Keywords: تردید جزئی; G protein-coupled receptors; partial agonism; biased agonism; rational ligand design; dynamic ligand binding; dualsteric binding
مقالات ISI تردید جزئی (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
From pyrrolidinyl-benzodioxane to pyrrolidinyl-pyridodioxanes, or from unselective antagonism to selective partial agonism at α4β2 nicotinic acetylcholine receptor
Keywords: تردید جزئی; α4β2 nAChR; α3β4 nAChR; Benzodioxane; Pyridodioxane; Partial agonism; Antagonism;
Vilazodone does not inhibit sexual behavior in male rats in contrast to paroxetine: A role for 5-HT1A receptors?
Keywords: تردید جزئی; Preclinical; Antidepressant; Serotonin receptor; Partial agonism;
ReviewSerotonin in antipsychotic drugs action
Keywords: تردید جزئی; 5-HT; 5-HT levels; Antipsychotic drugs; Microdialysis; Receptors; Affinity; Agonism; Antagonism; Partial agonism; Inverse agonism;
Non-specific binding and general cross-reactivity of Y receptor agonists are correlated and should importantly depend on their acidic sectors
Keywords: تردید جزئی; BIBP3226; (R)-N2-(diphenylacetyl)-N-[(4-hydroxyphenyl)methyl]d-arginineamide; BIIE0246; N-[(1S)-4-[(aminoiminomethyl)amino]-1-[([2-(3,5-dioxo-1,2-diphenyl-1,2,4-triazolidin-4-yl)ethyl]amino)carbonyl]butyl]-1-(2-[4-(6,11-dihydro-6-oxo-5H-dibenz[b,e]azepin-
Comparative biochemical and pharmacological characterization of a novel, NOP receptor selective hexapeptide, Ac-RYYRIR-ol
Keywords: تردید جزئی; N/OFQ; nociceptin/orphanin FQ; NOP receptor; N/OFQ peptide receptor; Ac-RYYRIK-ol; Acetyl-Arg-Tyr-Tyr-Arg-Ile-Lys-ol; Nociceptin/orphanin FQ (NOP) receptor; Hexapeptide ligands; Receptor binding; G-protein activation; In vitro pharmacology; Part
Synthesis and opioid activity of novel 6-substituted-6-demethoxy-ethenomorphinans
Keywords: تردید جزئی; Analgesics; Orvinols; Partial agonism; Drug abuse; DFT study
Characterization of new PPARγ agonists: Benzimidazole derivatives—importance of positions 5 and 6, and computational studies on the binding mode
Keywords: تردید جزئی; Benzimidazole derivatives; Partial agonism; Selective PPARγ modulators; Structure–activity relationship; Molecular modeling
Exploring kainate receptor pharmacology using molecular dynamics simulations
Keywords: تردید جزئی; Molecular dynamics; Agonism; Partial agonism; Antagonism; Kainate receptor; Ionotropic glutamate receptor;
Brain regional distribution of GABAA receptors exhibiting atypical GABA agonism: Roles of receptor subunits
Keywords: تردید جزئی; GABAA receptor; [35S]TBPS autoradiography; THIP; Gaboxadol; Partial agonism; Thalamus; Cerebellum
2-(4-Amino-3-methylphenyl)-5-fluorobenzothiazole is a ligand and shows species-specific partial agonism of the aryl hydrocarbon receptor
Keywords: تردید جزئی; 5F 203; 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole; TCAOB; tetrachloroazoxybenzene; TCDD; 2,3,7,8-tetrachlorodibenzo-p-dioxin; DMSO; dimethyl sulfoxide; MTT; 3-(4,5-Dimethylthiazol-2-yl)-2,5-diphenyltetrazolium bromide; AhR; aryl hydrocarbon recepto
Novel diastereomeric opioid tetrapeptides exhibit differing pharmacological activity profiles
Keywords: تردید جزئی; Opioid receptors; δ-Antagonists; Tritium labeling; Radioligand binding; G-protein activation; Partial agonism; Rat brain; CHO cells;
Partial and full agonism in endomorphin derivatives: Comparison by null and operational model
Keywords: تردید جزئی; Endomorphin derivatives; Partial agonism; Residual receptor fraction; β-Funaltrexamine; Mouse vas deferens; Null and operational model;
Aripiprazole and its human metabolite are partial agonists at the human dopamine D2 receptor, but the rodent metabolite displays antagonist properties
Keywords: تردید جزئی; Aripiprazole; Dopamine D2 receptor; Partial agonism