Keywords: کتوکونازول; Active freeze drying; Vacuum induce surface freezing; Drug nanocrystals; Nanosuspension; Ketoconazole; Wet media milling;
مقالات ISI کتوکونازول (ترجمه نشده)
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Keywords: کتوکونازول; HIV/aids; Dermatological conditions; Fixed-dose combination; Acyclovir; Ketoconazole; Transmucosal drug delivery; Stability; Labial mucosa; Vaginal mucosa;
Keywords: کتوکونازول; Cushing's syndrome; Cushing's disease; Ketoconazole; Metyrapone; Mitotane; Etomidate; Cabergoline; Pasireotide;
Keywords: کتوکونازول; Carbon paste electrode; Ketoconazole; AuNP; Voltammetric techniques;
Keywords: کتوکونازول; Microemulsion; Ketoconazole; Stability; Toxicity; Oral drug delivery;
Keywords: کتوکونازول; API; active pharmaceutical ingredient; BCS; biopharmaceutical classification system; Da; Dalton; DCS; developability classification system; DLS; dynamic light scattering; DMPEG; polyethylene glycol dimethyl ether; HPLC; high performance liquid chromatogra
Keywords: کتوکونازول; ACN; acetonitrile; API; active pharmaceutical ingredient; ASD; amorphous solid dispersion; BCS; biopharmaceutical classification system; CAP; cellulose acetate phthalate; DCM; dichloromethane; DMF; N,N-dimethylformamide; DL; drug load; DSC; differential s
Keywords: کتوکونازول; Fed state; Protein precipitation; Solid phase extraction; Biorelevantmedia; Drug analysis; Physicochemical properties; ÎCN; acetonitrile; API; active pharmaceutical ingredient; BA/BE; bioavailability/bioequivalence; CV; coefficient of variation; EtOH; et
Keywords: کتوکونازول; Silver; Ketoconazole; SERS; Computational;
Keywords: کتوکونازول; Itraconazole; Ketoconazole; Density functional theory; Infrared spectrum; Ultraviolet-visible spectrum; Natural bond orbital;
Keywords: کتوکونازول; Ketoconazole; Placenta; Estradiol-17β; Blood flow; Rat;
Keywords: کتوکونازول; Ketoconazole; Laccase; Enzymatic treatment; Biotransformation; Micro-toxicity;
Keywords: کتوکونازول; Ketoconazole; Hepatic injury; Oxidative stress; Apoptosis; Sesame Oil;
Keywords: کتوکونازول; Electron Paramagnetic Resonance; Electrochemistry; Drug Analysis; Graphite Electrode; Radicals; Ketoconazole
Keywords: کتوکونازول; Recurrent Ischemic Priapism; Stuttering Priapism; Ketoconazole; Sleep‐Related Erections; Priapism
Keywords: کتوکونازول; AhR; aryl hydrocarbon receptor; KET; ketoconazole; TCDD; 2,3,7,8-tetrachlorodibenzo-p-dioxin; Cytochrome P450; Drug-drug interactions; Dioxin receptor; Antifungal drugs;
Keywords: کتوکونازول; atopic dermatitis; contact dermatitis; eczema; fluconazole; head and neck dermatitis; itraconazole; ketoconazole; Malassezia; occupational dermatitis; seborrheic dermatitis; AD; atopic dermatitis; APT; atopy patch test; HND; head and neck dermatitis; SD;
Keywords: کتوکونازول; Cocrystal; Solubility; Ketoconazole
Keywords: کتوکونازول; Recurrent Ischemic Priapism; Stuttering Priapism; Ketoconazole; Sleep-Related Erections; Priapism; Induced Hypogonadal State and Recurrent Priapism
Keywords: کتوکونازول; Xanthine oxidase; Protein-drug interaction; Ketoconazole; Biosensor; Fluorescence;
Keywords: کتوکونازول; Hyperalgesia; Corticosterone; Microglia; IL-1β; Minocycline; Ketoconazole
Keywords: کتوکونازول; dipeptidyl peptidase-4 inhibitor; drug-drug interactions; ketoconazole; pharmacokinetics; teneligliptin;
Keywords: کتوکونازول; Midazolam; Raltegravir; Ketoconazole; Ritonavir; Rifampin;
Keywords: کتوکونازول; Ionic liquid; Ketoconazole; Solubility
Ascending Single-Dose Study of the Safety Profile, Tolerability, and Pharmacokinetics of Bosutinib Coadministered With Ketoconazole to Healthy Adult Subjects
Keywords: کتوکونازول; bosutinib; ketoconazole; pharmacokinetics; tyrosine kinase inhibitor;
Influence of proline and β-Cyclodextrin in ketoconazole physicochemical and microbiological performance
Keywords: کتوکونازول; Ketoconazole; Multicomponent complex; Solubility; Antifungal activity; Ketoconazole (PubChem CID: 47576); 46 β-cyclodextrin (PubChem CID: 444041); L-Proline (PubChem CID: 145742);
Design and synthesis of functionalized piperazin-1yl-(E)-stilbenes as inhibitors of 17α-hydroxylase-C17,20-lyase (Cyp17)
Keywords: کتوکونازول; Metabolic syndrome; Ketoconazole; Cortisol; 17αâHydroxylaseâC17,20âlyase (Cyp17);
Physiological based pharmacokinetic modeling to estimate in vivo Ki of ketoconazole on renal P-gp using human drug-drug interaction study result of fesoterodine and ketoconazole
Keywords: کتوکونازول; Physiological based pharmacokinetic model; P-gp; Renal excretion; Fesoterodine; Ketoconazole;
A Physiologically Based Pharmacokinetic Modeling Approach to Predict Drug-Drug Interactions of Buprenorphine After Subcutaneous Administration of CAM2038 With Perpetrators of CYP3A4
Keywords: کتوکونازول; buprenorphine; drug-drug interaction; physiologically based pharmacokinetics; ketoconazole; rifampin;
Study on adsorption behavior of ketoconazole on Q235 mild steel in 1.0â¯M HCl solution with electrochemical measurement
Keywords: کتوکونازول; Adsorption; Ketoconazole; Electrochemical noise;
W1038 near D-loop of NBD2 is a focal point for inter-domain communication in multidrug transporter Cdr1 of Candida albicans
Keywords: کتوکونازول; ABC; ATP-binding cassette; TMD; transmembrane domain; NBD; nucleotide binding domain; TMH; transmembrane helix; ICL; intracellular loop; Cdr1p; Candida drug resistance 1 protein; Pdr5p; pleiotropic drug resistance 5 protein; TAP; transporter associated wi
Exploring the feasibility of the use of biopolymers as a carrier in the formulation of amorphous solid dispersions - Part I: Gelatin
Keywords: کتوکونازول; Carbamazepine (2554); Cinnarizine (1547484); Darunavir (Ethanolate: 23725083); Fenofibrate (3339); Griseofulvin (441140); Indomethacin (3715); Itraconazole (55283); Ketoconazole (456201); Naproxen (156391); Nifedipine (4485); Ritonavir (392622); Diazepam
The Combination of GIS and Biphasic to Better Predict In Vivo Dissolution of BCS Class IIb Drugs, Ketoconazole and Raloxifene
Keywords: کتوکونازول; ASD; GIS; ketoconazole; raloxifene; BCS class II drug; simulation; in vivo performance;
In vitro ocular metabolism and bioactivation of ketoconazole in rat, rabbit and human
Keywords: کتوکونازول; Ocular metabolism; Ocular S9 fractions; Liver S9 fractions; Bioactivation; Potassium cyanide; [M+H]+; protonated molecular ion; KT; ketoconazole; RT; retention time; DAK; N-deacetylated ketoconazole; FMO; Flavin monooxygenase; LC; liquid chromatography; M
Processing of ketoconazole-4-aminobenzoic acid cocrystals using dense CO2 as an antisolvent
Keywords: کتوکونازول; Crystallization; Cocrystal; Ketoconazole; 4-amino benzoic acid; Gas;
Synergism between macrolide antibiotics and the azole fungicide ketoconazole in growth inhibition testing of the green alga Pseudokirchneriella subcapitata
Keywords: کتوکونازول; Azole fungicide; Clarithromycin; Erythromycin; Isobologram; Ketoconazole; Pseudokirchneriella subcapitata;
Metabolic-induced cytotoxicity of diosbulbin B in CYP3A4-expressing cells
Keywords: کتوکونازول; AP; Acetaminophen; CCK; 2H-Tetrazolium,5-(2,4-disulfophenyl)-3-(2-methoxy-4-nitrophenyl)-2-(4-nitrophenyl)-,innersalt,sodium salt; CYP450; Cytochrome P450; DB; Diosbulbin B; DMEM; Dulbecco's Modified Eagle Medium; DMF; N,N-Dimethylformamide; DMSO; D
Development and optimization of ketoconazole loaded nano-transfersomal gel for vaginal delivery using Box-Behnken design: In vitro, ex vivo characterization and antimicrobial evaluation
Keywords: کتوکونازول; Ketoconazole; Transfersome; Nanogel; Permeation; Antimicrobial studies;
In-vitro efficacies of topical microemulsions of clotrimazole and ketoconazole; and in-vivo performance of clotrimazole microemulsion
Keywords: کتوکونازول; Antifungal; Microemulsion; Topical; Clotrimazole; Ketoconazole; Candidiasis;
Y-shaped methoxy poly (ethylene glycol)-block-poly (epsilon-caprolactone)-based micelles for skin delivery of ketoconazole: in vitro study and in vivo evaluation
Keywords: کتوکونازول; Skin delivery; Micelles; Antifungal agent; Ketoconazole;
Enhanced effect in combination of curcumin- and ketoconazole-loaded methoxy poly (ethylene glycol)-poly (ε-caprolactone) micelles
Keywords: کتوکونازول; Curcumin; Ketoconazole; Synergistic effect; Micelles; MPEG-PCL;
The impact of supersaturation level for oral absorption of BCS class IIb drugs, dipyridamole and ketoconazole, using in vivo predictive dissolution system: Gastrointestinal Simulator (GIS)
Keywords: کتوکونازول; GIS; Ketoconazole; Dipyridamole; BCS class IIb drug; Supersaturation; Precipitation; In vivo performance;
Challenges in assignment of allosteric effects in cytochrome P450-catalyzed substrate oxidations to structural dynamics in the hemoprotein architecture
Keywords: کتوکونازول; Cytochrome P450; Allosteric effects; Cooperativity; Key determinants; Molecular modeling; 1PB; 1-pyrenebutanol; 4MP; 4-methylpyrazole; 7BQ; 7-benzyloxyquinoline; 7EC; 7-ethoxycoumarin; 7EFC; 7-ethoxy-4-trifluoromethylcoumarin; 9AP; 9-aminophenanthrene; 9E
Plant phenolics and terpenoids as adjuvants of antibacterial and antifungal drugs
Keywords: کتوکونازول; Potentiation; Low molecular weight natural products; Combination, Antibacterial drugs; Antifungal drugs; ABC; ATP-Binding Cassette; AMPH; Amphotericin B; AMC; Amoxicillin/Clavulanic acid; AMP; ampicillin; CAZ; ceftazidine; CD; clerodane diterpene 16α-hyd
Novel ex vivo protocol using porcine vagina to assess drug permeation from mucoadhesive and colloidal pharmaceutical systems
Keywords: کتوکونازول; Hung vagina; Ketoconazole; Mucoadhesive systems; Nanoparticle; Permeation protocol; Porcine vaginal mucosa;
Evaluation of selected Indian medicinal plants for antagonistic potential against Malassezia spp. and the synergistic effect of embelin in combination with ketoconazole
Keywords: کتوکونازول; Malassezia spp.; Secreted lipase; Embelia ribes; Embelin; Ketoconazole; Synergism;
Regulation of hepatic abcb4 and cyp3a65 gene expression and multidrug/multixenobiotic resistance (MDR/MXR) functional activity in the model teleost, Danio rerio (zebrafish)
Keywords: کتوکونازول; ABC; ATP-binding cassette; CYP; cytochrome P450; KTC; ketoconazole; MDR/MXR; multidrug/multixenobiotic resistance; P-gp; P-glycoprotein; PCN; pregnenolone 16α-carbonitrile; PXR; pregnane X-receptor; ARmax; maximum accumulation rate; Cmax; maximum concent
Simulations of Cytochrome P450 3A4-Mediated Drug-Drug Interactions by Simple Two-Compartment Model-Assisted Static Method
Keywords: کتوکونازول; bioavailability; cytochrome P450; drug interaction; dynamic simulation; first pass metabolism; hepatic clearance; intestinal metabolism; pharmacokinetics; simulations; parallel tube model; Ae (Ae,oral); dose fractions of urinary excreted unchanged drug af
Human intestine and liver microsomal metabolic differences between C19-diester and monoester diterpenoid alkaloids from the roots of Aconitum carmichaelii Debx.
Keywords: کتوکونازول; AC; Aconitine; BAC; 14-Benzoylaconine or 8-O-deacetyl aconitine; BHA; 14-Benzoylhypaconine or 8-O-deacetyl hypaconitine; BMA; 14-Benzoylmesaconine or 8-O-deacetyl mesaconitine; CHAPS; 3-[(3-cholamidopropyl) dimethyl-ammonio]-1-propane sulfonate; CYP450s;
Design, synthesis, and evaluation of (2S,4R)-Ketoconazole sulfonamide analogs as potential treatments for Metabolic Syndrome
Keywords: کتوکونازول; Metabolic Syndrome; Ketoconazole; Cortisol; 17αâHydroxylaseâC17,20âlyase (Cyp17);