دانلود مقالات ISI درباره DIPEA، diisopropylethylamine + ترجمه فارسی

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Synthesis of brassinosteroids with a keto group in the side chain

Keywords: DIPEA، diisopropylethylamine; BS, brassinosteroids; TBAB, tetrabutylammonium bromide; DIPEA, diisopropylethylamine; DMP, Dess–Martin periodinaneBrassinosteroids; 24-Epibrassinolide; Boric acid ester; 24-Epicryptolide; 22-Dehydro-24-epibrassinolide

دانلود رایگان متن کامل مقاله ISI 6 صفحه سال انتشار : 2015 سفارش ترجمه

طراحی پروب های لانتانیدهای پاسخگو مبتنی بر واکنش پذیر برای تشخیص چند رنگ در سیستم های بیولوژیکی

Designing reactivity-based responsive lanthanide probes for multicolor detection in biological systems

Keywords: DIPEA، diisopropylethylamine; Asc, ascorbate; BINAP, 2,2′-bis(diphenylphosphino)-1,1′-binaphthyl; CuAAC, Cu-catalyzed azide-alkyne cycloaddition; DIPEA, diisopropylethylamine; DO3A, 1,4,7-tris(carboxymethylaza)cyclododecane-10-azaacetylamid; DOTA, 1,4,7,10-tetraazacyclododecane-1,4,7,

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2014 سفارش ترجمه

Discovery of 4-(4-aminopyrazolo[1,5-a][1,3,5]triazin-8-yl)benzamides as novel, highly potent and selective, orally bioavailable inhibitors of Tyrosine Threonine Kinase, TTK

Keywords: DIPEA، diisopropylethylamine; Ar, aryl; ATP, Adenosine-5′-triphosphate; AUC, area under the curve; BA, bioavailability; CYP, Cytochrome P450; DBU, 1,8-diazabicyclo[5.4.0]undec-7-ene; DCM, dichloromethane; DIPEA, diisopropylethylamine; Δ, heat; DME, 1,2-dimethoxyethane; DMF, N,N-dimeth

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and antibacterial evaluation of novel 4″-glycyl linked quinolyl-azithromycins with potent activity against macrolide-resistant pathogens

Keywords: DIPEA، diisopropylethylamine; MLSB, macrolide–lincosamide–streptogramin B antibiotics; HBTU, O-(benzotriazol-1-yl)-N,N,N′,N′-tetramethyluronium hexafluorophosphate; DIPEA, diisopropylethylamine; SAR, structure–activity relationshipsMacrolide antibiotics; C-4″-substituted azithromycins

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2016 سفارش ترجمه

Synthesis and evaluation of a ligand targeting the somatostatin-2 receptor for drug delivery to neuroendocrine cancers

Keywords: DIPEA، diisopropylethylamine; ATCC, American Type Culture Collection; CDI, N,N′-carbonyldiimidazole; Dde, 2-acetyldimedone; DIPEA, diisopropylethylamine; Dmab, 4-{N-[1-(4,4-dimethyl-2,6-dioxocyclohexylidene)-3-methyl-butyl]-amino}benzyl ester; DMF, dimethylformamide; DSC, N,N′-disucci

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2015 سفارش ترجمه

Using click chemistry toward novel 1,2,3-triazole-linked dopamine D3 receptor ligands

Keywords: DIPEA، diisopropylethylamine; CuAAC, copper-catalyzed azide-alkyne cycloaddition; DIPEA, diisopropylethylamine; D2R, dopamine D2 receptor; D3R, dopamine D3 receptor; GPCR, G protein-coupled receptors; SAR, structure–activity relationship; TBTA, tris(benzyltriazolylmethyl)amineDopamine

دانلود رایگان متن کامل مقاله ISI 13 صفحه سال انتشار : 2015 سفارش ترجمه

Synthesis and biochemical activities of antiproliferative amino acid and phosphate derivatives of microtubule-disrupting β-lactam combretastatins

Keywords: DIPEA، diisopropylethylamine; Antiproliferative; Beta-lactam; Combretastatin A-4; Prodrug; Solubility; TubulinCA-1, combretastatin A-1; CA-4, combretastatin A-4; DIPEA, diisopropylethylamine; MTT, 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; NAC, N-acetylcolchicine; P

دانلود رایگان متن کامل مقاله ISI 17 صفحه سال انتشار : 2013 سفارش ترجمه

Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors

Keywords: DIPEA، diisopropylethylamine; Synthesis; Quinolones; Cannabinoid ligands; Partial agonists; Peripheral ligandsBBB, blood–brain barrier; CB1, cannabinoid type-1; CB2, cannabinoid type-2; CHO, chinese hamster ovary cell; CNS, central nervous system; DIPEA, diisopropylethylamine; DME, 1,

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2012 سفارش ترجمه

Small molecule antagonists of the urokinase (uPA): urokinase receptor (uPAR) interaction with high reported potencies show only weak effects in cell-based competition assays employing the native uPAR ligand

Keywords: DIPEA، diisopropylethylamine; ATF, amino-terminal fragment of uPA; Boc, tert-butyloxycarbonyl; DCC, N,N′-dicyclohexylcarbodiimide; DIPEA, diisopropylethylamine; DMAP, 4-(N,N-dimethylamino)pyridine; EGF, epidermal growth factor; GPI, glycophosphatidylinositol; HBTU, O-benzotriazole-N,N

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2011 سفارش ترجمه

The effect of a bromide leaving group on the properties of nitro analogs of the duocarmycins as hypoxia-activated prodrugs and phosphate pre-prodrugs for antitumor therapy

Keywords: DIPEA، diisopropylethylamine; CBI, seco-1,2,9,9a-tetrahydrocyclopropa[c]benz[e]indol-4-one; DEI, 5-[(dimethylamino)ethoxy]indole; DIPEA, diisopropylethylamine; DMA, dimethylacetamide; EDCI·HBr, N-ethyl-N′-(3-dimethylaminopropyl)carbodiimide hydrobromide; EWG, electron-withdrawing grou

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2011 سفارش ترجمه

Isomalyngamide A, A-1 and their analogs suppress cancer cell migration in vitro

Keywords: DIPEA، diisopropylethylamine; Antimetastatic agents; Cancer cell migration; Integrin signaling; Isomalyngamide; Marine metabolites; Sialyltransferase inhibitorDCM, dichloromethane; DIPEA, diisopropylethylamine; DMAP, 4-(dimethylamino)pyridine; DMEM, Dulbecco’s modified Eagle’s medium;

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2011 سفارش ترجمه

Does the combination of optimal substitutions at the C2-, N5- and N8-positions of the pyrazolo-triazolo-pyrimidine scaffold guarantee selective modulation of the human A3 adenosine receptors?

Keywords: DIPEA، diisopropylethylamine; APCI, atmospheric pressure chemical ionization; ATP, adenosine triphosphate; cAMP, cyclic adenosine monophosphate; CHO cells, Chinese hamster ovary cells; DIPEA, diisopropylethylamine; EL, extracellular loop; EGTA, ethylene glycol tetraacetic acid; Gi, in

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2011 سفارش ترجمه

Novel powerful water-soluble lipid immunoadjuvants inducing mouse dendritic cell maturation and B cell proliferation using TLR2 pathway

Keywords: DIPEA، diisopropylethylamine; Boc, tertiobutyloxycarbonyl; BOP, (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; CD, cluster of differentiation; DC, dendritic cell; DCC, dicyclohexylcarbodiimide; DIPEA, diisopropylethylamine; DMAP, dimethylaminopyridine; LPS,

دانلود رایگان متن کامل مقاله ISI 4 صفحه سال انتشار : 2010 سفارش ترجمه

E-selectin binding peptide–polymer–drug conjugates and their selective cytotoxicity against vascular endothelial cells

Keywords: DIPEA، diisopropylethylamine; Drug delivery systems; HPMA copolymers; E-selectin binding peptide; Multivalent interactions; Tumor vascular endothelium Polymer drug conjugatesAIBN, 2,2′-azobis(isobutyronitrile); CRD, carbohydrate recognition domain; DIPEA, diisopropylethylamine; DMF, d

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2009 سفارش ترجمه

NMR based structure–activity relationship analysis of an antimicrobial peptide, thanatin, engineered by site-specific chemical modification: Activity improvement and spectrum alteration

Keywords: DIPEA، diisopropylethylamine; ACN, acetonitrile; DIPEA, diisopropylethylamine; DMF, N,N-dimethylformamide; Fmoc, 9-fluorenylmethoxycarbonyl; HOBt, N-hydroxybenzotriazole; HPLC, high performance liquid chromatography; MALDI, matrix-assisted laser desorption/ionization; MIC, minimal inh

دانلود رایگان متن کامل مقاله ISI 7 صفحه سال انتشار : 2008 سفارش ترجمه

High-throughput evaluation of relative cell permeability between peptoids and peptides

Keywords: DIPEA، diisopropylethylamine; AEEA, acetyl-ethyleneglycol-ethyl-amine; BBB, blood–brain barrier; DBD, DNA-binding domain; Dex, dexamethasone; DIC, diisopropylcarbodiimide; DIPEA, diisopropylethylamine; EC50, half-maximal effective concentration; Fmoc, fluorenyl-methoxy-carbonyl; GR, g

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2008 سفارش ترجمه

The mechanism of oleic acid nitration by •NO2

Keywords: DIPEA، diisopropylethylamine; BSTFA, N,O-bis(trimethylsilyl)-trifluoroacetamide; DIPEA, diisopropylethylamine; EA, elaidic acid; IOX, isoxazole; GC/MS, gas chromatography mass spectrometry; LC/MS, liquid chromatography mass spectrometry; MRM, multiple reaction monitoring LC/MS; NO2FA,

دانلود رایگان متن کامل مقاله ISI 15 صفحه سال انتشار : 2008 سفارش ترجمه

Synthesis and biological evaluation of cyclic and branched peptide analogues as ligands for cholecystokinin type 1 receptor

Keywords: DIPEA، diisopropylethylamine; Boc, tert-butoxycarbonyl; DBU, (1,8-diazabicyclo[5.4.0]undec-7-ene); DIPEA, diisopropylethylamine; DMF, N,N-dimethylformamide; DTPA-Glu, N,N-bis[2-[bis(carboxyethyl)amino]-ethyl]-l-glutamic acid; EDT, 1,2-ethanedithiol; Fmoc, 9-fluorenylmethoxycarbonyl; H

دانلود رایگان متن کامل مقاله ISI 9 صفحه سال انتشار : 2007 سفارش ترجمه

Mapping Putative Contact Sites Between Subunits in a Bacterial ATP-binding Cassette (ABC) Transporter by Synthetic Peptide Libraries

Keywords: DIPEA، diisopropylethylamine; ABC, ATP-binding cassette; CAPE, cellulose-amino-hydroxypropyl ether; DIPEA, diisopropylethylamine; Fmoc-, 9-fluorenyl methoxy carbonyl-; RP-HPLC, reverse phase high pressure liquid chromatography; MALDI-TOF, matrix-assisted laser desorption ionisation-ti

دانلود رایگان متن کامل مقاله ISI 14 صفحه سال انتشار : 2007 سفارش ترجمه

Synthesis and evaluation of 3-aminopropionyl substituted fentanyl analogues for opioid activity

Keywords: DIPEA، diisopropylethylamine; Ac, acetyl; Ac2O, acetic anhydride; Boc, tert-butyloxycarbonyl; DCC, N,N-dicyclohexylcarbodiimide; DCM, dichloromethane; DCU, N,N-dicyclohexylurea; DEPT, decoupled edited phase transfer; DIPEA, diisopropylethylamine; DMF, N,N-dimethylformamide; DMSO, dime

دانلود رایگان متن کامل مقاله ISI 5 صفحه سال انتشار : 2006 سفارش ترجمه

Convenient synthesis of a sialylglycopeptide-thioester having an intact and homogeneous complex-type disialyl-oligosaccharide

Keywords: DIPEA، diisopropylethylamine; DEPBT, 3-(diethoxyphosphoryloxy)-1,2,3-benzotriazin-4(3H)-one; DIPCI, N,N′-diisopropylcarbodiimide; DIPEA, diisopropylethylamine; HBTU, 2-(1H-benzotriazole-1-yl)-1,1,3,3-tetramethyluronium hexafluorophosphate; HMPA, 4-hydroxymethylphenoxyacetic acid; HMPB

دانلود رایگان متن کامل مقاله ISI 8 صفحه سال انتشار : 2006 سفارش ترجمه

New highly potent GABA uptake inhibitors selective for GAT-1 and GAT-3 derived from (R)- and (S)-proline and homologous pyrrolidine-2-alkanoic acids

Keywords: DIPEA، diisopropylethylamine; GABA uptake inhibitors; antiepileptic; GAT-1; GAT-3; pyrrolidinesDBU, 1,8-diazabicyclo[5.4.0]un-7-decene; CC, column chromatography; DIBAH, diisobutylaluminiumhydride; DIPEA, diisopropylethylamine; DMF, N,N-dimethylformamide; DMSO, dimethylsulfoxide; GP,

دانلود رایگان متن کامل مقاله ISI 16 صفحه سال انتشار : 2006 سفارش ترجمه

A cyclic PNA-based compound targeting domain IV of HCV IRES RNA inhibits in vitro IRES-dependent translation

Keywords: DIPEA، diisopropylethylamine; Alloc, allyloxycarbonyl; Boc, tert-butyloxycarbonyl; DIPEA, diisopropylethylamine; DMF, dimethylformamide; HATU, O-(7-aza-1-benzotriazolyl)-N,N,N′,N′-tetramethyluronium hexa-fluorophosphate; HOAt, 1-hydroxy-7-azabenzotriazole; Mmt, monomethoxytrityl; PyBo

دانلود رایگان متن کامل مقاله ISI 10 صفحه سال انتشار : 2005 سفارش ترجمه