Keywords: تست کیناز; Antipsychotic drugs; Phosphoinositide 3-kinase delta; Mechanism of action; Kinase assay; Schizophrenia;
مقالات ISI تست کیناز (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: تست کیناز; Protein kinase activity; Chemosensor; Kinase assay; Microfluidic device;
Characterization of PKACα enzyme kinetics and inhibition in an HPLC assay with a chromophoric substrate
Keywords: تست کیناز; Kinase assay; cAMP-dependent protein kinase; Kinetics assay; Inhibition assay; HPLC; Chromophore;
Pervanadate induces Mammalian Ste20 Kinase 3 (MST3) tyrosine phosphorylation but not activation
Keywords: تست کیناز; Cys; cysteine; DMEM; Dulbecco's modified Eagle's medium; EGFR; epidermal growth factor receptor; GPCR; G protein-coupled receptor; HEK 293; human embryonic kidney 293; HPK1; hematopoietic progenitor kinase 1; MST; mammalian Ste20 kinase; MAP4K; MAP kinase
Design, synthesis and biological evaluation of 5-amino-4-(1H-benzoimidazol-2-yl)-phenyl-1,2-dihydro-pyrrol-3-ones as inhibitors of protein kinase FGFR1
Keywords: تست کیناز; Protein kinase FGFR1; Inhibitor; 5-Amino-4-(1H-benzoimidazol-2-yl)-phenyl-1,2-dihydro-pyrrol-3-ones; Virtual screening; Kinase assay
Functional analysis of anomeric sugar kinases
Keywords: تست کیناز; Sugar kinase; Galactokinase; Kinase assay
Bioluminescent kinase strips: A novel approach to targeted and flexible kinase inhibitor profiling
Keywords: تست کیناز; Kinase profiling; Bioluminescence; ADP detection; Selectivity profiles; Kinase assay; Kinase inhibitor; PTM; post-translational modification; FDA; U.S. Food and Drug Administration; BSA; bovine serum albumin; DMSO; dimethyl sulfoxide; TK; tyrosine kinase
Synthesis and biological evaluation of 5-(fluoro-substituted-6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)imidazoles as inhibitors of transforming growth factor-β type I receptor kinase
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay;
Identification of apoptosis signal-regulating kinase 1 (ASK1) inhibitors among the derivatives of benzothiazol-2-yl-3-hydroxy-5-phenyl-1,5-dihydro-pyrrol-2-one
Keywords: تست کیناز; ASK1; apoptosis signal-regulating kinase 1; MAPK; mitogen-activated protein kinase; ER; endoplasmic reticulum; TNF-α; tumor necrosis factor-alpha; AIP-1; ASK1-interacting protein 1; VEGF; vascular endothelial growth factor; Aβ; amyloid beta; CK2; protei
4-([1,2,4]Triazolo[1,5-a]pyridin-6-yl)-5(3)-(6-methylpyridin-2-yl)imidazole and -pyrazole derivatives as potent and selective inhibitors of transforming growth factor-β type I receptor kinase
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay; Cell-based luciferase reporter assay; Docking;
Leveraging text analytics in patent analysis to empower business decisions – A competitive differentiation of kinase assay technology platforms by I2E text mining software
Keywords: تست کیناز; Patent analysis; Drug discovery; Kinase assay; Text analytics; Mining software; Visualization software; Business decisions
Identification and in vitro evaluation of new leads as selective and competitive glycogen synthase kinase-3β inhibitors through ligand and structure based drug design
Keywords: تست کیناز; Structure based drug design (SBDD); Ligand based drug design (LBDD); Virtual screening; Glycogen synthase kinase-3β (GSK-3β); Cyclin dependent kinase 5/p25 (CDK5/p25); Kinase assay
Identification of a novel serum and glucocorticoid regulated kinase-1 (SGK1) ligand from virtual screening
Keywords: تست کیناز; SGK1; Foxo3a; Kinase assay; Docking; Structure-based virtual screening;
Synthesis and biological evaluation of 2-benzylamino-4(5)-(6-methylpyridin-2-yl)-5(4)-([1,2,4]triazolo[1,5-a]-pyridin-6-yl)thiazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay; Cell-based luciferase reporter assay; Docking;
Synthesis and biological evaluation of 1-substituted-3-(6-methylpyridin-2-yl)-4-([1,2,4]triazolo[1,5-a]pyridin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay; Cell-based luciferase reporter assay
A homogeneous and nonisotopic assay for phosphatidylinositol 4-kinases
Keywords: تست کیناز; Phosphoinositides; Phosphatidylinositol 4-kinase; Kinase assay; High-throughput screening assays;
Bacterial expression and purification of active hematopoietic cell kinase
Keywords: تست کیناز; Src-family kinase; Hematopoietic cell kinase; Bacterial expression; Kinase assay; Enzyme inhibition;
Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinolin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay; Cell-based luciferase reporter assay
Synthesis and biological evaluation of 1-substituted-3(5)-(6-methylpyridin-2-yl)-4-(quinoxalin-6-yl)pyrazoles as transforming growth factor-β type 1 receptor kinase inhibitors
Keywords: تست کیناز; TGF-β; ALK5 inhibitor; Fibrosis; Cancer; Kinase assay; Cell-based luciferase reporter assay; Docking
Development of a high-throughput AlphaScreen assay measuring full-length LRRK2(G2019S) kinase activity using moesin protein substrate
Keywords: تست کیناز; LRRK2; AlphaScreen; Luminescent oxygen channeling immunoassay; Kinase assay; High-throughput screening
Evaluating the utility of the HTRF® Transcreener™ ADP assay technology: A comparison with the standard HTRF assay technology
Keywords: تست کیناز; HTRF; Transcreener; ADP; Kinase assay; ATPase; Inhibitor
An intracellular conformational sensor assay for Abl T315I
Keywords: تست کیناز; Kinase conformational sensor; Biosensor; Bcr-Abl; Abl315I; Split luciferase; Kinase assay; HTS; CAP-SH3-SH2;
A solid-phase Bcr-Abl kinase assay in 96-well hydrogel plates
Keywords: تست کیناز; Kinase assay; Imatinib mesylate (IM); Peptide substrate; Protein tyrosine kinase
Activation of ROCK by RhoA is regulated by cell adhesion, shape, and cytoskeletal tension
Keywords: تست کیناز; Rho; ROCK; Kinase assay; Myosin phosphorylation; Cell shape; Focal adhesions; FAK; Hypertension
Serine 714 might be implicated in the regulation of the phosphorylation in other areas of mPer1 protein
Keywords: تست کیناز; Circadian clock; Casein kinase 1ε (CK1ε); Period 1 (per1); Phosphorylation; Pulse-chase; Kinase assay
Use of pseudosubstrate affinity to measure active protein kinase A
Keywords: تست کیناز; Protein kinase A; Kinase assay; Protein kinase inhibitor; H89
Time-resolved fluorescence resonance energy transfer kinase assays using physiological protein substrates: Applications of terbium–fluorescein and terbium–green fluorescent protein fluorescence resonance energy transfer pairs
Keywords: تست کیناز; Green fluorescent protein; Kinase assay; TR-FRET
Homogeneous time-resolved fluorescence and its applications for kinase assays in drug discovery
Keywords: تست کیناز; HTRF; Kinase assay; Kinetics; Inhibitor; Mechanism
Utilization of luminescent technology to develop a kinase assay: Cdk4 as a model system
Keywords: تست کیناز; Kinase assay; Cd4k; Luminescence; ATP depletion;
Novel C-Raf phosphorylation sites: serine 296 and 301 participate in Raf regulation
Keywords: تست کیناز; MS; mass spectrometry; RBD; Ras-binding domain; CRD; cysteine rich domain; NP-40; Nonidet P-40; LC; liquid chromatography; LC/MS-MS/MS; data-dependent tandem LC/MS; C-Raf kinase; Kinase assay; Phosphorylation; Mass spectrometry;
Assaying Bcr-Abl kinase activity and inhibition in whole cell extracts by phosphorylation of substrates immobilized on agarose beads
Keywords: تست کیناز; Bcr-Abl; Protein tyrosine kinase; Kinase assay; Imatinib mesylate;