Synthesis and evaluation of bifunctional nitrocatechol inhibitors of pig liver catechol-O-methyltransferase Fulltext Access 10 Pages 2005
Dual DNA recognition codes of a short peptide derived from the basic leucine zipper protein EmBP1 Fulltext Access 10 Pages 2005
Novel cytotoxic monotetrahydrofuranic Annonaceous acetogenins from Annona montana Fulltext Access 10 Pages 2005
Furoxan analogues of the histamine H3-receptor antagonist imoproxifan and related furazan derivatives Fulltext Access 10 Pages 2005
Design, modelling, synthesis and biological evaluation of peptidomimetic phosphinates as inhibitors of matrix metalloproteinases MMP-2 and MMP-8 Fulltext Access 10 Pages 2005
Design, synthesis, and biological evaluation of N-acetyl-2-(or 3-)carboxymethylbenzenesulfonamides as cyclooxygenase isozyme inhibitors Fulltext Access 10 Pages 2005
A new structural alternative in benzo[b]furans for antimicrobial activity Fulltext Access 10 Pages 2005
Density-functional theory and ab initio Hartree–Fork studies on the structural parameters and chemical activity of the free radicals generated by benzoquinone and hydroquinone Fulltext Access 10 Pages 2005
Synthesis and antitumor evaluation of novel 5-substituted-4-hydroxy-8-nitroquinazolines as EGFR signaling-targeted inhibitors Fulltext Access 10 Pages 2005
Synthesis and antitrichinellosis activity of some 2-substituted-[1,3]thiazolo[3,2-a]benzimidazol-3(2H)-ones Fulltext Access 10 Pages 2005
Design, synthesis, and biological characterization of potential antiatherogenic nitric oxide releasing tocopherol analogs Fulltext Access 10 Pages 2005
Improved synthesis of daunomycin conjugates with triplex-forming oligonucleotides. The polypurine tract of HIV-1 as a target Fulltext Access 10 Pages 2005
A cyclic PNA-based compound targeting domain IV of HCV IRES RNA inhibits in vitro IRES-dependent translation Fulltext Access 10 Pages 2005
Synthetic multifunctional pores that open and close in response to chemical stimulation Fulltext Access 10 Pages 2005
Design, synthesis, and biological evaluation of linear 1-(4-, 3- or 2-methylsulfonylphenyl)-2-phenylacetylenes: A novel class of cyclooxygenase-2 inhibitors Fulltext Access 10 Pages 2005
Homology modelling and active-site-mutagenesis study of the catalytic domain of the pneumococcal phosphorylcholine esterase Fulltext Access 10 Pages 2005
Structure–activity studies of uptake and phototoxicity with heavy-chalcogen analogues of tetramethylrosamine in vitro in chemosensitive and multidrug-resistant cells Fulltext Access 10 Pages 2005
9-Oxime-3-ketolides: Modification at the C-11,12-diol moiety and antibacterial activities against key respiratory pathogens Fulltext Access 10 Pages 2005
Antitumor activity and distribution of pyrroloiminoquinones in the sponge genus Zyzzya Fulltext Access 10 Pages 2005
Synthesis and cytotoxicity of epoxide and pyrazole analogs of the combretastatins Fulltext Access 10 Pages 2005
Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides: Antiviral activity and cellular toxicity Fulltext Access 10 Pages 2005
Design, synthesis, and biological evaluation of folic acid targeted tetraphenylporphyrin as novel photosensitizers for selective photodynamic therapy Fulltext Access 10 Pages 2005
Reaction of caesium 4-chlorophenate and chlorohydrins from threonines: synthesis of clofibrate analogues Fulltext Access 10 Pages 2005
New β-amino thiols as efficient catalysts for highly enantioselective alkenylzinc addition to aldehydes Fulltext Access 10 Pages 2005
Complexation between poly(acrylic acid) and poly(vinylpyrrolidone): Influence of the molecular weight of poly(acrylic acid) and small molecule salt on the complexation Fulltext Access 10 Pages 2005
Synthesis and properties of biodegradable elastomeric epoxy modified polyurethanes based on poly(ε-caprolactone) and poly(ethylene glycol) Fulltext Access 10 Pages 2005
Preparation and characterization of thiophene copolymers with second order non-linear optical properties Fulltext Access 10 Pages 2005
1H NMR studies of homo and mixed ligand complexes of Tl+ ion with several polyazamacrocycles Fulltext Access 10 Pages 2005
Properties and structure–activity studies of cyclic β-hairpin peptidomimetics based on the cationic antimicrobial peptide protegrin I Fulltext Access 10 Pages 2005
Cooperative lectin recognition of periodical glycoclusters along DNA duplexes: alternate hybridization and full hybridization Fulltext Access 10 Pages 2005
Synthesis of 9-alkyl and 9-heteroalkyl substituted 2-amino-6-guanidinopurines and their influence on the NO-production in macrophages Fulltext Access 10 Pages 2005
Synthesis and human NKT cell stimulating properties of 3-O-sulfo-α/β-galactosylceramides Fulltext Access 10 Pages 2005
Novel non-steroidal/non-anilide type androgen antagonists: discovery of 4-substituted pyrrole-2-carboxamides as a new scaffold for androgen receptor ligands Fulltext Access 10 Pages 2005
Preparation of highly substituted γ-lactam follicle stimulating hormone receptor agonists Fulltext Access 10 Pages 2005
3D-QSAR CoMFA studies on trypsin-like serine protease inhibitors: a comparative selectivity analysis Fulltext Access 10 Pages 2005
Design, synthesis, and structure–activity relationships of potent GPIIb/IIIa antagonists: discovery of FK419 Fulltext Access 10 Pages 2005
Combinatorial approach to identification of tyrphostin inhibitors of cytokine signaling Fulltext Access 10 Pages 2005
5-Arylidene-2-imino-4-thiazolidinones: Design and synthesis of novel anti-inflammatory agents Fulltext Access 10 Pages 2005
Synthesis of gossypol atropisomers and derivatives and evaluation of their anti-proliferative and anti-oxidant activity Fulltext Access 10 Pages 2005
Combinatorial design of nonsymmetrical cyclic urea inhibitors of aspartic protease of HIV-1 Fulltext Access 10 Pages 2005
Methyltrioxorhenium: a new catalyst for the activation of hydrogen peroxide to the oxidation of lignin and lignin model compounds Fulltext Access 10 Pages 2005
Structural modification of phenylpropanoid-derived compounds and the effects on their participation in redox processes Fulltext Access 10 Pages 2005
Design, synthesis, and biological evaluation of N-acetyl-2-carboxybenzenesulfonamides: a novel class of cyclooxygenase-2 (COX-2) inhibitors Fulltext Access 10 Pages 2005
Zidampidine, an aryl phosphate derivative of AZT: in vivo pharmacokinetics, metabolism, toxicity, and anti-viral efficacy against hemorrhagic fever caused by Lassa virus Fulltext Access 10 Pages 2005
New metal aminocarbene-substituted cyclopentadienyliron half sandwich complexes Fulltext Access 10 Pages 2005
Cluster-containing carbon-rich molecules: Reactions of ruthenium cluster carbonyls with {Au(PR3)}2(μ-CCCC) (R = Ph, tol) Fulltext Access 10 Pages 2005
Cationic arene ruthenium complexes containing chelating 1,10-phenanthroline ligands Fulltext Access 10 Pages 2005
Mechanistic studies on the formation of Pt(II) hydroformylation catalysts in imidazolium-based ionic liquids Fulltext Access 10 Pages 2005
Conformational behaviour of dinuclear Rh(I) complexes of the open-chain tetrapyrrolic ligand 2,2′-bidipyrrin (H2BDP) Fulltext Access 10 Pages 2005
Synthesis and structure of potential Lewis acid–Lewis base bifunctional catalysts: 2-N,N-Diisopropylaminophenylboronate derivatives Fulltext Access 10 Pages 2005
(Tetramethylcyclobutadiene)cobalt complexes with monoanionic carborane ligands [9-L-7,8-C2B9H10]− (L = SMe2, NMe3 and py) Fulltext Access 10 Pages 2005
Photochemical synthesis and spectroscopic characteristic of the first vinylsilane carbonyl complexes of tungsten(0) Fulltext Access 10 Pages 2005
Preparation of rhenium hydride complexes with pyrazole and pyrazolato ligands Fulltext Access 10 Pages 2005
Synthesis, reactivity and stereochemistry of new phosphorus heterocycles with 5- or 6-membered rings Fulltext Access 10 Pages 2005
Furan- and thiophene-functionalised bis-carbene ligands: Synthesis, silver(I) complexes, and catalysis Fulltext Access 10 Pages 2005
The first synthesis of cyclopropanone acetals from the reaction of Fischer carbene complexes with ketene acetals Fulltext Access 10 Pages 2005
On the ligand properties of the P- versus the N-heterocyclic carbene for a Grubbs catalyst in olefin metathesis Fulltext Access 10 Pages 2005
Luminescent coordination polymers with extended Au(I)–Ag(I) interactions supported by a pyridyl-substituted NHC ligand Fulltext Access 10 Pages 2005
Synthesis, structure and electronic properties of N-dialkylamino- and N-alkoxy-1,2,4-triazol-3-ylidene ligands Fulltext Access 10 Pages 2005
Synthesis and characterization of a free phenylene bis(N-heterocyclic carbene) and its di-Rh complex: Catalytic activity of the di-Rh and CCC–NHC Rh pincer complexes in intermolecular hydrosilylation of alkynes Fulltext Access 10 Pages 2005
The effect of substituents at silicon on the cross-metathesis of trisubstituted vinylsilanes with olefins Fulltext Access 10 Pages 2005
Synthesis and asymmetric catalytic application of chiral imidazolium–phosphines derived from (1R,2R)-trans-diaminocyclohexane Fulltext Access 10 Pages 2005
Silver alkoxide and amino N-heterocyclic carbenes; syntheses and crystal structures Fulltext Access 10 Pages 2005
Rhodium complexes of PCNHCP: Oxidative addition of dichloromethane and catalytic hydrosilylation of alkynes affording (E)-alkenylsilanes Fulltext Access 10 Pages 2005
Synthesis of hydrophilic Fischer carbene complexes as organometallic marker and PEGylating agent for proteins Fulltext Access 10 Pages 2005
Synthesis and NMR characterization of dinuclear Fe(II) organometallic complexes containing a non-equivalently bridging 5-aryl tetrazolate ligand Fulltext Access 10 Pages 2005
An anionic inositol phosphate glycan pseudotetrasaccharide exhibits high insulin-mimetic activity in rat adipocytes Fulltext Access 10 Pages 2005
Optimized N-phenyl-N′-(2-chloroethyl)ureas as potential antineoplastic agents: Synthesis and growth inhibition activity Fulltext Access 10 Pages 2005
Aza-bicyclic amino acid carboxamides as α4β1/α4β7 integrin receptor antagonists Fulltext Access 10 Pages 2005
Donepezil–tacrine hybrid related derivatives as new dual binding site inhibitors of AChE Fulltext Access 10 Pages 2005
Preparation of single-enantiomer semiochemicals using 2-methoxy-2-(1-naphthyl)propionic acid and 2-methoxy-2-(9-phenanthryl)propionic acid Fulltext Access 10 Pages 2005
Configurational assignment of vic-amino alcohols from their circular dichroism spectra with dirhodium tetracetate as an auxiliary chromophore Fulltext Access 10 Pages 2005
A new stereocontrolled approach to fused polycyclic compounds containing a diketopiperazine ring Fulltext Access 10 Pages 2005
Synthesis and structural characterization of diastereomeric isomers of RNA trimer adenylyl(3′-5′)adenylyl(3′-5′)adenosine Fulltext Access 10 Pages 2005
2-Chlorobicyclo[2.2.1]hept-5-ene-2-carboxamide and 2-chlorobicyclo[2.2.1]heptane-2-carboxamide as precursors of bicyclo[2.2.1]hept-5-en-2-one and bicyclo[2.2.1]heptan-2-one: resolution, absolute configuration and hydrogen-bonding properties Fulltext Access 10 Pages 2005
Asymmetric oxidation of sulfenates to sulfinates as a new route to optically active ortho-phosphorylated phenyl sulfoxides Fulltext Access 10 Pages 2005
α-Diimines as nitrogen ligands for ruthenium-catalyzed allylation reactions and related (pentamethylcyclopentadienyl) ruthenium complexes Fulltext Access 10 Pages 2005
Novel (η6-arene)-ruthenium(II) complexes containing bis(iminophosphorano)methanide and methandiide ligands Fulltext Access 10 Pages 2005
Copper, silver and gold-based catalysts for carbene addition or insertion reactions Fulltext Access 10 Pages 2005
Copper(I) complexes supported by a heavily fluorinated bis(pyrazolyl)borate: syntheses and characterization of [H2B(3,5-(CF3)2Pz)2]CuL (where L = PPh3, NCCH3, HCCPh, H2CCHPh) and {[H2B(3,5-(CF3)2Pz)2]Cu}2(1,5-COD) Fulltext Access 10 Pages 2005
Iridium mediated methyl and phenyl C–H activation of 2-(arylazo)phenols. Synthesis, structure, and spectral and electrochemical properties of some organoiridium complexes Fulltext Access 10 Pages 2005
Reactivity of [CpCr(CO)3]2 towards thione (CS) moieties in some sulfur-containing substrates Fulltext Access 10 Pages 2005
Reaction of Fe3(CO)12 with but-2-yn-1,4-diol, 1,4-dichloro-but-2-yne, propargyl-alcohol and propargyl-chloride.: The X-ray structures of [Fe2(CO)6{H2CCCCH2}], [Fe2(CO)6{H2CCC(H)C(OCH3)O}] and Fe3(CO)10{H2CCC(H)C(O)C{CH2(O)CH3}CCH2}] Fulltext Access 10 Pages 2005
New mononuclear ruthenium complexes of η5-cyclichydrocarbon containing azine ligands: Syntheses, spectral and structural studies Fulltext Access 10 Pages 2005
Synthesis and structural characterization of carbon-centered tris(pentafluorophenyl)silyl derivatives Fulltext Access 10 Pages 2005
Synthesis and structural characterization of unsymmetrical osmocenes containing the pentamethylcyclopentadienyl ligand Fulltext Access 10 Pages 2005
Synthesis and reactivity of cyclometallated platinum (II) compounds containing [C,N,Nâ²] terdentate ligands: Crystal structures of [PtCl{(CH3)2N(CH2)3NCH(4-ClC 6H3)}], [PtCl{(CH3)2N(CH2)3NCH(2-ClC6H3)}] and [PtCl{(CH3)2N(CH2)3NCH(3-(CH3)C6H3)}] Fulltext Access 10 Pages 2005
Part 1: 1,3-Dipolar addition of activated alkyne towards coordinated azido group in ruthenium(II) complexes containing η5-cyclichydrocarbons Fulltext Access 10 Pages 2005
Copper-mediated displacements of allylic THP ethers on a bisphosphonate template Fulltext Access 10 Pages 2005