Synthesis and evaluation of novel 1H-pyrrolo[2,3-b]pyridine-5-carboxamide derivatives as potent and orally efficacious immunomodulators targeting JAK3
Keywords: JAK (Janus kinase); JAK3 inhibitor; Immunomodulator; Transplant rejection; Docking calculation; hERG (human ether-a-go-go-related gene);