Keywords: متابولیسم درون بدن; Itraconazole; In vitro metabolism; Metabolomics; Liquid chromatography-mass spectrometry;
مقالات ISI متابولیسم درون بدن (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: متابولیسم درون بدن; Enzymatic kinetics; In vitro metabolism; Microsomes; Sigmoidal profile; Piplartine
Keywords: متابولیسم درون بدن; Pesticides; Toxicokinetics; P450; In vitro metabolism; Risk assessment;
Keywords: متابولیسم درون بدن; MS-supported automated method development; In vitro metabolism; Cocktail approach; UHPLC-MS; UHPSFC-MS; Compact single quadrupole;
Elucidation of pharmacokinetics of novel DNA ligase I inhibitor, S012-1332 in rats: Integration of in vitro and in vivo findings
Keywords: متابولیسم درون بدن; S012-1332; LC-ESI-MS/MS; Preclinical pharmacokinetics; Plasma protein binding; In vitro metabolism;
Suspect and untargeted screening of bisphenol S metabolites produced by in vitro human liver metabolism
Keywords: متابولیسم درون بدن; Bisphenol S; In vitro metabolism; Human liver microsomes; High-resolution mass spectrometry; MZmine; Emerging contaminants;
GABAA receptor activity modulating piperine analogs: In vitro metabolic stability, metabolite identification, CYP450 reaction phenotyping, and protein binding
Keywords: متابولیسم درون بدن; au; arbitrary units; BBB; blood brain barrier; CNS; central nervous system; CYP450; cytochrome P450; DMSO; dimethyl sulfoxide; ESI; electrospray ionization; GABAA; γ- aminobutyric acid type A receptor; HPLC; high performance liquid chromatography; HR; hi
Insight into stereoselective disposition of enantiomers of a potent antithrombotic agent, S002-333 following administration of the racemic compound to mice
Keywords: متابولیسم درون بدن; S002-333; Stereoselective pharmacokinetics; Tissue distribution; Plasma protein binding; In vitro metabolism; Enantiomer-enantiomer interaction;
Characterization of oxycodone in vitro metabolism by human cytochromes P450 and UDP-glucuronosyltransferases
Keywords: متابولیسم درون بدن; Oxycodone; Cytochromes P450; UDP-glucuronosyltransferases; In vitro metabolism;
Characterization of the phase I and phase II metabolic profile of tolvaptan by in vitro studies and liquid chromatography-mass spectrometry profiling: Relevance to doping control analysis
Keywords: متابولیسم درون بدن; Tolvaptan; In vitro metabolism; LC-MS/(MS); Anti-Doping analysis; Drug-drug interactions; Azole antifungals;
In vitro metabolism of a novel synthetic cannabinoid, EAM-2201, in human liver microsomes and human recombinant cytochrome P450s
Keywords: متابولیسم درون بدن; EAM-2201; Synthetic cannabinoid; In vitro metabolism; LC–HRMS; Human liver microsomes; Cytochrome P450
Identification of in vitro metabolites of ethylphenidate by liquid chromatography coupled to quadrupole time-of-flight mass spectrometry
Keywords: متابولیسم درون بدن; Ethylphenidate; High-resolution mass spectrometry; In vitro metabolism; Methylphenidate; New psychoactive substances;
Mitochondrial toxicity of selective COX-2 inhibitors via inhibition of oxidative phosphorylation (ATP synthesis) in rat liver mitochondria
Keywords: متابولیسم درون بدن; Drug induced liver injury; Selective COX-2 inhibitors; Rat liver mitochondria; Oxidative phosphorylation; ATP; In vitro metabolism;
JWH-018 Ï-OH, a shared hydroxy metabolite of the two synthetic cannabinoids JWH-018 and AM-2201, undergoes oxidation by alcohol dehydrogenase and aldehyde dehydrogenase enzymes in vitro forming the carboxylic acid metabolite
Keywords: متابولیسم درون بدن; ADH; alcohol dehydrogenase; ALDH; aldehyde dehydrogenase; AO; aldehyde oxidase; Clint.micr; microsomal intrinsic clearance; CYP; cytochrome P450; EIC; extracted ion chromatogram; EMCDDA; European Monitoring Centre for Drugs and Drug Addiction; ESI; electr
Comprehensive characterization of the in vitro and in vivo metabolites of ziyuglycoside I in rat microsome, intestinal flora, excretion specimen and fresh tissues based on LC-Q-TOF/MS
Keywords: متابولیسم درون بدن; Ziyuglycoside I; LC-Q-TOF/MS; In vivo metabolism; In vitro metabolism; Ziyuglycoside II;
In-line coupling of an achiral-chiral column to investigate the enantioselective in vitro metabolism of the pesticide Fenamiphos by human liver microsomes
Keywords: متابولیسم درون بدن; Pesticide; Chiral analysis; In vitro metabolism; Human liver microsomes; Metabolites; Predicted toxicokinetic parameters;
Pharmacokinetic properties, in vitro metabolism and plasma protein binding of govaniadine an alkaloid isolated from Corydalis govaniana Wall
Keywords: متابولیسم درون بدن; Govaniadine; in vitro metabolism; Pharmacokinetics; Two-compartment model;
In vitro metabolism of rebaudioside E under anaerobic conditions: Comparison with rebaudioside A
Keywords: متابولیسم درون بدن; LLOQ; lower limit of quantitation; Rebaudiosides; Steviol; Stevia extract; Stevia leaf extract; Purified stevia leaf extract; In vitro metabolism; Human;
Evaluation of simple in vitro to in vivo extrapolation approaches for environmental compounds
Keywords: متابولیسم درون بدن; IVIVE; In vitro metabolism; Reverse dosimetry; Css;
6:2 Fluorotelomer iodide in vitro metabolism by rat liver microsomes: Comparison with [1,2-14C] 6:2 fluorotelomer alcohol
Keywords: متابولیسم درون بدن; 6:2 Fluorotelomer iodide (6:2 FTI); 6:2 Fluorotelomer alcohol (6:2 FTOH); 5:3 Acid; Perfluorocarboxylic acids (PFCAs); In vitro metabolism; Rat liver microsomes;
Determination of major metabolites of MAM-2201 and JWH-122 in in vitro and in vivo studies to distinguish their intake
Keywords: متابولیسم درون بدن; Synthetic cannabinoid; JWH-122; MAM-2201; In vitro metabolism; Urine;
A non-michaelian behavior of the in vitro metabolism of the pentacyclic triterpene alfa and beta amyrins by employing rat liver microsomes
Keywords: متابولیسم درون بدن; Amyrins; Atypical enzymatic kinetics; In vitro metabolism; Hill profile; Natural product;
In vitro metabolism study of the promising anticancer agent the lignan (−)-grandisin
Keywords: متابولیسم درون بدن; Grandisin; In vitro metabolism; Method validation; CYP450; Rat liver microsomes; Dihydro-grandisin metabolite
In vitro metabolism of di(2-ethylhexyl) phthalate (DEHP) by various tissues and cytochrome P450s of human and rat
Keywords: متابولیسم درون بدن; DEHP; In vitro metabolism; Human tissues; Rat tissues; Cytochrome P450; LC-MS/MS;
Investigation of piceid metabolites in rat by liquid chromatography tandem mass spectrometry
Keywords: متابولیسم درون بدن; Piceid; HPLC-MS-MS; In vitro metabolism; Urinary metabolite;
Drug metabolism of CYP3A4, CYP2C9 and CYP2D6 substrates in pigs and humans
Keywords: متابولیسم درون بدن; Verapamil; Testosterone; Pig pharmacokinetics; Dextromethorphan; In vitro metabolism; Pig mRNA expressisonPK, pharmacokinetics; CD, candidate drug; CYP, cytochrome P450; VER, verapamil; NOR, norverapamil; BDDCS, Biopharmaceutic drug disposition classifica
Stereoselective determination of drugs and metabolites in body fluids, tissues and microsomal preparations by capillary electrophoresis (2000–2010)
Keywords: متابولیسم درون بدن; Capillary electrophoresis; Enantiomers; Chirality; Drugs; Body fluids; Stereoselective metabolism; Pharmacokinetics; In vitro metabolism
In vitro liver metabolism of aclidinium bromide in preclinical animal species and humans: Identification of the human enzymes involved in its oxidative metabolism
Keywords: متابولیسم درون بدن; AB; aclidinium bromide; BChE; butyrylcholinesterase; CID; collision-induced dissociation; P450; cytochrome P450; ESI; electrospray ionization; FMO; flavin-containing monooxigenases; glyc; glycolyl; Kh; hydrolysis rate constant; LC; liquid chromatography;
Metabolism of carbosulfan II. Human interindividual variability in its in vitro hepatic biotransformation and the identification of the cytochrome P450 isoforms involved
Keywords: متابولیسم درون بدن; Pesticides; Xenobiotic; Risk assessment; In vitro metabolism; P450; LC–MS
In vitro metabolism study of a new nitrosyl ruthenium complex [Ru(NH·NHq)(terpy)NO]3+ nitric oxide donor using rat microsomes
Keywords: متابولیسم درون بدن; In vitro metabolism; Nitric oxide; Nitrosyl ruthenium complex;
Inhibition of acetylcholinesterase by metabolites of copper pyrithione (CuPT) and its possible involvement in vertebral deformity of a CuPT-exposed marine teleostean fish
Keywords: متابولیسم درون بدن; 2,2′-dipyridyldisulfide; 2,2′-dithiobispyridine-N-oxide; Antifouling biocide; Fundulus heteroclitus; In vitro metabolism; Liver microsomes; Thin-layer chromatography
In vitro hepatic metabolism of 2,2′,4,4′,5-pentabromodiphenyl ether (BDE 99) in Chinook Salmon (Onchorhynchus tshawytscha)
Keywords: متابولیسم درون بدن; NOAA, National Oceanographic and Atmospheric Administration; GST, glutathione S-transferase; CYP, cytochrome P450; PBDE, polybrominated diphenyl etherChinook salmon; Polybrominated diphenyl ethers; In vitro metabolism
The role of diet in the metabolism of daidzein by human faecal microbiota sampled from Italian volunteers
Keywords: متابولیسم درون بدن; Daidzein; Diet; Equol; Human; In vitro metabolism; LC-MS
In vitro studies on the metabolism of trabectedin (YONDELIS®) in monkey and man, including human CYP reaction phenotyping
Keywords: متابولیسم درون بدن; Trabectedin; In vitro metabolism; Human; Monkey; CYP reaction phenotyping
Safety evaluation to support First-In-Man investigations I: Kinetic and safety pharmacology studies
Keywords: متابولیسم درون بدن; In vitro metabolism; CYP enzyme; Pharmacokinetics; Mass balance; Toxicokinetics; hERG assay; Anaesthetised animal; Telemetry animal; QT prolongation
Biotransformation of bisphenol F by human and rat liver subcellular fractions
Keywords: متابولیسم درون بدن; Bisphenol F; In vitro metabolism; Endocrine disrupter
Characterization of the in vitro metabolic profile of amlodipine in rat using liquid chromatography–mass spectrometry
Keywords: متابولیسم درون بدن; In vitro metabolism; Amlodipine; LC/MS; LC–MS/MS; Rat hepatocyte; Accurate mass measurement
An in vitro study on metabolism of 17β-boldenone and boldione using cattle liver and kidney subcellular fractions
Keywords: متابولیسم درون بدن; 17β-Boldenone; Boldione; In vitro metabolism; Cattle; Liver; Kidney; High performance liquid chromatography; Liquid chromatography tandem mass spectrometry
In vitro metabolism of BYZX in human liver microsomes and the structural elucidation of metabolite by liquid chromatography–mass spectrometry method
Keywords: متابولیسم درون بدن; BYZX; In vitro metabolism; HPLC–MS-MS; Human liver microsomes (HLM)
Microbial metabolism of caffeic acid and its esters chlorogenic and caftaric acids by human faecal microbiota in vitro
Keywords: متابولیسم درون بدن; Polyphenols; Caffeic acid; Chlorogenic acid; Caftaric acid; Faecal microbiota; In vitro metabolism
Cobalamin as an analytical tool for analysis of oxirane metabolites of 1,3-butadiene: Development and validation of the method
Keywords: متابولیسم درون بدن; Cobalamin; Diepoxybutane; Butadiene; In vitro metabolism
Species differences in metabolites of PET ligands: serotonergic 5-HT1A receptor antagonists 3-trans-FCWAY and 3-cis-FCWAY
Keywords: متابولیسم درون بدن; PET; 5-HT1A; FCWAY; In vitro metabolism
The tyrosine kinase inhibitor PD153035: implication of labeling position on radiometabolites formed in vitro
Keywords: متابولیسم درون بدن; Epidermal growth factor receptor; Tyrosine kinase inhibitor; In vitro metabolism; PD153035; Anilinoquinazoline; Positron emission tomography
Synthesis and evaluation of 4-[18F]fluorothalidomide for the in vivo studies of angiogenesis
Keywords: متابولیسم درون بدن; Angiogenesis; 4-[18F]Fluorothalidomide; HUVEC; PET; In vitro metabolism
Thiodiglycol, the hydrolysis product of sulfur mustard: Analysis of in vitro biotransformation by mammalian alcohol dehydrogenases using nuclear magnetic resonance
Keywords: متابولیسم درون بدن; Sulfur mustard; Thiodiglycol; In vitro metabolism; Alcohol dehydrogenase; NMR;
Enantioselective analysis of the metabolites of hydroxychloroquine and application to an in vitro metabolic study
Keywords: متابولیسم درون بدن; Hydroxychloroquine; Desethylchloroquine; Desethylhydroxychloroquine; Enantioselective separation; In vitro metabolism;
A novel incubation direct injection LC/MS/MS technique for in vitro drug metabolism screening studies involving the CYP 2D6 and the CYP 3A4 isozymes
Keywords: متابولیسم درون بدن; LC/MS/MS; In vitro metabolism; Dextromethorphan; CYP 3A4;
Repeated Glucuronidation at One Hydroxyl Group Leads to Structurally Novel Diglucuronides of Steroid Sex Hormones
Keywords: متابولیسم درون بدن; liver microsomes; in vitro metabolism; diglucuronide; UGT; steroid hormone; species differences;
In vitro metabolic fate of a novel structural class: Evidence for the formation of a reactive intermediate on a benzothiophene moiety
Keywords: متابولیسم درون بدن; In vitro metabolism; Hepatocytes; Arene oxide; Exact-mass mass spectrometry;