Keywords: تست اتصال; Fragment-based drug discovery; Affinity capillary electrophoresis; Binding assay; Weak interaction drug-target; % inh; percentage of inhibition; μep; electrophoretic mobility; ACE; affinity capillary electrophoresis; AGB; 4-acetamidophenyl 4-guanidinoben
مقالات ISI تست اتصال (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: تست اتصال; Dual specific antibody; Bispecific antibody; Bioassay; Cell proliferation; Signaling pathways; Binding assay;
Keywords: تست اتصال; Nicotine analogues; Mycobacterium; Pharmacokinetics; Anti-TB activity; Binding assay; Deaddiction; MABA
Keywords: تست اتصال; Withania somnifera; Morphine; Antinociception; Hyperalgesia; Binding assay
Keywords: تست اتصال; Force spectroscopy; Protein–ligand interaction; Protein unfolding; Mechanical stability; Binding assay
Keywords: تست اتصال; Binding mechanism; Kinetics; Histone deacetylases; Inhibitors; Binding assay
Keywords: تست اتصال; High-performance liquid chromatography; Dissociation constant; Binding assay; High affinity;
In vitro and in vivo activity of cyclopeptide Dmt-c[d-Lys-Phe-Asp]NH2, a mu opioid receptor agonist biased toward β-arrestin
Keywords: تست اتصال; Cyclic opioid peptides; Binding assay; Calcium mobilization assay; Bioluminescence resonance energy transfer assay; Hot-plate test; Whole gastrointestinal transit test;
Development and validation of a bioassay to evaluate binding of adalimumab to cell membrane-anchored TNFα using flow cytometry detection
Keywords: تست اتصال; Adalimumab; Binding assay; Bioassay validation; Flow cytometry; Membrane TNFα;
Okaramine insecticidal alkaloids show similar activity on both exon 3c and exon 3b variants of glutamate-gated chloride channels of the larval silkworm, Bombyx mori
Keywords: تست اتصال; BmGluCl; Bombyx mori glutamate-gated chloride channel; Okaramines; Ivermectin; Glutamate-gated chloride channels; Silkworm (Bombyx mori); Voltage-clamp electrophysiology; Binding assay;
Herbicide and insect resistant Bt cotton pollen assessment finds no detrimental effects on adult honey bees
Keywords: تست اتصال; Apis mellifera; Cry toxin; qRT-PCR; Binding assay;
Research PaperSynthesis and activity of opioid peptidomimetics with β2- and β3-amino acids
Keywords: تست اتصال; β-amino acids; Peptide synthesis; Binding assay; Calcium mobilization assay; Writhing test; Enzymatic degradation;
Assessment of new triplet forming artificial nucleobases as RNA ligands directed towards HCV IRES IIId loop
Keywords: تست اتصال; Hepatitis virus C; IRES IIId loop; RNA ligands; Inhibitors; Binding assay;
A novel method for detection of IFN-lambda 3 binding to cells for quantifying IFN-lambda receptor expression
Keywords: تست اتصال; Interferon-lambda; Interferon-lambda receptor; Flow cytometry; Binding assay; Interferon-stimulated genes;
Expression, characterisation and antigenicity of a truncated Hendra virus attachment protein expressed in the protozoan host Leishmania tarentolae
Keywords: تست اتصال; Hendra virus; Attachment protein; Leishmania tarentolae; Protein expression; Binding assay;
Identification and functional characterization of tumor necrosis factor receptor 1 (TNFR1) of grass carp (Ctenopharyngodon idella)
Keywords: تست اتصال; TNF-α receptor 1; Molecular characterization; Binding assay; Functional identification; Grass carp;
Discovery of 2-(3,4-dichlorophenoxy)-N-(2-morpholin-4-ylethyl)acetamide: A selective σ1 receptor ligand with antinociceptive effect
Keywords: تست اتصال; Pain; σ receptors; Binding assay; Formalin test
New 2-Aminothiazoline derivatives lower blood pressure of spontaneously hypertensive rats (SHR) via I1-imidazoline and alpha-2 adrenergic receptors activation
Keywords: تست اتصال; Imidazoline receptor; Aminothiazoline; Hypertension; PC12 cells; Binding assay;
Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABAA receptors containing the α5 subunit
Keywords: تست اتصال; Amide compound; Receptor efficacy; Binding assay; Free brain concentration; Rat kinetics; Basic behavior;
Development of microfluidic-based assays to estimate the binding between osteocalcin (BGLAP) and fluorescent antibodies
Keywords: تست اتصال; Osteocalcin (BGLAP); Binding assay; Fluorescent antibodies
'Turn On/Off' fluorescence probe for the screening of unactivated Bruton's tyrosine kinase
Keywords: تست اتصال; Bruton's tyrosine kinase; Fluorescence probe; Kinase inhibitor; Binding assay;
Radiosynthesis and in vitro validation of 3H-NS14492 as a novel high affinity alpha7 nicotinic receptor radioligand
Keywords: تست اتصال; Bmax; maximum density; 125I-BTX; 125I-α-bungarotoxin; Kd; dissociation constant; Ki; inhibition constant; NSB; non-specific binding; OD; optical density; PAM; positive allosteric modulator; SB; specific binding; TB; total binding; TE; tissue equivalent;
In vitro and ex vivo characterization of (−)-TZ659 as a ligand for imaging the vesicular acetylcholine transporter
Keywords: تست اتصال; Vesicular acetylcholine transporter; Radioligand; Binding assay; Autoradiography
Novel agonists of benzodiazepine receptors: Design, synthesis, binding assay and pharmacological evaluation of 1,2,4-triazolo[1,5-a]pyrimidinone and 3-amino-1,2,4-triazole derivatives
Keywords: تست اتصال; Synthesis; Benzodiazepine agonists; Binding assay; Hypnotic activity
Basic neuroscienceUse of radiolabeled antagonist assays for assessing agonism at D2 and D3 dopamine receptors: Comparison with functional GTPγS assays
Keywords: تست اتصال; Dopamine receptors; [3H]spiperone binding; [35S] GTPγS binding; GTP shift; Efficacy; Affinity; Binding assay; Functional assay; D2 receptors; D3 receptors;
Separation and peroxisome proliferator-activated receptor-γ agonist activity evaluation of synthetic racemic bavachinin enantiomers
Keywords: تست اتصال; ALWPIHGZAXQYLV-ZCLATKBISA-N; Bavachinin; PPAR-γ; Supercritical fluid chromatography; Binding assay; Molecular docking;
Homoisoflavonoids as potential imaging agents for β-amyloid plaques in Alzheimer's disease
Keywords: تست اتصال; Alzheimer's disease; Amyloid; Imaging agent; Homoisoflavonoid; Binding assay
FACS binding assay for analysing GDNF interactions
Keywords: تست اتصال; DOL; Degree of labelling; FACS; Fluorescent-activated cell sorting; GDNF; Glial cell-line derived neurotrophic factor; G-CSF; granulocyte-colony stimulating factor; GFRα; GDNF Family receptor alpha; GDNF488; GDNF conjugated with Alexa 488; 293T-GFR1; 293
Development of a fluorescence polarization binding assay for folate receptor
Keywords: تست اتصال; Binding assay; Membrane extracts; KB cells
Evaluation of potential Myt1 kinase inhibitors by TR-FRET based binding assay
Keywords: تست اتصال; Protein kinase Myt1; Binding assay; Inhibitor; Organic synthesis; DockingBCA, bicinchoninic acid; Cdk1, cyclin dependent kinase 1; CycB, cyclin B; DMSO, dimethylsulfoxide; DTT, dithiothreitol; GGL, glycoglycerolipid; HEK, human embryonic kidney; HR-MS, hi
Förster resonance energy transfer competitive displacement assay for human soluble epoxide hydrolase
Keywords: تست اتصال; Soluble epoxide hydrolase; Binding assay; Competitive displacement assay; Förster resonance energy transfer (FRET); Fluorescent assay
Development of a fluorescence polarization binding assay for asialoglycoprotein receptor
Keywords: تست اتصال; Binding assay; Membrane extracts; Crude receptor extract
A versatile method to measure the binding to basic proteins by surface plasmon resonance
Keywords: تست اتصال; SPR; Binding assay; TATA box-binding protein (TBP); Histone; Ribosomal protein;
Synthesis and evaluation of 17α-(dimethylphenyl)vinyl estradiols as probes of the estrogen receptor-α ligand binding domain
Keywords: تست اتصال; Steroidal estrogens; Estrogen receptor; Ligand binding domain; Synthesis; Molecular modeling; Binding assay;
Design and synthesis of marine fungal phthalide derivatives as PPAR-γ agonists
Keywords: تست اتصال; PPAR-γ; Phthalide; Marine fungus; Binding assay; Luciferase assay
Frontal affinity chromatography with MS detection of the ligand binding domain of PPARγ receptor: Ligand affinity screening and stereoselective ligand–macromolecule interaction
Keywords: تست اتصال; HPAC; FAC–MS; Immobilized PPARγ receptor; Binding assay; Ligand affinity screening; Enantioselective binding
Three pheromone-binding proteins help segregation between two Helicoverpa species utilizing the same pheromone components
Keywords: تست اتصال; Pheromone-binding protein; Helicoverpa armigera; Helicoverpa assulta; Western blot; Conformational change; Binding assay
Novel quinoxaline derivatives for in vivo imaging of β-amyloid plaques in the brain
Keywords: تست اتصال; Alzheimer’s disease; β-Amyloid; Imaging agent; Binding assay; Autoradiography
Comparative analysis of binding affinities to epidermal growth factor receptor of monoclonal antibodies nimotuzumab and cetuximab using different experimental animal models
Keywords: تست اتصال; Binding assay; Cetuximab; EGF receptor; Nimotuzumab; Placenta
Parecoxib and its metabolite valdecoxib directly interact with cannabinoid binding sites in CB1-expressing HEK 293 cells and rat brain tissue
Keywords: تست اتصال; COX 2 inhibitor; Cannabinoid receptor; Binding assay; HEK 293 cells; Brain
Inflammation Triggers Constitutive Activity and Agonist-induced Negative Responses at M3 Muscarinic Receptor in Dental Pulp
Keywords: تست اتصال; Binding assay; constitutive receptor activity; dental pulp; M3 muscarinic receptor; nitric oxide synthase; pilocarpine; pulpitis;
Synthesis and evaluation of benzofuran-2-yl(phenyl)methanone derivatives as ligands for β-amyloid plaques
Keywords: تست اتصال; Alzheimer’s disease; β-Amyloid; Imaging agent; Binding assay; Autoradiography
Novel (E)-5-styryl-2,2′-bithiophene derivatives as ligands for β-amyloid plaques
Keywords: تست اتصال; Alzheimer’s disease; β-amyloid plaques; Imaging agent; Bithiophene; Binding assay
Bisubstrate fluorescent probes and biosensors in binding assays for HTS of protein kinase inhibitors
Keywords: تست اتصال; ARC; adenosine analogue-oligoarginine conjugate; CHO; Chinese Hamster Ovary; EFC; enzyme fragment complementation technology; FA; fluorescence anisotropy; FITC; Fluorescein isothiocyanate; FRET; Förster-resonance energy transfer; GST; glutathione S-tra
A fluorescence polarization-based assay for the identification and evaluation of calmodulin antagonists
Keywords: تست اتصال; Fluorescence polarization; Calmodulin; Cy5–W-7; Fluorescent labeling; Binding assay; Binding affinity; High-throughput screening
Modified binding assay for improved sensitivity and specificity in the detection of residual pertussis toxin in vaccine preparations
Keywords: تست اتصال; Pertussis toxin; Pertussis vaccine; Binding assay; Alternative to animal testing
Development of a selective competitive receptor binding assay for the determination of the affinity to NR2B containing NMDA receptors
Keywords: تست اتصال; NMDA receptor; NR2B; Ifenprodil; Recombinant receptor; Binding assay
In vitro determination of tetanus toxicity by an endopeptidase assay linked to a ganglioside-binding step
Keywords: تست اتصال; Clostridial neurotoxins; Tetanus neurotoxin; In vitro; Endopeptidase assay; Binding assay; Synaptobrevin; Gangliosides; BoNT; botulinum neurotoxin; BSA; bovine serum albumin; EP; European Pharmacopoeia; H-chain; heavy chain; L-chain; light chain; Lf; limi
Assessment of a recombinant androgen receptor binding assay: Initial steps towards validation
Keywords: تست اتصال; Rat recombinant androgen receptor; Binding assay; Screening for endocrine active compounds;
Generating artificial homologous proteins according to the representative family character in molecular mechanics properties – an attempt in validating an underlying rule of protein evolution
Keywords: تست اتصال; Protein evolution; Protein design; Hydrophobic interaction; Hydration; Binding assay