Keywords: اکسازولیدین; Gram-positive bacteria; Japanese; Methicillin-resistant Staphylococcus aureus; Oxazolidinone; Skin and soft tissue infection; Tedizolid phosphate;
مقالات ISI اکسازولیدین (ترجمه نشده)
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Keywords: اکسازولیدین; Spiropyrimidinetrione; Oxazolidinone; [1,5]-Hydride shift; Drug resistance;
Keywords: اکسازولیدین; Azomethine; Haircolor; Oxidation dye; Oxazolidinone; Phthalimide; Coupler; PPD; 1 = p-phenylenediamine = benzene-1,4-diamine; MPD; m-phenylenediamine = benzene-1,3-diamine; MAP; m-aminophenol; AHT; 3 = 4-amino-2-hydroxytoluene = 5-amino-2-methylpheno
Keywords: اکسازولیدین; bioavailability; healthy Korean subjects; oxazolidinone; pharmacokinetics; tedizolid;
Keywords: اکسازولیدین; Antimicrobials; Oxazolidinone; Mycobacterium tuberculosis; Staphylococcus aureus; E. faecalis
Keywords: اکسازولیدین; Methicillin-resistant Staphylococcus aureus; Pulmonary infection; Murine model; Oxazolidinone;
Keywords: اکسازولیدین; ECG; QT prolongation; Safety; Oxazolidinone; Antibacterial; Heart;
Keywords: اکسازولیدین; sp3-rich; Library; Bicyclic; Scaffold; Oxazolidinone;
Keywords: اکسازولیدین; Migraine; CGRP; Oxazolidinone; Class B GPCR; Scaffold hopping;
Keywords: اکسازولیدین; Tedizolid; Linezolid; cfr; Surveillance; Oxazolidinone
Keywords: اکسازولیدین; Lipases; Kinetic resolution; Oxazolidinone; Asymmetric synthesis;
Keywords: اکسازولیدین; nAChR; Carbachol; Ligand; Affinity; Carbamoyl; Oxazolidinone;
Keywords: اکسازولیدین; Oxazolidinone; Kinetic resolution; Asymmetric, synthesis; Candida antarctica lipase B; Cascade alkoxycarbonylation
Keywords: اکسازولیدین; ABSSSI; Latino ethnicity; Oxazolidinone; Tedizolid
Toward polymers with oxazolidin-2-one building blocks through tetra-n-butyl-ammonium halides (Cl, Br, I) catalyzed coupling of epoxides with isocyanates
Keywords: اکسازولیدین; Oxazolidinone; Isocyanurate; Homogeneous catalysis; Epoxide prepolymer;
In vivo efficacy and pharmacokinetics of bi-aryl oxazolidinone RBx 11760 loaded polylactic acid-polyethylene glycol nanoparticles in mouse hematogenous bronchopneumonia and rat groin abscess caused by Staphylococcus aureus
Keywords: اکسازولیدین; Nanoparticles; PLA-PEG; Oxazolidinone; Staphylococcus aureus; Antibacterial; Nanomedicine; ATCC; American type culture collection; ATR-FTIR; attenuated total reflectance-Fourier transforms infrared spectroscopy; ACN; acetonitrile; ADME; absorption, dist
Stereoselective synthesis and transformations of pinane-based 1,3-diaminoalcohols
Keywords: اکسازولیدین; Diaminoalcohol; Catalyst; Oxazolidinone; Monoterpene; Stereochemistry;
Promising in vitro and in vivo inhibition of multidrug-resistant Helicobacter pylori by linezolid and novel oxazolidinone analogues
Keywords: اکسازولیدین; Oxazolidinone; Antimicrobial agent; Helicobacter pylori; Multidrug resistance;
Synthesis and evaluation of pretomanid (PA-824) oxazolidinone hybrids
Keywords: اکسازولیدین; Tuberculosis; Antituberculosis; Oxazolidinone; Pretomanid; PA-824; Antibiotic;
Novel metabolites from the roots of Cadaba natalensis
Keywords: اکسازولیدین; Cadaba natalensis; Diazacyclododecanedione; Oxazolidinone; Isoquiniline alkaloids; Isolation; Structure elucidation;
Sialylation with systematically protected allyl galactoside acceptors using sialyl phosphate donors
Keywords: اکسازولیدین; Sialylation; Carbohydrate; Sialyl phosphate donor; Oxazolidinone;
Structure–activity relationship study of a series of novel oxazolidinone derivatives as IL-6 signaling blockers
Keywords: اکسازولیدین; Rheumatoid arthritis; IL-6 antagonists; IL-6 signaling inhibitor; STAT3; gp130; Oxazolidinone
How to explain low molar masses in PolyHydroxyUrethanes (PHUs)
Keywords: اکسازولیدین; PolyHydroxyUrethanes; Oxazolidinone; Ureas; Molar masses; Side-reactions; Carbonates
Chemical approach for the syntheses of GM4 isomers with sialic acid to non-natural linkage positions on galactose
Keywords: اکسازولیدین; Sialylation; Oxazolidinone; Anomeric configuration; GM4
Lactam and oxazolidinone derived potent 5-hydroxytryptamine 6 receptor antagonists
Keywords: اکسازولیدین; 5-Hydroxytryptamine; Antagonist; Lactam; Oxazolidinone; CNS;
A novel one-pot synthesis of oxazolidinones through direct introduction of CO2 into allylamine derivatives
Keywords: اکسازولیدین; Oxazolidinone; Allylamine; Carbon dioxide fixation; One-pot synthesis; Supercritical fluids;
Synthesis of α-chiral-β,γ-unsaturated carboxylic acid derivatives using chiral auxiliaries
Keywords: اکسازولیدین; Chiral auxiliary; Diastereoselective alkylation; Pseudoephedrine; Oxazolidinone;
Thermally induced substrate release via intramolecular cyclizations of Amino esters and Amino carbonates
Keywords: اکسازولیدین; Lactam; Oxazolidinone; Drug delivery; Poly(dimethylsiloxane) microchannel;
Dehydrative synthesis of chiral oxazolidinones catalyzed by alkali metal carbonates under low pressure of CO2
Keywords: اکسازولیدین; Carbon dioxide; Amino alcohol; Dehydration; Cesium carbonate; Alkali metal carbonate; Oxazolidinone;
Synthesis and antibacterial activities of new piperidine substituted (5R)-[1,2,3]triazolylmethyl and (5R)-[(4-F-[1,2,3]triazolyl)methyl] oxazolidinones
Keywords: اکسازولیدین; Oxazolidinone; Antibiotics; Synthesis; Antibacterial activity;
Design and synthesis of N-alkyldeoxynojirimycin derivatives with improved metabolic stability as inhibitors of BVDV and Tacaribe virus
Keywords: اکسازولیدین; N-Alkyldeoxynojirimycin; Sulfonamide; Urea; Oxazolidinone; Metabolic stability; Antiviral; BVDV; Tacaribe;
Novel 3-O-carbamoyl erythromycin A derivatives (carbamolides) with activity against resistant staphylococcal and streptococcal isolates
Keywords: اکسازولیدین; Bacterial resistance; cfr; erm; MLSb; MRSA; Macrolide; Carbamolide; Clarithromycin; Oxazolidinone; Linezolid; Ribosome X-ray; Deinococcus radiodurans
Design of task-specific ionic liquids for catalytic conversion of CO2 with aziridines under mild conditions
Keywords: اکسازولیدین; Polyethylene glycol; Ionic liquids; Carbon dioxide; Aziridine; Oxazolidinone
Novel promising linezolid analogues: Rational design, synthesis and biological evaluation
Keywords: اکسازولیدین; Linezolid; Oxazolidinone; Thiourea; Antibacterial; Structure–activity relationship
Nuevos fármacos antituberculosos en la tuberculosis resistente y multirresistente
Keywords: اکسازولیدین; Tuberculosis multirresistente; Nuevos fármacos; Fluoroquinolonas; Nitroimidazoles; Diarilquinolina; Oxazolidinona; SQ109Multidrug-resistant tuberculosis; New drugs; Fluoroquinolone; Nitroimidazole; Diarylquinoline; Oxazolidinone; SQ109
Antibacterial oxazolidinone analogues having a N-hydroxyacetyl-substituted seven-membered [1,2,5]triazepane or [1,2,5]oxadiazepane C-ring unit
Keywords: اکسازولیدین; Antibacterial; Oxazolidinone; [1,2,5]Triazepane; [1,2,5]Oxadiazepane;
Synthesis and in vitro/in vivo antibacterial activity of oxazolidinones having thiocarbamate at C-5 on the A-ring and an amide- or urea-substituted [1,2,5]triazepane or [1,2,5]oxadiazepane as the C-ring
Keywords: اکسازولیدین; Antibacterial; Oxazolidinone; Methicillin-resistant Staphylococcus aureus; [1,2,5]Triazepane; [1,2,5]Oxadiazepane
Copper (I) catalyzed synthesis of 1,3-oxazolidin-2-ones from alkynes, amines, and carbon dioxide under solvent-free conditions
Keywords: اکسازولیدین; Carbon dioxide; Oxazolidinone; Solvent-free; Copper-catalyzed;
Antibacterial activity of LCB01-0062, a novel oxazolidinone
Keywords: اکسازولیدین; LCB01-0062; Oxazolidinone; MIC; Time-kill; Systemic infection;
Syntheses and biological studies of novel spiropiperazinyl oxazolidinone antibacterial agents using a spirocyclic diene derived acylnitroso DielsâAlder reaction
Keywords: اکسازولیدین; Oxazolidinone; Antibiotics; Nitroso DielsâAlder reaction; Spirocyclic diene; MRSA;
Synthesis and preliminary antibacterial evaluation of Linezolid-like 1,2,4-oxadiazole derivatives
Keywords: اکسازولیدین; Oxazolidinone; 1,2,4-Oxadiazole; Linezolid; Antimicrobial activity; Fluorinated heterocycles
Résistance au linézolide chez les staphylocoques
Keywords: اکسازولیدین; Linezolide; ARNr 23S; Gène cfr; Oxazolidinones; Ribosome; Staphylocoques; Linezolid; 23S rRNA; Cfr gene; Oxazolidinone; Ribosom; Staphylococci;
Efficient synthesis and anti-enteroviral activity of 9-arylpurines
Keywords: اکسازولیدین; Purines; Microwave-assisted synthesis; Oxazolidinone; Enterovirus; Coxsackie virus B3CVB3, coxsackie virus type B3; MAOS, microwave-assisted organic synthesisVHJZZHRWGKIDIH-UHFFFAOYSA-N; KFRLPTRPEAWAJZ-UHFFFAOYSA-N; IUDVIGAJZAHZLJ-UHFFFAOYSA-N; XVZMLNVQHL
Shape memory polymers based on cyanate ester-epoxy-poly (tetramethyleneoxide) co-reacted system
Keywords: اکسازولیدین; Shape memory polymer; Cyanate ester-epoxy blend; Oxazolidinone; Poly(tetramethyleneoxide)
Structure–activity studies of RNA-binding oxazolidinone derivatives
Keywords: اکسازولیدین; RNA; Oxazolidinone; Antiterminator; T-box riboswitch; FRET
Novel 3-chlorooxazolidin-2-ones as antimicrobial agents
Keywords: اکسازولیدین; Antibacterial; Antifungal; Antimicrobial; Oxazolidinone; Topical
Discovery of a novel nitroimidazolyl-oxazolidinone hybrid with potent anti Gram-positive activity: Synthesis and antibacterial evaluation
Keywords: اکسازولیدین; Oxazolidinone; Nitroimidazole; In vitro antibacterial activity; Cytotoxicity;
Interaction of substrate and catalyst during the formation of oxazolidinones from 2-aminoalcohols and diethyl carbonate using recyclable 1,3-dichlorodistannoxanes
Keywords: اکسازولیدین; Oxazolidinone; Recyclable distannoxane; Diethylcarbonate; 2-Aminoalcohols; Catalyst–substrate interaction
Design, synthesis and docking studies of quinoline-oxazolidinone hybrid molecules and their antitubercular properties
Keywords: اکسازولیدین; 4-Aminoquinoline; Oxazolidinone; Antibacterial; Antimycobacterial activity; Docking studies
Discovery of torezolid as a novel 5-hydroxymethyl-oxazolidinone antibacterial agent
Keywords: اکسازولیدین; Oxazolidinone; Pyridine; Antibiotics; Prodrug; Antibacterial activity; DA-7867