Keywords: کولین استراز; AChE; acetylcholinesterase; BChE; butyrylcholinesterase; ChEs; cholinesterases; CWA; chemical warfare agents; CWNA; chemical warfare nerve agent; EI; enzyme-inhibitor conjugate; EVB; empirical valence bond; FE; free energy; MD; molecular dynamics; NA; ner
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Keywords: کولین استراز; Ion-selective electrode; Potentiometry; Cholinesterases; Binding affinity; Anticholinesterase; Neostigmine;
Keywords: کولین استراز; AADAC; arylacetamide deacetylase; AChE; acetylcholinesterase; AEA; arachidonoylethanolamide; 2-AG; 2-arachidonoylglycerol; BChE; butyrylcholinesterase; BBB; blood-brain barrier; CES1; carboxylesterases 1; CES2; carboxylesterases 2; CNS; central nervous sy
Keywords: کولین استراز; Taurine; Cognitive impairment; Cholinesterases; Inflammatory cytokines; ROCK-II; ChAT;
Keywords: کولین استراز; NG-Nitro-l-arginine methyl ester; 7-Nitroindazole; Malathion; Oxidative stress; Cholinesterases; Comet assay;
Synthesis of readily available fluorophenylalanine derivatives and investigation of their biological activity
Keywords: کولین استراز; AChE; acetylcholinesterase; BAC; bacitracin; BChE; butyrylcholinesterase; ChE; cholinesterases; DMAP; 4-(dimethylamino)pyridine; EDC; N-(3-dimethylaminopropyl)-Nâ²-ethylcarbodiimide hydrochloride; ESBL; extended-spectrum β-lactamase; FLU; fluconazole; m
Keywords: کولین استراز; ACh; acetylcholine; ChEs; cholinesterases; AChE; acetylcholinesterase; EeAChE; AChE from Electrophorus electricus; hAChE; human acetylcholinesterase; BuChE; butyrylcholinesterase; eqBuChE; BChE from equine serum; ChEI; ChE inhibitor; AChEI; AChE inhibitor
Keywords: کولین استراز; Organophosphorus compounds; pesticides; mass spectrometry; in silico; cholinesterases; alpha/beta hydrolases;
Keywords: کولین استراز; Cannabis sativa; Tramadol; Cholinesterases; Memory; Cognitive decline;
Keywords: کولین استراز; Esterases; Paraoxonase-1; Cholinesterases; Pesticides; SNPs;
Keywords: کولین استراز; Aβ; β-amyloid; AD; Alzheimer's disease; AChE; acetylcholinesterase; BuChE; butyrylcholinesterase; BuLi; butyl lithium; DTNB; 5,5â²-dithiobis 2-nitrobenzoic acid; HPLC; high performance liquid chromatography; HRMS; high resolution mass spectrum; LRMS;
Keywords: کولین استراز; Cholinesterases; Biochemical biomarkers; Pseudosida ramosa; Native species; Tropical ecotoxicology
Keywords: کولین استراز; Pyrazolobenzothiazine; Benzimidazole; Hybrid compounds; Cholinesterases; Docking studies
Keywords: کولین استراز; JTLGJFBDQUBICH-UHFFFAOYSA-N; FEBATDALCUAQCM-UHFFFAOYSA-N; KZASLSLPFQAZRC-UHFFFAOYSA-N; APTXIDCPFDQWLD-UHFFFAOYSA-N; ZPMMPPBRCTWMHF-UHFFFAOYSA-N; LYXYENKXUDZGBB-UHFFFAOYSA-N; JKJRTNOOSNWMJV-UHFFFAOYSA-N; REFAZYLZAXUBGI-UHFFFAOYSA-N; RONHWZKWQSMGNP-UHFFFAOY
Keywords: کولین استراز; AChE; acetylcholinesterase; BChE; butyrylcholinesterase; BChE â/â mouse; butyrylcholinesterase knock-out mouse; ChE; cholinesterases; DTNB; 5,5-dithiobis(2-nitrobenzoic acid); isoOMPA; tetraisopropylpyrophosphoramide; Mouse butyrylcholinesterase; Mono
Keywords: کولین استراز; Enzyme kinetics; Cholinesterases; Parameter estimation;
Keywords: کولین استراز; CES; carboxylesterases; ChE; cholinesterase; CI50; concentration that produce 50% of inhibition; DTNB; 5,5´-dithio-2-bis-nitrobenzoate; G; gonads; GST; glutation S-transferase; OP; organophosphate insecticide; p-NPA; p-nitrophenyl acetate; p-NPB; p-nitro
The organophosphorus pesticide dimethoate decreases cell viability and induces changes in different biochemical parameters of rat pancreatic stellate cells
Keywords: کولین استراز; Calcium; Dimethoate; Esterase activity; Organophosphorus insecticide; Pancreatic stellate cells; ACh; Acetylcholine; AChE; Acetylcholinesterase; BChE; Butyrylcholinesterase; [Ca2+]i; Intracellular free Ca2+ concentration; CbEs; Carboxylesterases; ChE; Cho
Biological, chemical and in silico fingerprints of Dianthus calocephalus Boiss.: A novel source for rutin
Keywords: کولین استراز; α-amylase; Cholinesterases; Tyrosinase; Phenolics; Molecular docking and dynamics; Natural agents;
Design and synthesis of novel coumarin-pyridinium hybrids: In vitro cholinesterase inhibitory activity
Keywords: کولین استراز; Cholinesterases; Coumarins; Docking study; Kinetic study; Pyridinium salts; β-secretase (BACE1);
Synthesis and characterization of new inhibitors of cholinesterases based on N-phenylcarbamates: In vitro study of inhibitory effect, type of inhibition, lipophilicity and molecular docking
Keywords: کولین استراز; Carbamates; Monosaccharide derivatives; Cholinesterases; IC50; Molecular modeling; Water bridge;
Cholinesterase-inhibitory effect and in silico analysis of alkaloids from bulbs of Hieronymiella species
Keywords: کولین استراز; Amaryllidaceae; Hieronymiella; Cholinesterases; In silico; Alkaloids; Argentina; AChE; acetylcholinesterase enzyme; BChE; butyrylcholinesterase enzyme; E; extracts;
Synthesis, structure-activity relationship and molecular docking studies of 3-O-flavonol glycosides as cholinesterase inhibitors
Keywords: کولین استراز; Flavonoids; Flavonols; 3-Hydroxyflavones; Glycosides; Cholinesterases; AChE/BChE inhibitors; Molecular docking studies;
Design, facile synthesis, and evaluation of novel spiro- and pyrazolo[1,5-c]quinazolines as cholinesterase inhibitors: Molecular docking and MM/GBSA studies
Keywords: کولین استراز; Spiro-pyrazolo[1,5-c]quinazolines; MW irradiation; Cholinesterases; Molecular docking; MM/GBSA calculations;
Superior efficacy of HI-6 dimethanesulfonate over pralidoxime methylsulfate against Russian VX poisoning in cynomolgus monkeys (Macaca fascicularis)
Keywords: کولین استراز; AIBC; dual-chambered autoinjector; AS; atropine sulfate; AVZ; avizafone chlorhydrate; HI-6 DMS; HI-6 dimethanesulfonate; OPNA; organophosphorus nerve agents; i.m.; intramuscular; i.v.; intravenous; LD50; lethal dose 50%; ChEs; cholinesterases; AChEs; acet
Evaluation of oxidative stress and antioxidant status, serum trace mineral levels and cholinesterases activity in cattle infected with Anaplasma marginale
Keywords: کولین استراز; Anaplasma marginale; Antioxidants; Oxidative stress; Serum trace minerals; Cholinesterases;
Quercetin treatment regulates the Na+,K+-ATPase activity, peripheral cholinergic enzymes, and oxidative stress in a rat model of demyelination
Keywords: کولین استراز; ACh; acetylcholine; AChE; acetylcholinesterase; AcSCh; acetylthiocholine; BuChE; butyrylcholinesterase; CAT; catalase; CNS; central nervous system; DTNB; 5,5â²-dithio-bis-2-nitrobenzoic acid; EB; ethidium bromide; Hb; hemoglobin; MDA; malondialdehyde; MS
Novel in vitro and in silico insights of the multi-biological activities and chemical composition of Bidens tripartita L.
Keywords: کولین استراز; Anti-proliferative; Antioxidant; α-glucosidase; DNA protection; Anti-cancer; Cholinesterases;
Aflatoxins produced by Aspergillus parasiticus present in the diet of quails increase the activities of cholinesterase and adenosine deaminase
Keywords: کولین استراز; Aspergillus parasiticus; Adenosine deaminase; Aflatoxins; Cholinesterases; Quails;
Synthesis, crystal structure determination, biological screening and docking studies of N1-substituted derivatives of 2,3-dihydroquinazolin-4(1H)-one as inhibitors of cholinesterases
Keywords: کولین استراز; N-alkylated-2,3-dihydroquinazolin-4(1H)-one; Cholinesterases; Alzheimer's disease; Benzylation; Computational studies;
Synthesis, biological evaluation and docking studies of 2,3-dihydroquinazolin-4(1H)-one derivatives as inhibitors of cholinesterases
Keywords: کولین استراز; 2,3-Dihydroquinazolin-4(1H)-one; Dual inhibitors; Cholinesterases; Alzheimer's disease;
Design, synthesis and biological activity of novel donepezil derivatives bearing N-benzyl pyridinium moiety as potent and dual binding site acetylcholinesterase inhibitors
Keywords: کولین استراز; Alzheimer's disease; Donepezil; Benzylpyridinium; Acetylcholinesterase inhibitors antioxidant; β-Amyloid aggregation; Neuroprotection; AD; Alzheimer's disease; ChEs; Cholinesterases; ACh; acetylcholine; AChE; acetylcholinesterase; BuChE; butyrylcholinest
N-acetylcysteine protects memory decline induced by streptozotocin in mice
Keywords: کولین استراز; Cognition; Cholinesterases; Acetylcholine; Behavioral
Alterations of Na+/K+-ATPase, cholinergic and antioxidant enzymes activity by protocatechuic acid in cadmium-induced neurotoxicity and oxidative stress in Wistar rats
Keywords: کولین استراز; Cadmium; Protocatechuic acid; Enzymes; Na+/K+ ATPase; Cholinesterases; Antioxidant
Use of cholinesterase activity as an ecotoxicological marker to assess anatoxin-a(s) exposure: Responses of two cladoceran species belonging to contrasting geographical regions
Keywords: کولین استراز; Anatoxin-a(s); Microcystins; Cholinesterases; Biochemical biomarkers; Cyanobacterial blooms; Native species
Iminosugars as a new class of cholinesterase inhibitors
Keywords: کولین استراز; Iminosugars; Cholinesterases; Inhibitors; Alzheimer disease;
Evaluation of ecotoxicological effects of drugs on Daphnia magna using different enzymatic biomarkers
Keywords: کولین استراز; Acetaminophen; Chlorpromazine; Diclofenac; Propranolol; Cholinesterases; Oxidative stress
Does zebra mussel (Dreissena polymorpha) represent the freshwater counterpart of Mytilus in ecotoxicological studies? A critical review
Keywords: کولین استراز; Bivalve; Biological model; Biomarker; Proteomics; Transcriptomics; MTT; 3(4,5-dimethyl-2thiazholyl)-2,5-diphenyl-2H-tetrazolium bromide); MDMA; 3,4-methylenedioxymethamphetamine; AChE; acetylcholinesterase; ABM; active biomonitoring; ALP; alkaline phospha
(â)-Meptazinol-melatonin hybrids as novel dual inhibitors of cholinesterases and amyloid-β aggregation with high antioxidant potency for Alzheimer's therapy
Keywords: کولین استراز; AD; Alzheimer's disease; Aβ; amyloid-β; ACh; acetylcholine; AChE; acetylcholinesterase; AChEIs; acetylcholinesterase inhibitors; BChE; butyrylcholinesterase; BBB; blood-brain barrier; CAS; catalytic anionic site; ChEs; cholinesterases; CCK-8; cell c
Synthesis, biological evaluation and molecular docking study of novel piperidine and piperazine derivatives as multi-targeted agents to treat Alzheimer's disease
Keywords: کولین استراز; Alzheimer's disease; Multi-target directed ligands; Cholinesterases; Aβ aggregation; Antioxidants; Molecular docking;
Assessing Jasminum grandiflorum L. authenticity by HPLC-DAD-ESI/MSn and effects on physiological enzymes and oxidative species
Keywords: کولین استراز; Jasminum grandiflorum L.; HPLC-DAD-ESI/MSn; Phenolic compounds; Cholinesterases; MAO-A; Oxidative species;
Design, synthesis and evaluation of novel tacrine-(β-carboline) hybrids as multifunctional agents for the treatment of Alzheimer's disease
Keywords: کولین استراز; OLKLOVAJULLISR-UHFFFAOYSA-N; WUZJRHKAIFSDMM-UHFFFAOYSA-N; XKKFXCKMPXLPKK-UHFFFAOYSA-N; WKAJCZZPMZGMDI-UHFFFAOYSA-N; ZXEXKQSBZMYPAQ-UHFFFAOYSA-N; UTSQNVLOMVPCIW-YTTGMZPUSA-N; LBOYVYBBAFDIGX-NDEPHWFRSA-N; HLSFNIKGKKTOIA-TWAVRPEISA-N; HSQBZWURRKNSMR-TXMUIZFD
Modulation of the endogenous antioxidants paraoxonase-1 and urate by pesticide exposure and genetic variants of xenobiotic-metabolizing enzymes
Keywords: کولین استراز; Pesticide exposure; Cholinesterases; Endogenous antioxidants; Pesticidemetabolising gene variants; Occupational health
Intérêt du dosage des cholinestérases dans le cadre des intoxications aux organophosphorés
Keywords: کولین استراز; Biomarqueurs; Cholinestérases; Exposition; Neurotoxiques organophosphorésBiomarkers; Cholinesterases; Exposure; Organophosphorus agents
Evaluation of pesticide-induced oxidative stress from a gene–environment interaction perspective
Keywords: کولین استراز; Pesticide exposure; Cholinesterases; Pesticide-metabolizing genes; Biomarkers of susceptibility; Occupational health
Effect of different extraction methodologies on the recovery of bioactive metabolites from Satureja parvifolia (Phil.) Epling (Lamiaceae)
Keywords: کولین استراز; Satureja parvifolia (Phil.) Epling; Phenolic compounds; Volatile compounds; Antioxidant; Cholinesterases
Characterization of type “B” esterases and hepatic CYP450 isoenzimes in Senegalese sole for their further application in monitoring studies
Keywords: کولین استراز; Characterization; Cholinesterases; Carboxylesterases Solea senegalensis; CYPs; Fluorimetric substrates
Acute toxic effects of pyrene on Pomatoschistus microps (Teleostei, Gobiidae): Mortality, biomarkers and swimming performance
Keywords: کولین استراز; Polycyclic aromatic hydrocarbons; Pyrene; Common goby; Biomarkers; Behavior; Cholinesterases
Isatin-3-N4-benzilthiosemicarbazone, a non-toxic thiosemicarbazone derivative, protects and reactivates rat and human cholinesterases inhibited by methamidophos in vitro and in silico
Keywords: کولین استراز; Antioxidant; Cholinesterases; Molecular docking; Thiosemicarbazones; Methamidophos;
Synthesis and in vitro evaluation of 7-methoxy-N-(pent-4-enyl)-1,2,3,4-tetrahydroacridin-9-amine—new tacrine derivate with cholinergic properties
Keywords: کولین استراز; 7-Methoxytacrine; Cholinesterases; Alzheimer disease; Molecular modelling; Cholinesterase inhibitors