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Pharmacology Research Articles

Evodiamine inhibits gastrointestinal motility via CCK and CCK1 receptor in water-avoidence stress rat model
Fulltext Access 7 Pages 2018
Cilostazol alleviates streptozotocin-induced testicular injury in rats via PI3K/Akt pathway
Fulltext Access 7 Pages 2018
Lipoxin A4 may attenuate the progression of obesity-related glomerulopathy by inhibiting NF-κB and ERK/p38 MAPK-dependent inflammation
Fulltext Access 7 Pages 2018
γ-Glutamylcysteine synthetase (γ-GCS) as a target for overcoming chemo- and radio-resistance of human hepatocellular carcinoma cells
Fulltext Access 7 Pages 2018
Strong carcinogenic stress response induction of preneoplastic cells positive for GST-P in the rat liver: Physiological mechanism for initiation
Fulltext Access 7 Pages 2018
Mild aerobic training with blood flow restriction increases the hypertrophy index and MuSK in both slow and fast muscles of old rats: Role of PGC-1α
Fulltext Access 7 Pages 2018
Growth-inhibition of S180 residual-tumor by combination of cyclophosphamide and chitosan oligosaccharides in vivo
Fulltext Access 7 Pages 2018
Astragaloside suppresses apoptosis of the podocytes in rats with diabetic nephropathy via miR-378/TRAF5 signaling pathway
Fulltext Access 7 Pages 2018
Exercise induced improvements in insulin sensitivity are concurrent with reduced NFE2/miR-432-5p and increased FAM3A
Fulltext Access 7 Pages 2018
Polymorphisms of human T cell epitopes of Mycobacterium tuberculosis indicate divergence of host immune pressure on different categories of proteins
Fulltext Access 7 Pages 2018
Pimozide suppresses colorectal cancer via inhibition of Wnt/β-catenin signaling pathway
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Down-regulation of lncRNA MEG3 promotes endothelial differentiation of bone marrow derived mesenchymal stem cells in repairing erectile dysfunction
Fulltext Access 7 Pages 2018
Clinical significance and functions of microRNA-93/CDKN1A axis in human cervical cancer
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Quercetin suppresses breast cancer stem cells (CD44+/CD24−) by inhibiting the PI3K/Akt/mTOR-signaling pathway
Fulltext Access 7 Pages 2018
Altered expression of Aquaporin-2 in one-kidney, one-clip hypertension
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Icariin alleviates murine lupus nephritis via inhibiting NF-κB activation pathway and NLRP3 inflammasome
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Immunomodulatory effects of Sceletium tortuosum (Trimesemine™) elucidated in vitro: Implications for chronic disease
Fulltext Access 7 Pages 2018
Immunomodulatory effects of a bioactive fraction of Strobilanthes crispus in NMU-induced rat mammary tumor model
Fulltext Access 7 Pages 2018
Extracts of Cordyceps sinensis inhibit breast cancer cell metastasis via down-regulation of metastasis-related cytokines expression
Fulltext Access 7 Pages 2018
D-chiro-inositol enriched Fagopyrum tataricum (L.) Gaench extract alleviates mitochondrial malfunction and inhibits ER stress/JNK associated inflammation in the endothelium
Fulltext Access 7 Pages 2018
Inhibitory effects of Aconiti Lateralis Radix Preparata on chronic intermittent cold-induced inflammation in the mouse hypothalamus
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Phytochemical characterization and biological activity evaluation of ethanolic extract of Cinnamomum zeylanicum
Fulltext Access 7 Pages 2018
Effect of Zembrin® and four of its alkaloid constituents on electric excitability of the rat hippocampus
Fulltext Access 7 Pages 2018
A new Alzheimer's disease cell model using B cells to induce beta amyloid plaque formation and increase TNF alpha expression
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Magnolol abrogates chronic mild stress-induced depressive-like behaviors by inhibiting neuroinflammation and oxidative stress in the prefrontal cortex of mice
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Carotid intima-media thickness and anti-hypertensive treatment: Focus on angiotensin II receptor blockers
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LC-MS guided isolation of gracilistones A and B, a pair of diastereomeric sesquiterpenoids with an unusual tetrahydrofuran-fused tricyclic skeleton from Acanthopanax gracilistylus and their potential anti-inflammatory activities
Fulltext Access 7 Pages 2018
Racemic phenylpropanoids from the root barks of Ailanthus altissima (Mill.) Swingle with cytotoxicity against hepatoma cells
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Acclimation of C2C12 myoblasts to physiological glucose concentrations for in vitro diabetes research
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Thermo-sensitive gel in glaucoma therapy for enhanced bioavailability: In vitro characterization, in vivo pharmacokinetics and pharmacodynamics study
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Systemic delivery of mesenchymal stem cells condition media in repeated doses acts as magic bullets in restoring IFN-γ/IL-4 balance in asthmatic rats
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Clinical utility of ABCB1 genotyping for preventing toxicity in treatment with irinotecan
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Lycodine-type alkaloids from Lycopodiastrum casuarinoides and their cholinesterase inhibitory activities
Fulltext Access 7 Pages 2018
New tetracyclic triterpenoids from Jatropha gossypiifolia induce cell-cycle arrest and apoptosis in RKO cells
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Terpenoids from the stems of Celastrus hindsii and their anti-RSV activities
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Chemical constituents from Daphne tangutica and their cytotoxicity against nasopharyngeal carcinoma cells
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Apigenin as neuroprotective agent: Of mice and men
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Treatment of hypertension: The ESH/ESC guidelines recommendations
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JMJD3 is involved in neutrophil membrane proteinase 3 overexpression during the hyperinflammatory response in early sepsis
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Enantiomer-specific positive allosteric modulation of CB1 signaling in autaptic hippocampal neurons
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Impact of adenosine A2a receptor polymorphism rs5751876 on platelet reactivity in ticagrelor treated patients
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Pharmacological intervention in hypertension using beta-blockers: Real‐world evidence for long-term effectiveness
Fulltext Access 7 Pages 2018
Cardiovascular diseases, NLRP3 inflammasome, and western dietary patterns
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Dihydroartemisinin induced caspase-dependent apoptosis through inhibiting the specificity protein 1 pathway in hepatocellular carcinoma SK-Hep-1 cells
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The α1,3-fucosyltransferase FUT7 regulates IL-1β-induced monocyte-endothelial adhesion via fucosylation of endomucin
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Delta-like homolog1/GATA binding protein 2 axis mediates leptin inhibition of PPARγ2 expression in hepatic stellate cells in vitro
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Increase in Ca2 + current by sustained cAMP levels enhances proliferation rate in GH3 cells
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TRPV1 alterations in urinary bladder dysfunction in a rat model of STZ-induced diabetes
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Triptolide inhibits pituitary adenoma cell viability, migration and invasion via ADAM12/EGFR signaling pathway
Fulltext Access 7 Pages 2018
Transferrin targeted liposomal 5-fluorouracil induced apoptosis via mitochondria signaling pathway in cancer cells
Fulltext Access 7 Pages 2018
New 4-methylidene sterols from the marine sponge Theonella swinhoei
Fulltext Access 7 Pages 2018
Flavonoid glycosides and alkaloids from the embryos of Nelumbo nucifera seeds and their antioxidant activity
Fulltext Access 7 Pages 2018
Monoterpenoid indole alkaloids from the leaves of Alstonia scholaris and their NF-κB inhibitory activity
Fulltext Access 7 Pages 2018
Isobenzofuranones from the aerial parts of Leontopodium leontopodioides (Wild.) Beauv.
Fulltext Access 7 Pages 2018
Silybin counteracts doxorubicin resistance by inhibiting GLUT1 expression
Fulltext Access 7 Pages 2018
New natural inhibitors of hexokinase 2 (HK2): Steroids from Ganoderma sinense
Fulltext Access 7 Pages 2018
Bioactive chemical constituents of Duboscia macrocarpa Bocq., and X-ray diffraction study of 11β, 12β-epoxyfriedours-14-en-3α-ol
Fulltext Access 7 Pages 2018
Chemodiversity of Cirsium fruits: Antiproliferative lignans, neolignans and sesquineolignans as chemotaxonomic markers
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Pursuing sesterterpene lactams in Australian Irciniidae sponges
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Caroguaianolide A-E, five new cytotoxic sesquiterpene lactones from Carpesium abrotanoides L.
Fulltext Access 7 Pages 2018
Cytotoxic carbazole alkaloid derivatives from the leaves and stems of Murraya microphylla
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Phenylpropanoids from the fruit of Crataegus pinnatifida exhibit cytotoxicity on hepatic carcinoma cells through apoptosis induction
Fulltext Access 7 Pages 2018
Racemic meroterpenoids from Ganoderma cochlear
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Two novel bioactive sulfated guaiane sesquiterpenoid salt alkaloids from the aerial parts of Scorzonera divaricata
Fulltext Access 7 Pages 2018
Cassaine diterpenoids from the seeds of Erythrophleum fordii and their cytotoxic activities
Fulltext Access 7 Pages 2018
An endophytic Fungi of Ginkgo biloba L. produces antimicrobial metabolites as potential inhibitors of FtsZ of Staphylococcus aureus
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Tanzawaic acid derivatives from freshwater sediment-derived fungus Penicillium sp.
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Three new quinazolines from Evodia rutaecarpa and their biological activity
Fulltext Access 7 Pages 2018
Variation of the alkaloid content of Peumus boldus (boldo)
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Spongian diterpenes from Chinese marine sponge Spongia officinalis
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Two new flavonoid-triterpene saponin meroterpenoids from Clinopodium chinense and their protective effects against anoxia/reoxygenation-induced apoptosis in H9c2 cells
Fulltext Access 7 Pages 2018
Cytotoxic indole alkaloids from Melodinus khasianus and Melodinus tenuicaudatus
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Trypanocidal activity of polysaccharide extract from Genipa americana leaves
Fulltext Access 7 Pages 2018
Evaluation of the aphrodisiac potential of a chemically characterized aqueous extract of Tamarindus indica pulp
Fulltext Access 7 Pages 2018
Hemostasis and uterine contraction promoting effect of the extract from drugs in the Zi-Yin-Tiao-Jing granule, a traditional Chinese compound preparation
Fulltext Access 7 Pages 2018
Cisatracurium induces mast cell activation and pseudo-allergic reactions via MRGPRX2
Fulltext Access 7 Pages 2018
IL-9 exhibits elevated expression in osteonecrosis of femoral head patients and promotes cartilage degradation through activation of JAK-STAT signaling in vitro
Fulltext Access 7 Pages 2018
Effects of ceftriaxone-induced intestinal dysbacteriosis on regulatory T cells validated by anaphylactic mice
Fulltext Access 7 Pages 2018
Regulatory T cells increase after treatment with poly (ADP-ribose) polymerase-1 inhibitor in ischemic stroke patients
Fulltext Access 7 Pages 2018
Treatment of Guillain-Barré syndrome with Bifidobacterium infantis through regulation of T helper cells subsets
Fulltext Access 7 Pages 2018
Costunolide ameliorates lipoteichoic acid-induced acute lung injury via attenuating MAPK signaling pathway
Fulltext Access 7 Pages 2018
Intestinal dysbacteriosis potentiates ovalbumin-induced allergic airway inflammation by inhibiting microRNA-130a to upregulate tumor necrosis factor α
Fulltext Access 7 Pages 2018
Montelukast inhibits inflammatory response in rheumatoid arthritis fibroblast-like synoviocytes
Fulltext Access 7 Pages 2018
Low-dose naltrexone (LDN): A promising treatment in immune-related diseases and cancer therapy
Fulltext Access 7 Pages 2018
Bone marrow derived M2 macrophages protected against lipopolysaccharide-induced acute lung injury through inhibiting oxidative stress and inflammation by modulating neutrophils and T lymphocytes responses
Fulltext Access 7 Pages 2018
IL-34 regulates IL-6 and IL-8 production in human lung fibroblasts via MAPK, PI3K-Akt, JAK and NF-κB signaling pathways
Fulltext Access 7 Pages 2018
Curcumin attenuates sepsis-induced acute organ dysfunction by preventing inflammation and enhancing the suppressive function of Tregs
Fulltext Access 7 Pages 2018
Activation of PPARγ by Curcumin protects mice from ischemia/reperfusion injury induced by orthotopic liver transplantation via modulating polarization of Kupffer cells
Fulltext Access 7 Pages 2018
Anti-inflammatory effects of Perillae Herba ethanolic extract against TNF-α/IFN-γ-stimulated human keratinocyte HaCaT cells
Fulltext Access 7 Pages 2018
Immunomodulatory effect of 1, 25 dihydroxy vitamin D3 on the expression of RNA sensing pattern recognition receptor genes and cytokine response in dengue virus infected U937-DC-SIGN cells and THP-1 macrophages
Fulltext Access 7 Pages 2018
Regulatory effects of chrysophanol, a bioactive compound of AST2017-01 in a mouse model of 2,4-dinitrofluorobenzene-induced atopic dermatitis
Fulltext Access 7 Pages 2018
The characteristics of beta 2-glycoprotein I-dependent anticardiolipin antibody and blood coagulation status in subjects with classical biological false-positive syphilis reactions
Fulltext Access 7 Pages 2018
Evaluation of a lymphocyte transformation test and cytokine detection assay to identify phenytoin and carbamazepine provoked DRESS or SJS/TEN in epilepsy patients
Fulltext Access 7 Pages 2018
Heme oxygenase-2 suppresses acute inflammation and improves the survival of skin allografts
Fulltext Access 7 Pages 2018
A cell-based test system for the assessment of pharmacokinetics of NOD1 and NOD2 receptor agonists
Fulltext Access 7 Pages 2018
Impairment of regulatory T cells in patients with neonatal necrotizing enterocolitis
Fulltext Access 7 Pages 2018
Monoamine oxidases inhibitors from Colvillea racemosa: Isolation, biological evaluation, and computational study
Fulltext Access 7 Pages 2018
C21-steroidal glycosides and sesquiterpenes from the roots of Cynanchum bungei and their inhibitory activities against the proliferation of B and T lymphocytes
Fulltext Access 7 Pages 2018
Diketopiperazines and 2H-pyran-2-ones with antioxidant activity from the rice fermented with Aspergillus luchuensis
Fulltext Access 7 Pages 2018
Identification of tagitinin C from Tithonia diversifolia as antitrypanosomal compound using bioactivity-guided fractionation
Fulltext Access 7 Pages 2018
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