Keywords: دامنه کیناز; aFAK; active FAK; AL; activation loop; CL; catalytic loop; CMD; classical molecular dynamics; FAK; focal adhesion kinase; FAT; focal adhesion targeting domain; FERM; 4.1 ezrin radixin moesin; GL; glycine rich loop; H; helix; hFAK; hyperactive FAK; iFAK; i
مقالات ISI دامنه کیناز (ترجمه نشده)
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Keywords: دامنه کیناز; AS; activation segment; CS or C-spine; catalytic spine; CL; catalytic loop; CTT; carboxyterminal tail; D1; immunoglobulin-like domain-1; EGFR; epidermal growth factor receptor; GIST; gastrointestinal stromal tumors; GK; gatekeeper; GRL; Gly-rich loop; KD;
Structural characterization of recombinant human fibroblast growth factor receptor 2b kinase domain upon interaction with omega fatty acids
Keywords: دامنه کیناز; hFGFR2b; human fibroblast growth factor receptor 2b; UFAs; unsaturated fatty acids; CD; circular dichroism; FGFRs; fibroblast growth factor receptors; RTK; receptor tyrosine kinase; Ig; immunoglobulin; PLCγ; phospholipase Cγ; FRS2; fibroblast growth fac
Keywords: دامنه کیناز; ARMS; alveolar rhabdomyosarcoma; BSS; Beare Stevenson cutis gyrata syndrome; CFS; chromosomal fragile site; CC; coiled coil domain; EMS; 8p11 myeloproliferative syndrome (EMS); ERMS; embryonal rhabdomyosarcoma; FN; fibronectin domain; Ig; immunoglobulin-l
Keywords: دامنه کیناز; TRPM7; Breast cancer; Migration; Kinase domain;
Analysis of ABL kinase domain mutations as a probable cause of imatinib resistance in Chronic Myeloid Leukemia patients of Kashmir
Keywords: دامنه کیناز; Imatinib resistance; Fusion transcript; Kinase domain; cDNA; BCR-ABL; Complete cytogenetic response;
Identification of PKMYT1 inhibitors by screening the GSK published protein kinase inhibitor set I and II
Keywords: دامنه کیناز; Cdk1; Cyclin-dependent kinase 1; EFS; embryonal FYN-associated substrate; (6-FAM); 6-carboxyfluorescein; FL; full-length; FP; fluorescence polarization; FPIA; fluorescence polarization based immunoassay; KD; kinase domain; PKIS; protein kinase inhibitor s
Cloning, expression and purification of kinase domains of cacao PR-1 receptor-like kinases
Keywords: دامنه کیناز; Receptor-like protein kinase; Pathogenesis-related protein 1; Ligation-independent cloning; Protein expression; Cacao; DDM; dodecyl maltoside; FPR; frosty pod rot; HEPES; 4-(2-hydroxyethyl)-1-piperazineethanesulfonic acid; KD; kinase domain; LB; Lysogeny
Crystal structure of the kinase and UBA domains of SNRK reveals a distinct UBA binding mode in the AMPK family
Keywords: دامنه کیناز; SNRK; AMPK family; KD-UBA; Structural diversity; SNRK; sucrose non-fermenting (snf1)-related kinase; AMPK; AMP-activated protein kinase; BRSK; brain-specific kinase; MARK; microtubule affinity regulating kinase; SIK; salt-inducible kinase; NUAK; nuclear A
Role of RET protein-tyrosine kinase inhibitors in the treatment RET-driven thyroid and lung cancers
Keywords: دامنه کیناز; ARTN; artemin; AS; activation segment; CD; cadherin-like domain; CDK; cyclin-dependent protein kinase; CL; catalytic loop; CS or C-spine; catalytic spine; CTT; carboxyterminal tail; EGFR; epidermal growth factor receptor; FGFR; fibroblast growth factor re
The role of small molecule platelet-derived growth factor receptor (PDGFR) inhibitors in the treatment of neoplastic disorders
Keywords: دامنه کیناز; Axitinib: (PubMED CID: 6450551); Dasatinib: (PubMED CID: 3062316); Imatinib: (PubMED CID: 5291); Lenvatinib: (PubMED CID: 9823820); Nilotinib: (PubMed CID: 644241); Nintedanib: (PubMed CID: 9809715); Ponatinib: (PubMed CID: 24826799); Sorafenib: (PubMed C
Efficient sortase-mediated N-terminal labeling of TEV protease cleaved recombinant proteins
Keywords: دامنه کیناز; Sortase; Post-labeling purification; TEV; LPXTG; Affinity tag; TEV; Tobacco Etch Virus; EGFR; epidermal growth factor receptor; MSP; membrane scaffold protein; HER; Human Epidermal growth factor Receptor; KD; kinase domain; SrtA; Sortase A; ACP; acyl carr
Characterization and enzymatic properties of protein kinase ACR4 from Arabidopsis thaliana
Keywords: دامنه کیناز; ACR4; Kinase domain; Enzymatic property; Arabidopsis thaliana;
De novo ALK kinase domain mutations are uncommon in kinase inhibitor-naïve ALK rearranged lung cancers
Keywords: دامنه کیناز; Mutation; Lung cancer; Adenocarcinoma; ALK; Kinase domain; Crizotinib;
Recent progress in the identification of adenosine monophosphate-activated protein kinase (AMPK) activators
Keywords: دامنه کیناز; ACC; acetyl-CoA carboxylase; ADaM; allosteric drug and metabolite; AID; auto-inhibitory domain; α-RIM; α-regulatory interacting motif; AMPK; adenosine monophosphate-activated protein kinase; ASMS; affinity selection mass spectrometry; CamKKβ; Ca2+/calm
Threonine 34 phosphorylation by phosphoinositide-dependent protein kinase 1 facilitates dissociation of Akt from the plasma membrane
Keywords: دامنه کیناز; Akt; protein kinase B; IGF; insulin-like growth factor; KD; kinase domain; MAPKAPK2; mitogen-activated protein kinase-activated protein kinase 2; MS; mass spectrometry; PDK; phosphoinositide-dependent protein kinase; PH; pleckstrin homology; PIK3; phospha
Polo-like kinase 3 (PLK3) mediates the clearance of the accumulated PrP mutants transiently expressed in cultured cells and pathogenic PrPSc in prion infected cell line via protein interaction
Keywords: دامنه کیناز; PLKs; polo-like kinases; KD; kinase domain; PBD; polo-box domain; TSE; transmissible spongiform encephalopathies; CJD; Creutzfeldt-Jakob disease; GSS; Gerstmann-Straüssler-Scheinker; FFI; fatal familial insomnia; BSE; bovine spongiform encephalopat
Molecular dynamics of the asymmetric dimers of EGFR: Simulations on the active and inactive conformations of the kinase domain
Keywords: دامنه کیناز; EGFR; Kinase domain; Asymmetric dimers; Molecular dynamics; Essential dynamics; Intermolecular interactions
HER family kinase domain mutations promote tumor progression and can predict response to treatment in human breast cancer
Keywords: دامنه کیناز; HER family mutation; Kinase domain; Lapatinib; Drug resistance; Biomarker; TKI; tyrosine kinase inhibitors;
The early manifestation, tumor-specific occurrence and prognostic significance of TGFBR2 aberrant splicing in oral carcinoma
Keywords: دامنه کیناز; Oral cancer; TGFβ signaling; Alternative splicing; TGFBR2; Kinase domain; Sequencing;
Implications of BCR-ABL1 kinase domain-mediated resistance in chronic myeloid leukemia
Keywords: دامنه کیناز; BCR-ABL1; Kinase domain; Tyrosine kinase inhibitors; Philadelphia chromosome; Chronic myeloid leukemia; Resistance; Mutations;
Ectopic expression of ZmSIMK1 leads to improved drought tolerance and activation of systematic acquired resistance in transgenic tobacco
Keywords: دامنه کیناز; MAPK; mitogen-activated protein kinase; qRT-PCR; quantitative real-time PCR; RT-PCR; reverse transcription PCR; Pst DC3000; Pseudomonas syringae pv. tomato DC3000; ROS; reactive oxygen species; PR; pathogen related genes; SAR; systemic acquired resistance
Novel small-molecule AMPK activator orally exerts beneficial effects on diabetic db/db mice
Keywords: دامنه کیناز; AMPK; AMP-activated protein kinase; ACC; acetyl-CoA carboxylase; CNTF; ciliary neurotrophic factor; AICAR; 5-aminoimidazole-4-carboxamide ribonucleoside; KD; kinase domain; AID; autoinhibitory domain; GBD; glycogen-binding domain; CaMKKα/β; calmodulin-d
The type 2 anti-Müllerian hormone receptor has splice variants that are dominant-negative inhibitors
Keywords: دامنه کیناز; Amhr2; Dominant-negative; Kinase domain; Ligand binding domain; Bone-morphogenetic protein responsive element
Benzimidazole inhibitors of the protein kinase CHK2: Clarification of the binding mode by flexible side chain docking and protein-ligand crystallography
Keywords: دامنه کیناز; ADP; adenosine diphosphate; ATM; ataxia telangiectasia mutated; ATP; adenosine triphosphate; CHK2; checkpoint kinase 2; GOLD; genetic optimisation for ligand docking; GST; glutathione S-transferase; KD; kinase domain; MOE; molecular operating environment;
LOV2-linker-kinase phosphorylates LOV1-containing N-terminal polypeptide substrate via photoreaction of LOV2 in Arabidopsis phototropin1
Keywords: دامنه کیناز; At; Arabidopsis thaliana; BL; blue light; CBB; Coomassie brilliant blue; D450; ground state of phototropin; FMN; flavin mononucleotide; GFP; Green Fluorescent Protein; GST; glutathione S-transferase; KD; kinase domain; L; linker; LOV; light-oxygen-voltage
Detection and molecular characterization of a novel BRAF activated domain mutation in follicular variant of papillary thyroid carcinoma
Keywords: دامنه کیناز; BRAF mutations; Follicular variant papillary thyroid carcinoma; Kinase domain; Modeling
Requirement of the SH4 and tyrosine-kinase domains but not the kinase activity of Lyn for its biosynthetic targeting to caveolin-positive Golgi membranes
Keywords: دامنه کیناز; Golgi caveolin; Kinase domain; Lipid modification; Lyn; Src-family tyrosine kinase; Targeting;
High-resolution melt curve analysis: Initial screening for mutations in BCR-ABL kinase domain
Keywords: دامنه کیناز; CML; BCR-ABL; HRM; Kinase domain; Mutation; Resistance
Characterization and development of a peptide substrate-based phosphate transfer assay for the human vascular endothelial growth factor receptor-2 tyrosine kinase
Keywords: دامنه کیناز; VEGF; Kdr; Receptor tyrosine kinase; Phosphorylation assay; Autophosphorylation; Angiogenesis; Kinase domain
Structure of human Fyn kinase domain complexed with staurosporine
Keywords: دامنه کیناز; Fyn; Kinase domain; Non-receptor tyrosine kinase; Src family; Staurosporine; Inhibitor; X-ray crystal structure