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Pharmacology Research Articles

Kaempferol increases apoptosis in human cervical cancer HeLa cells via PI3K/AKT and telomerase pathways
Fulltext Access 5 Pages 2017
Vitamin D3 intake as regulator of insulin degrading enzyme and insulin receptor phosphorylation in diabetic rats
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Eupatilin prevents H2O2-induced oxidative stress and apoptosis in human retinal pigment epithelial cells
Fulltext Access 5 Pages 2017
Asymptomatic hyperuricemia is a strong risk factor for resistant hypertension in elderly subjects from general population
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The effect of Searsia chirindensis stem-bark extract on renal and liver function in a rat model of neurotoxicity
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Effectiveness of a Nintendo Wii balance board exercise programme on standing balance of children with cerebral palsy: A randomised clinical trial protocol
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Evaluation of hepatoprotective and antidiabetic activity of Alchemilla mollis
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Contrary influence of clinically applied sorafenib concentrations among hepatocellular carcinoma patients
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In vivo and in silico sedative-hypnotic like activity of 7-methyljuglone isolated from Diospyros lotus L.
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Knockdown of FOXR2 suppresses the tumorigenesis, growth and metastasis of prostate cancer
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Gastrodia elata attenuates inflammatory response by inhibiting the NF-κB pathway in rheumatoid arthritis fibroblast-like synoviocytes
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Phytochemicals of Pogostemon Cablin (Blanco) Benth. aqueous extract: Their xanthine oxidase inhibitory activities
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Neuroprotective effects of octreotide on diabetic neuropathy in rats
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H2S causes contraction and relaxation of major arteries of the rabbit
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Anatomic trisegmentectomy: An alternative treatment for huge or multiple hepatocellular carcinoma of right liver
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COMMD7 promotes hepatocellular carcinoma through regulating CXCL10
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Neuroprotection against hydrogen peroxide-induced toxicity by Dictyophora echinovolvata polysaccharide via inhibiting the mitochondria-dependent apoptotic pathway
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Sedative-hypnotic-like effect and molecular docking of di-naphthodiospyrol from Diospyros lotus in an animal model
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Effects of Paeonia emodi on hepatic cytochrome P450 (CYP3A2 and CYP2C11) expression and pharmacokinetics of carbamazepine in rats
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Antihyperlipidemic effect of Pistacia khinjuk
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Editorial overview: Use of PK-PD for antibacterial drug development: decreasing risk and paths forward for resistant pathogens
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Novel treatments for chronic hepatitis C: closing the remaining gaps
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Editorial overview: Gastrointestinal: New frontiers in therapeutics for GI diseases and disorders - from microRNAs to novel pharmaceutics, to low FODMAP diets and microbiome
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Two new steroidal saponins isolated from Anemarrhena asphodeloides
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New diterpenoids isolated from Leonurus japonicus and their acetylcholinesterase inhibitory activity
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Cycloartane triterpenoid and its glucoside isolated from Cassia occidentalis
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Clavuridins A and B, two new trinor-guaiane sesquiterpenes isolated from the Xisha soft coral Clavularia viridis
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Preparation and physicochemical characterization of T-OA PLGA microspheres
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Grape seed procyanidin B2 inhibits adipogenesis of 3T3-L1 cells by targeting peroxisome proliferator-activated receptor γ with miR-483-5p involved mechanism
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Efficacy of antiviral drug AV2 in the treatment of human papillomavirus-associated precancerous lesions of the uterine cervix: A randomized placebo-controlled clinical trial in Kinshasa, DR Congo. (KINVAV study)
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Recent advances in drug discovery of GPCR allosteric modulators for neurodegenerative disorders
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Measuring G protein-coupled receptor signalling in the brain with resonance energy transfer based biosensors
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Islet G-protein coupled receptors: therapeutic potential for diabetes
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Changes in Asthma Maintenance Therapy Prescribing Patterns Following the 2006 Long-acting β-Agonist FDA Drug Warning
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Risk Evaluation and Mitigation Strategies (REMS), Pemoline, and What Is a Signal?
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2017, Sexual Dimorphism, Sexual Pluralism, and More
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Vitamins C and D
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Dexmedetomidine inhibits activation of the MAPK pathway and protects PC12 and NG108-15 cells from lidocaine-induced cytotoxicity at its maximum safe dose
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Wearable technology to reduce sedentary behavior and CVD risk in older adults: Design of a randomized controlled trial
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The design and rationale of the Beijing Vascular Disease Patients Evaluation Study (BEST study)
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Assessing Community Cancer care after insurance ExpanSionS (ACCESS) study protocol
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Development of validated high-performance thin layer chromatography for quantification of aristolochic acid in different species of the Aristolochiaceae family
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Extending FDA guidance to include consumer medication information (CMI) delivery on mobile devices
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Modulation of proteolytic polyprotein processing by coxsackievirus mutants resistant to inhibitors targeting phosphatidylinositol-4-kinase IIIβ or oxysterol binding protein
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Replication of the Zika virus in different iPSC-derived neuronal cells and implications to assess efficacy of antivirals
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Enhanced protection against experimental Junin virus infection through the use of a modified favipiravir loading dose strategy
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Modeling HCV cure after an ultra-short duration of therapy with direct acting agents
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5-Hydroxytyrosol inhibits HIV-1 replication in primary cells of the lower and upper female reproductive tract
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Antiviral activity of the adenosine analogue BCX4430 against West Nile virus and tick-borne flaviviruses
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Comparison of three cell-based drug screening platforms for HSV-1 infection
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Herpes simplex virus type 1 abrogates the antiviral activity of Ch25h via its virion host shutoff protein
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Transmission of hepatitis E virus infection to human-liver chimeric FRG mice using patient plasma
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Co-administration of recombinant major envelope proteins (rA27L and rH3L) of buffalopox virus provides enhanced immunogenicity and protective efficacy in animal models
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Cost-benefit effectiveness of angiotensin-II receptor blockers in patients with uncomplicated hypertension: A comparative analysis
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Tenofovir alafenamide (TAF) does not deplete mitochondrial DNA in human T-cell lines at intracellular concentrations exceeding clinically relevant drug exposures
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Scoparone attenuates hepatic stellate cell activation through inhibiting TGF-β/Smad signaling pathway
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Molecular assessment of protective effect of Vitex negundo in ISO induced myocardial infarction in rats
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Omentin-1 prevents cartilage matrix destruction by regulating matrix metalloproteinases
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Flavonoids from Carya cathayensis Sarg. leaves inhibit carotid artery lesion formation induced by low blood flow
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Different profiles of the mRNA levels of DNA repair genes in MCF-7 and SH-SY5Y cells after treatment with combination of cisplatin, 50-Hz electromagnetic field and bleomycin
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Lianqinjiedu decoction attenuates LPS-induced inflammation and acute lung injury in rats via TLR4/NF-κB pathway
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Oxidative stress and some biochemical alterations due to scorpion (Leiurus quinquestriatus) crude venom in rats
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Buccal viral DNA as a trigger for brincidofovir therapy in the mousepox model of smallpox
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Inhibitory effect of Triperygium wilfordii polyglucoside on dipeptidyl peptidase I in vivo and in vitro
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Meeting report: Third Summer School on Innovative Approaches for Identification of Antiviral Agents (IAAASS)
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Immunomodulatory activities of phlorizin metabolites in lipopolysaccharide-stimulated RAW264.7 cells
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Role of pathogen-associated molecular patterns (PAMPS) in immune responses to fungal infections
Fulltext Access 6 Pages 2017
Naringin ameliorates diabetic nephropathy by inhibiting NADPH oxidase 4
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Stimulation of μ-opioid receptors dilates retinal arterioles by neuronal nitric oxide synthase-derived nitric oxide in rats
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l-carnitine preserves cardiac function by activating p38 MAPK/Nrf2 signalling in hearts exposed to irradiation
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Astilbin from Engelhardtia chrysolepis enhances intestinal barrier functions in Caco-2 cell monolayers
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ZD0947, a sulphonylurea receptor modulator, detects functional sulphonylurea receptor subunits in murine vascular smooth muscle ATP-sensitive K+ channels
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Oxidative stress inactivates ecto-5'-nucleotidase by inhibiting protein kinase C in rat hearts in vivo
Fulltext Access 6 Pages 2017
Effects of the 5-HT6 receptor antagonist idalopirdine on extracellular levels of monoamines, glutamate and acetylcholine in the rat medial prefrontal cortex
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Role of A1 and A2A adenosine receptor agonists in adipose tissue inflammation induced by obesity in mice
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MPP+ inhibits mGluR1/5-mediated long-term depression in mouse hippocampus by calpain activation
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Bis(benzofuran-thiazolidinone)s and bis(benzofuran-thiazinanone)s as inhibiting agents for chikungunya virus
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Conditioning neoadjuvant therapies for improved immunotherapy of cancer
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Detection of the hepatitis B virus (HBV) covalently-closed-circular DNA (cccDNA) in mice transduced with a recombinant AAV-HBV vector
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Protective effects of Donepezil against endothelial permeability
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Pre-and post-pandemic trends in antiviral use in hospitalized patients with laboratory-confirmed influenza: 2004/05-2013/14, Toronto, Canada
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Identification and evaluation of potent Middle East respiratory syndrome coronavirus (MERS-CoV) 3CLPro inhibitors
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Antileishmanial activity of verbascoside: Selective arginase inhibition of intracellular amastigotes of Leishmania (Leishmania) amazonensis with resistance induced by LPS plus IFN-γ
Fulltext Access 6 Pages 2017
4′-Azidocytidine (R1479) inhibits henipaviruses and other paramyxoviruses with high potency
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RO0504985 is an inhibitor of CMGC kinase proteins and has anti-human cytomegalovirus activity
Fulltext Access 6 Pages 2017
Full length articleChronic D609 treatment interferes with cell cycle and targets the expression of Olig2 in Glioma Stem like Cells
Fulltext Access 6 Pages 2017
Full length articlePTPN21 protects PC12 cell against oxygen-glucose deprivation by activating cdk5 through ERK1/2 signaling pathway
Fulltext Access 6 Pages 2017
Diosmin prevents left ventricular hypertrophy, adenosine triphosphatases dysfunction and electrolyte imbalance in experimentally induced myocardial infarcted rats
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Platycodin D suppressed LPS-induced inflammatory response by activating LXRα in LPS-stimulated primary bovine mammary epithelial cells
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Protective effect of forsythiaside A on OVA-induced asthma in mice
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miR-938 promotes colorectal cancer cell proliferation via targeting tumor suppressor PHLPP2
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Synergic stimulation of serotonin 5-HT1A receptor and α2-adrenoceptors for neuropathic pain relief: Preclinical effects of 2-substituted imidazoline derivatives
Fulltext Access 6 Pages 2017
Arctigenin improves vascular tone and decreases inflammation in human saphenous vein
Fulltext Access 6 Pages 2017
Hsp27 promotes ABCA1 expression and cholesterol efflux through the PI3K/PKCζ/Sp1 pathway in THP-1 macrophages
Fulltext Access 6 Pages 2017
The inhibitory effects of levo-tetrahydropalmatine on rat Kv1.5 channels expressed in HEK293 cells
Fulltext Access 6 Pages 2017
Psychopharmacology of combined activation of the serotonin1A and σ1 receptors
Fulltext Access 6 Pages 2017
Rimonabant, a selective cannabinoid1 receptor antagonist, protects against light-induced retinal degeneration in vitro and in vivo
Fulltext Access 6 Pages 2017
Effect of antiarrhythmic drugs on small conductance calcium - activated potassium channels
Fulltext Access 6 Pages 2017
Role of prostanoid EP3/1 receptors in mechanisms of emesis and defaecation in ferrets
Fulltext Access 6 Pages 2017
miR-455 inhibits breast cancer cell proliferation through targeting CDK14
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