Chemical Structure on Conjunctival Drug Permeability: Adopting Porcine Conjunctiva and Cassette Dosing for Construction of In Silico Model
Fulltext Access 27 Pages 2017
Influence of a Small Amount of Glycerol on the Trehalose Bioprotective Action Analyzed In Situ During Freeze-Drying of Lyzozyme Formulations by Micro-Raman Spectroscopy
Fulltext Access 27 Pages 2017
Graphical contents list
Fulltext Access 27 Pages 2017
A benzothiazole/piperazine derivative with acetylcholinesterase inhibitory activity: Improvement in streptozotocin-induced cognitive deficits in rats
Fulltext Access 27 Pages 2017
Synthesis and biological evaluation of largazole zinc-binding group analogs
Fulltext Access 27 Pages 2017
Advances in the design of solid lipid nanoparticles and nanostructured lipid carriers for targeting brain diseases
Fulltext Access 27 Pages 2017
Cutaneous vaccination with coated microneedles prevents development of airway allergy
Fulltext Access 27 Pages 2017
Phytantriol based smart nano-carriers for drug delivery applications
Fulltext Access 27 Pages 2017
Simultaneously overcome tumor vascular endothelium and extracellular matrix barriers via a non-destructive size-controlled nanomedicine
Fulltext Access 27 Pages 2017
1,3,5-Triazines: A promising scaffold for anticancer drugs development
Fulltext Access 27 Pages 2017
Nebulizers and spacers for aerosol delivery through adult nasal cannula at low oxygen flow rate: An in-vitro study
Fulltext Access 27 Pages 2017
Attitudes and attributes of pharmacists in relation to practice change - A scoping review and discussion
Fulltext Access 27 Pages 2017
Surging footprints of mathematical modeling for prediction of transdermal permeability
Fulltext Access 27 Pages 2017
A High-Throughput Bioluminescent Assay to Monitor the Deamidation of Asparagine and Isomerization of Aspartate Residues in Therapeutic Proteins and Antibodies
Fulltext Access 27 Pages 2017
Supervised pelvic floor muscle training versus attention-control massage treatment in patients with faecal incontinence: Statistical analysis plan for a randomised controlled trial
Fulltext Access 27 Pages 2017
Pharmaceutical Amorphous Nanoparticles
Fulltext Access 27 Pages 2017
Development and characterization of the voriconazole loaded lipid-based nanoparticles
Fulltext Access 27 Pages 2017
On the Post-Compaction Evolution of Tensile Strength of Sodium Chloride-Starch Mixture Tablets
Fulltext Access 27 Pages 2017
Microflow Imaging Analyses Reflect Mechanisms of Aggregate Formation: Comparing Protein Particle Data Sets Using the Kullback-Leibler Divergence
Fulltext Access 27 Pages 2017
A Demonstration of Mixing Robustness in a Direct Compression Continuous Manufacturing Process
Fulltext Access 27 Pages 2017
Smart chemistry-based nanosized drug delivery systems for systemic applications: A comprehensive review
Fulltext Access 28 Pages 2017
Ibuprofen nanocrystals developed by 22 factorial design experiment: A new approach for poorly water-soluble drugs
Fulltext Access 28 Pages 2017
Supercritical fluid chromatography approach for a sustainable manufacture of new stereoisomeric anticancer agent
Fulltext Access 28 Pages 2017
Turning the screw even further to increase microparticle retention and ocular bioavailability of associated drugs: The bioadhesion goal
Fulltext Access 28 Pages 2017
In situ hydrogels enhancing postoperative functional recovery by reducing iron overload after intracerebral haemorrhage
Fulltext Access 28 Pages 2017
A chemiluminescence reagent free method for the determination of captopril in medicine and urine samples by using trivalent silver
Fulltext Access 28 Pages 2017
Simultaneous separation and determination of four uncaria alkaloids by capillary electrophoresis using dual cyclodextrin system
Fulltext Access 28 Pages 2017
Evaluation of ornidazole-loaded nanofibers as an alternative material for direct pulp capping
Fulltext Access 28 Pages 2017
Antimicrobial mangosteen extract infused alginate-coated gauze wound dressing
Fulltext Access 28 Pages 2017
Open innovation: Towards sharing of data, models and workflows
Fulltext Access 28 Pages 2017
On-Chip Preparation of Streptokinase Entrapped in Chitosan Nanoparticles Used in Thrombolytic Therapy Potentially
Fulltext Access 28 Pages 2017
Neuroprotective effect of cannabinoids nanoplatforms in neurodegenerative diseases
Fulltext Access 28 Pages 2017
Repurposing antipsychotic drugs into antifungal agents: Synergistic combinations of azoles and bromperidol derivatives in the treatment of various fungal infections
Fulltext Access 28 Pages 2017
Novel methyl indolinone-6-carboxylates containing an indole moiety as angiokinase inhibitors
Fulltext Access 28 Pages 2017
Melatonin pharmacokinetics after transdermal administration changes according to the time of the day
Fulltext Access 28 Pages 2017
Clinical translation of stem cell based interventions for spinal cord injury - Are we there yet?
Fulltext Access 28 Pages 2017
4-Aminoquinoline-ferrocenyl-chalcone conjugates: Synthesis and anti-plasmodial evaluation
Fulltext Access 28 Pages 2017
Phenyl butyrate inhibits pyruvate dehydrogenase kinase 1 and contributes to its anti-cancer effect
Fulltext Access 29 Pages 2017
Allometric size: The scientific theory and extension to normal fat mass
Fulltext Access 29 Pages 2017
Enhanced dissolution of poorly soluble antiviral drugs from nanoparticles of cellulose acetate based solid dispersion matrices
Fulltext Access 29 Pages 2017
Cardioprotective action of the aqueous extract of Terminalia arjuna bark against toxicity induced by doxorubicin
Fulltext Access 29 Pages 2017
Design, synthesis and antithrombotic evaluation of novel non-peptide thrombin inhibitors
Fulltext Access 29 Pages 2017
Simplified stratum corneum model membranes for studying the effects of permeation enhancers
Fulltext Access 29 Pages 2017
A Novel Approach for the Development of a Nanostructured Lipid Carrier Formulation by Hot-Melt Extrusion Technology
Fulltext Access 29 Pages 2017
Evaluation of Different Holder Devices for Freeze-Drying in Dual-Chamber Cartridges With a Focus on Energy Transfer
Fulltext Access 29 Pages 2017
Investigation of binding behaviour of procainamide hydrochloride with human serum albumin using synchronous, 3D fluorescence and circular dichroism
Fulltext Access 29 Pages 2017
Synthesis and in vitro degradation studies of substituted poly(organophosphazenes) for drug delivery applications
Fulltext Access 29 Pages 2017
Study of Rheology and Polymer Adsorption Onto Drug Nanoparticles in Pharmaceutical Suspensions Produced by Nanomilling
Fulltext Access 29 Pages 2017
Fill volume, humidification and heat effects on aerosol delivery and fugitive emissions during noninvasive ventilation
Fulltext Access 29 Pages 2017
Simultaneous quantification of endothelin receptor antagonists and phosphodiesterase 5 inhibitors currently used in pulmonary arterial hypertension
Fulltext Access 29 Pages 2017
Optimization of a new methodology for trace determination of elements in biological fluids: Application for speciation of inorganic selenium in children's blood
Fulltext Access 29 Pages 2017
Achievable separation performance and analysis time in current liquid chromatographic practice for monoclonal antibody separations
Fulltext Access 29 Pages 2017
Development and validation of a liquid chromatographic method for the analysis of squaric acid dibutyl ester and its impurities
Fulltext Access 29 Pages 2017
Enantiomeric separation of the antiuremic drug colchicine by electrokinetic chromatography. Method development and quantitative analysis
Fulltext Access 29 Pages 2017
Raman spectroscopy and capillary zone electrophoresis for the analysis of degradation processes in commercial effervescent tablets containing acetylsalicylic acid and ascorbic acid
Fulltext Access 29 Pages 2017
A comparison report of three advanced methods for drug-cyclodextrin interaction measurements
Fulltext Access 29 Pages 2017
Antibody-free detection of infectious bacteria using quantum dots-based barcode assay
Fulltext Access 29 Pages 2017
Determination of pharmaceutical residues in wastewater using high performance liquid chromatography coupled to quadrupole-Orbitrap mass spectrometry
Fulltext Access 29 Pages 2017
Serendipitous discovery of potent human head and neck squamous cell carcinoma anti-cancer molecules: A fortunate failure of a rational molecular design
Fulltext Access 29 Pages 2017
Therapeutic investigations of novel indoxyl-based indolines: A drug target validation and Structure-Activity Relationship of angiotensin-converting enzyme inhibitors with cardiovascular regulation and thrombolytic potential
Fulltext Access 29 Pages 2017
2-Aminothiophene scaffolds: Diverse biological and pharmacological attributes in medicinal chemistry
Fulltext Access 29 Pages 2017
Design, synthesis and biological evaluation of some novel sulfonamide derivatives as apoptosis inducers
Fulltext Access 29 Pages 2017
Amino acid or peptide conjugates of acridine/acridone and quinoline/quinolone-containing drugs. A critical examination of their clinical effectiveness within a twenty-year timeframe in antitumor chemotherapy and treatment of infectious diseases
Fulltext Access 29 Pages 2017
Comparative stability-indicating chromatographic methods for determination of 4-hexylresorcinol in pharmaceutical formulation and shrimps
Fulltext Access 29 Pages 2017
Potential of insulin nanoparticle formulations for oral delivery and diabetes treatment
Fulltext Access 29 Pages 2017
The release kinetics, antimicrobial activity and cytocompatibility of differently prepared collagen/hydroxyapatite/vancomycin layers: Microstructure vs. nanostructure
Fulltext Access 29 Pages 2017
Synthesis and biological evaluation of a new series of benzimidazole derivatives as antimicrobial, antiquorum-sensing and antitumor agents
Fulltext Access 29 Pages 2017
Sodium hydrogen exchanger inhibitory activity of benzotriazole derivatives
Fulltext Access 29 Pages 2017
Design, synthesis and structure-activity relationship studies of a novel focused library of 2,3,4-substituted oxazolidines with antiproliferative activity against cancer cell lines
Fulltext Access 29 Pages 2017
The role of hyaluronan as a drug carrier to enhance the bioavailability of extended release ophthalmic formulations. Hyaluronan-timolol ionic complexes as a model case
Fulltext Access 30 Pages 2017
Impact of Formulation Properties and Process Parameters on the Dispensing and Depositioning of Drug Nanosuspensions Using Micro-Valve Technology
Fulltext Access 30 Pages 2017
Hydrophilic interaction liquid chromatography method development and validation for the assay of HEPES zwitterionic buffer
Fulltext Access 30 Pages 2017
Development of new efficient method for isolation of phenolics from sea algae prior to their rapid resolution liquid chromatographic-tandem mass spectrometric determination
Fulltext Access 30 Pages 2017
Light-switchable systems for remotely controlled drug delivery
Fulltext Access 30 Pages 2017
Chemical analysis and potential endocrine activities of aluminium coatings intended to be in contact with cosmetic water
Fulltext Access 30 Pages 2017
Overview of solidification techniques for self-emulsifying drug delivery systems from industrial perspective
Fulltext Access 30 Pages 2017
Modeling in the quality by design environment: Regulatory requirements and recommendations for design space and control strategy appointment
Fulltext Access 30 Pages 2017
Use of ionic liquids as headspace gas chromatography diluents for the analysis of residual solvents in pharmaceuticals
Fulltext Access 30 Pages 2017
Asymmetric synthesis of novel triazole derivatives and their in vitro antiviral activity and mechanism of action
Fulltext Access 30 Pages 2017
Metabolic profiles of exudates from chronic leg ulcerations
Fulltext Access 30 Pages 2017
A Mechanism-Based Pharmacokinetic Enzyme Turnover Model for Dichloroacetic Acid Autoinhibition in Rats
Fulltext Access 30 Pages 2017
Biological and structural studies of phosphonium 'masked thiolate' compounds
Fulltext Access 30 Pages 2017
Paclitaxel-Loaded Magnetic Nanoparticles: Synthesis, Characterization, and Application in Targeting
Fulltext Access 30 Pages 2017
Re-evaluating the presumed superiority of amorphous nanoparticles over amorphous microscale solid dispersion in solubility enhancement of poorly soluble drugs
Fulltext Access 30 Pages 2017
Model Systems for Studying the Role of Canalicular Efflux Transporters in Drug-Induced Cholestatic Liver Disease
Fulltext Access 30 Pages 2017
Diurnal variation in the pharmacokinetics and brain distribution of morphine and its major metabolite
Fulltext Access 30 Pages 2017
Development of Maltodextrin-Based Immediate-Release Tablets Using an Integrated Twin-Screw Hot-Melt Extrusion and Injection-Molding Continuous Manufacturing Process
Fulltext Access 30 Pages 2017
Jet-vortex spray freeze drying for the production of inhalable lyophilisate powders
Fulltext Access 30 Pages 2017
Parameters Affecting the Enhanced Permeability and Retention Effect: The Need for Patient Selection
Fulltext Access 30 Pages 2017
Design, synthesis and evaluation of aromatic heterocyclic derivatives as potent antifungal agents
Fulltext Access 30 Pages 2017
Hot-melt extrusion as a continuous manufacturing process to form ternary cyclodextrin inclusion complexes
Fulltext Access 30 Pages 2017
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