مهار ثابت

در این صفحه تعداد 131 مقاله تخصصی درباره مهار ثابت که در نشریه های معتبر علمی و پایگاه ساینس دایرکت (Science Direct) منتشر شده، نمایش داده شده است. برخی از این مقالات، پیش تر به زبان فارسی ترجمه شده اند که با مراجعه به هر یک از آنها، می توانید متن کامل مقاله انگلیسی همراه با ترجمه فارسی آن را دریافت فرمایید.
در صورتی که مقاله مورد نظر شما هنوز به فارسی ترجمه نشده باشد، مترجمان با تجربه ما آمادگی دارند آن را در اسرع وقت برای شما ترجمه نمایند.
مقالات ISI مهار ثابت (ترجمه نشده)
مقالات زیر هنوز به فارسی ترجمه نشده اند.
در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
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Keywords: مهار ثابت; THR; Thrombin; EC; Epicatechin; EGC; Epigallocatechin; ECG; Epicatechin gallate; EGCG; Epigallocatechin gallate; CE; Capillary electrophoresis; EMMA; Electrophoretically mediated microanalysis; IMER; Immobilized enzyme microreaction; pNA; para-nitroanilin
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Keywords: مهار ثابت; Phosphodiesterase-6; Inhibitor; Inhibition constant; Retina; Photoreceptors; Ex vivo electroretinography; A; activation coefficient; cAMP; adenosine 3′,5′ cyclic monophosphate; cGMP; guanosine 3′,5′ cyclic monophosphate; CNG channel; cyclic nucleo
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Keywords: مهار ثابت; AD; Alzheimer's disease; DA; dopamine; DAergic; dopaminergic; hMAO-A; human monoamine oxidase A; hMAO-B; human monoamine oxidase B; HRP; horseradish peroxidase; IC50; the half maximal inhibitory concentration; i.p.; intraperitoneal; Ki; inhibition const
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Keywords: مهار ثابت; ADAM; advanced dissolution, absorption, and metabolism; AED; antiepileptic drug; AUC; area-under-the-curve; B/P; blood to plasma ratio; BID; twice daily; BMI; body mass index; CBZ; carbamazepine; CLint; intrinsic clearance; CLR; renal clearance; CL; clear
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Keywords: مهار ثابت; Dissociation constant; Inhibition constant; Affinity; Nonspecific binding; Nontarget site binding; Adsorption; Ki; enzyme inhibition constant; AChE; acetylcholinesterase; eeAChE; Electrophorus electricus AChE; ATCh; acetylthiocholine chloride; bis(7)-tacr
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Keywords: مهار ثابت; Scorpion; Venom; Neurotoxin; Neuropeptide; Ion channels; AC50; toxin concentration for activation to 50%; Cav; voltage-gated calcium channel; EC50; half maximal effective concentration; ED50; median effective dose; ER; endoplasmic reticulum; IC50; half ma
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Keywords: مهار ثابت; AnPRT; anthranilate phosphoribosyltransferase; IC50; absolute IC50, that is the concentration of inhibitor which decreased enzyme activity by 50%; Km; Michaelis-Menten constant; Ki; inhibition constant; Mtb; Mycobacterium tuberculosis; PPi; pyrophosphate;
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Keywords: مهار ثابت; Carbonic anhydrase inhibitors; Isoforms I, II, IV, IX; Benzenesulfonamide; 1,2,3-Triazole; CA; Carbonic anhydrase; hCA; human carbonic anhydrase; CAIs; Carbonic anhydrase inhibitors; AAZ; Acetazolamide; Ki; Inhibition constant; nM; nanomolar; μM; micromo
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Keywords: مهار ثابت; AChR; nicotinic acetylcholine receptor; ACh; acetylcholine; TCAs; tricyclic antidepressants; α-BTx; α-bungarotoxin; MLA; methyllycaconitine; RT; room temperature; IC50; ligand concentration that produces 50% inhibition (of binding or of agonist activati
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Keywords: مهار ثابت; SBC; Apoptosis; Docking; ADME; Stomach cancer cell line (AGS); Anti-proliferative; MTT; 3-(4,5-dimethylthiazol-2-yl)-2,5-diphenyl tetrazolium bromide; ADME; absorption, distribution, metabolism and excretion; FBS; fetal bovine serum; RPMI; rosewell park m
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Keywords: مهار ثابت; GPCR; G protein-coupled receptor; EP4; prostaglandin E2 receptor EP4 subtype; LPAR; lysophosphatidic acid receptor; DTI; drug-target interaction; ADE; adverse drug event; MoA; mechanism of action; Ki; inhibition constant; Kd; dissociation constant; IC50;
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Keywords: مهار ثابت; A2aR; adenosine A2a receptor; CAF; cancer-associated fibroblast; CHO; Chinese hamster ovary; IC50; concentration of compound that displaces the binding of radioligand by 50%; Kb; binding constant; Ki; inhibition constant; NECA; 5″-N-ethylcarboxamidoaden
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Keywords: مهار ثابت; AUC; area under the curve; DDI; drug-drug interaction; fu; fraction unbound; IC50; inhibition constant; IV; intravenous; IVIVE; in vitro/in vivo extrapolation; Ki; inhibition constant; OAT; organic anion transporter; PBPK; physiologically based pharmacoki
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Keywords: مهار ثابت; drug interaction; cytochrome P450s; membrane transport/transporters; regulatory; guidance/guideline; ADME; absorption, distribution, metabolism and excretion; BCRP; breast cancer resistance protein; CYP; cytochrome P-450; d; induction calibration factor;
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Keywords: مهار ثابت; PTP1B; protein tyrosine phosphatase 1B; IC50; the inhibitor concentration leading 50% activity loss; Ki; inhibition constant; Kiapp; apparent Ki; Vmax; maximum velocity; Km; Michaelis-Menten constant; Kobs; apparent first-order rate constant for the trans
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Keywords: مهار ثابت; clinical trial simulations; drug interactions; pharmacokinetics; physiologically based pharmacokinetic modeling; organic anion-transporting polypeptide transporters; CYP enzymes; AUC; area under the blood concentration-time curve; AUCR; area under the b
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Keywords: مهار ثابت; AChR; nicotinic acetylcholine receptor; ACh; acetylcholine; NCA; noncompetitive antagonist; RT; room temperature; MHb; medial habenula; VI; ventral inferior; Ki; inhibition constant; Kd; dissociation constant; IC50; ligand concentration that produces 50%
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Keywords: مهار ثابت; drug transport; drug interactions; organic anion-transporting polypeptide transporters; hepatocytes; hepatic transport; pharmacokinetics; physiologically based pharmacokinetic modeling; AUC; area under the plasma concentration-time curve; CsA; cyclosporin
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Keywords: مهار ثابت; cytochrome P450; drug interaction; hepatic clearance; mathematical model; organic anion-transporting polypeptide transporters; pharmacokinetics; AUC; area under the plasma concentration-time curve; CL; clearance; CLint,all; overall hepatic intrinsic cle
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Keywords: مهار ثابت; Human α4β2 nicotinic acetylcholine receptor; Bupropion; (±)-SADU-3-72; Molecular docking; Luminal and non-luminal sites; Ca2+ influx; AChR; nicotinic acetylcholine receptor; NCA; noncompetitive antagonist; (±)-BP; (±)-bupropion [(±)-2-(tert-butylami
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Keywords: مهار ثابت; 5-HT; 5-hydroxytryptamine (serotonin); m5-HT3AR; murine serotonin type 3A receptor; AChR; nicotinic acetylcholine receptor; ACh; acetylcholine; NMDAR; N-methyl-D-aspartate receptor; AMPAR; α-amino-3-hydroxy-5-methyl-4-isoxazolepropionic acid receptor; NI
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Keywords: مهار ثابت; COX-2; Cyclooxygenase 2; E2; Estradiol; ERα, ERβ; estrogen receptor alpha and beta; ERE; estrogen responsive element; GC; granulosa cells; 5-HT; Serotonin; 5-HT1-7; Serotonin receptors 1-7; IC50; median inhibitory concentration; Ki; Inhibition constant;
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Keywords: مهار ثابت; CA; carbonic anhydrase; hCA; human carbonic anhydrase; Quinacrine; (RS)-N′-(6-Chloro-2-methoxy-acridin-9-yl)-N,N-diethylpentane-1,4-diamine; Proflavine; acridine-3,6-di-amine; Amsacrine; N-(4-(acridin-9-ylamino)-3-methoxyphenyl)methanesulfonamide; IR; i
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Keywords: مهار ثابت; Bmax; maximum density; 125I-BTX; 125I-α-bungarotoxin; Kd; dissociation constant; Ki; inhibition constant; NSB; non-specific binding; OD; optical density; PAM; positive allosteric modulator; SB; specific binding; TB; total binding; TE; tissue equivalent;
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Keywords: مهار ثابت; ADP; adenosine-diphosphate; ATP; adenosine triphosphate; GK; glucokinase; TlGK; glucokinase from Thermococcus litoralis; glucose-6-P; glucose-6-phosphate; KM; Michaelis constant; kcat; turnover rate; Ki; inhibition constant; Ka; activation constant; KD; d
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Keywords: مهار ثابت; Alpha-glucosidase; Glucose diffusion; Restructured pork; Inhibition mechanism; Hypoglycaemic effects; CVD; cardiovascular disease; CRP; control-RP; GOD; glucose oxidase; Ki; inhibition constant; Km; Michaelis-Menten constant; NRP; restructured pork cont
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Keywords: مهار ثابت; VKOR; vitamin K epoxide reductase; VKORC1; vitamin K epoxide reductase complex subunit 1; Vitamin K > O; vitamin K epoxide; Ferula communis L. (Apiaceae); Ferulenol; Ferprenin; VKORC1; Inhibition constant; Interspecies variability;
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Keywords: مهار ثابت; AChR; nicotinic acetylcholine receptor; NCA; noncompetitive antagonist; RT; room temperature; Ki; inhibition constant; Kd; dissociation constant; IC50; ligand concentration that produces 50% inhibition of binding (or of agonist activation); nH; Hill coeff
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Keywords: مهار ثابت; AChR; nicotinic acetylcholine receptor; (−)-lobeline (α-lobeline) (−); -2S, 6R, 8S-lobeline, Ct-AChBP, acetylcholine binding protein from Capitella teleta; Ac-AChBP; acetylcholine binding protein from Aplysia californica; CCh; carbamylcholine; RT; ro
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Keywords: مهار ثابت; BBI; Bowman-Birk inhibitor; CD; circular dichroism; DTT; dithiothreitol; RP-HPLC; reversed-phase high performance liquid chromatography; Ki; inhibition constant; MALDI-TOF; matrix assisted laser desorption ionisation time of flight mass spectrometry; PI
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Keywords: مهار ثابت; aa; amino acid; AMC; 7-amino 4-methyl coumarin; Amu; atomic mass unit; Au; arbitrary unit; Aufs; absorption units full scale; IMS; iso-coumarinyl methyl sulfone; Eda; enediyne amino acid; h; human; IC50; inhibitor concentration required for 50% inhibition
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Keywords: مهار ثابت; Cooperativity; Protein-ligand binding; Ligand binding affinity; Scoring functions; B-factor; Thrombin; Non-additivity; Me; methyl; Bn; benzyl; Boc; tert-butoxycarbonyl; ΔG˚; standard Gibbs free energy; Ki; inhibition constant; EDCI; 1-(3-dimethylaminopr
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Keywords: مهار ثابت; BAPNA; N-α-benzoyl-DL-arginine-p-nitroanilide; BBI; Bowman-Birk inhibitors; BBIC; Bowman-Birk inhibitor concentrate; BTEE; N-benzoyl-L-tyrosine ethyl ester; CIA; chymotrypsin inhibitor activity; CIU; chymotrypsin inhibitor units; CRC; colorectal cancer;
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Keywords: مهار ثابت; SARS-CoV; Severe Acute Respiratory Syndrome coronavirus; 3CLpro; 3 Chymotrypsin-like cysteine protease; MD; molecular dynamics; VS; virtual screening; CSM; computational solvent mapping; ROC; receiver operating characteristic; RMSD; root mean square devia
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Keywords: مهار ثابت; 5-HT; 5-hydroxy tryptamine (serotonin); 5-HTT; serotonin transporter; AAP; atypical antipsychotics; ACH; acetylcholine; ADR; adverse drug reaction; AP; antipsychotic; CDSR; cochrane database of systematic reviews; CTZ; chemotrigger zone; DAT; dopamine tra
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Keywords: مهار ثابت; P2X3 receptor; Desensitization; Mechanism of antagonism; Drug screening; Calcium imaging; αß-meATP; αß-methylene-ATP; CI; confidence interval; EC50; 50% effective concentration; IC50; 50% inhibitory concentration; Ki; inhibition constant; pA2; negativ
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Keywords: مهار ثابت; HQRJJHXKCFABSI-UONOGXRCSA-N; SAR; structure and activity relationship; NS2B-NS3; nonstructural protein 2B and 3; DENV; dengue virus; Ki; inhibition constant; TFA; trifluoroacetic acid; EtOAc; ethyl acetate; DCM; dichloromethylene; EtOH; ethyl alcohol; DMA
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Keywords: مهار ثابت; S. baicalensis; Scutellaria baicalensis; CYP; cytochrome P450; CYP2D; cytochrome P450 2D; CYP3A; cytochrome P450 3A; DXM; dextromethorphan; BG; baicalin; RLMs; rat liver microsomes; Km; substrate concentration at half-maximal product formation rate; Ki; i
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Keywords: مهار ثابت; Bioinsecticidal; Kunitz trypsin inhibitor; Insect pests; Piptadenia moniliformis; ED50; effective dose to inhibit 50% of an enzymatic pool; HPLC; high-performance liquid chromatography; TCA; trichloroacetic acid; Ki; inhibition constant; DTT; dithiothreit