Keywords: آگونیست های جزئی; Agonistas parciales; Buprenorfina; Vareniclina; Aripiprazol; Memantina; Partial agonists; Buprenorphine; Varenicline; Aripiprazole; Memantine;
مقالات ISI آگونیست های جزئی (ترجمه نشده)
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Assessments of cellular melatonin receptor signaling pathways: β-arrestin recruitment, receptor internalization, and impedance variations
Keywords: آگونیست های جزئی; Melatonin receptors; Technical assessments; β-arrestin; Internalization; CellKey®; Partial agonists;
Molecular determinants of PPARγ partial agonism and related in silico/in vivo studies of natural saponins as potential type 2 diabetes modulators
Keywords: آگونیست های جزئی; Type 2 diabetes; Saponins; PPARγ; Partial agonists; Pharmacophore; Docking; CAT; catalase; GSH; reduced glutathione; HB; hydrogen bond; MDA; malondialdehyde; NADPH; beta-nicotinamide adenine dinucleotide 2â²-phosphate; PDB; Protein Data Bank; PPARγ;
Synthesis and biological evaluation of novel hybrids of highly potent and selective α4β2-Nicotinic acetylcholine receptor (nAChR) partial agonists
Keywords: آگونیست های جزئی; α4β2-nAChRs; Partial agonists; Hybrids; Antidepressant-like effects; CNS; central nervous system; AD; Alzheimer's disease; ADHD; attention deficit hyperactivity disorder; NIMH-PDSP; National Institute of Mental Health Psychoactive Drug Screening Program
Synthesis and SAR of aminothiazole fused benzazepines as selective dopamine D2 partial agonists
Keywords: آگونیست های جزئی; Dopamine; Partial agonists;
Conformational restriction in a series of GPR119 agonists: Differences in pharmacology between mouse and human
Keywords: آگونیست های جزئی; G-protein coupled receptors; GPR119 agonists; Pharmacology; Partial agonists
Novel azulene derivatives for the treatment of erectile dysfunction
Keywords: آگونیست های جزئی; Penile erection; Erectile dysfunction; Azulene; Dopamine D4; Partial agonists;
Use of an α3β4 nicotinic acetylcholine receptor subunit concatamer to characterize ganglionic receptor subtypes with specific subunit composition reveals species-specific pharmacologic properties
Keywords: آگونیست های جزئی; Smoking cessation; Drug screening; Ganglionic receptors; Partial agonists; BTMPS; [bis-(2,2,6,6-tetramethyl-4-piperidinyl)-sebacate]; TMPH; 2,2,6,6-tetramethylpiperidin-4-yl heptanoate; GTS-21; (3-(2,4dimethoxybenzylidene)anabaseine); SNP; single nucleoti
Synthesis and P2Y2 receptor agonist activities of uridine 5â²-phosphonate analogues
Keywords: آگونیست های جزئی; NBS; N-bromosuccinimide; TMSBr; trimethylsilyl bromide; TFA; trifluoroacetic acid; NMO; N-methylmorpholine-N-oxide; P2Y2 receptor; G protein-coupled receptor; Uracil nucleotides; Nucleoside phosphonates; Partial agonists;
Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors
Keywords: آگونیست های جزئی; Synthesis; Quinolones; Cannabinoid ligands; Partial agonists; Peripheral ligandsBBB, blood–brain barrier; CB1, cannabinoid type-1; CB2, cannabinoid type-2; CHO, chinese hamster ovary cell; CNS, central nervous system; DIPEA, diisopropylethylamine; DME, 1,
Positive modulation of α7 nAChR responses in rat hippocampal interneurons to full agonists and the α7-selective partial agonists, 4OH-GTS-21 and S 24795
Keywords: آگونیست های جزئی; Brain slices; Patch-clamp; nAChRs; Partial agonists; Full agonists; Hippocampus; Positive allosteric modulators;
NMR Spectroscopy of the Ligand-Binding Core of Ionotropic Glutamate Receptor 2 Bound to 5-Substituted Willardiine Partial Agonists
Keywords: آگونیست های جزئی; AMPA, α-amino-3-hydroxy-5-methylisoxazole-4-propionic acid; GluR, glutamate receptorglutamate receptor; AMPA; partial agonists; NMR; chemical exchange
The novel antidyskinetic drug sarizotan elicits different functional responses at human D2-like dopamine receptors
Keywords: آگونیست های جزئی; Parkinson's disease; Dyskinesia; GIRK channels; Adenylyl cyclase; Sarizotan; Signaling; Functional selectivity; Dopamine receptors; AtT-20 neuroendocrine cells; Partial agonists; Electrophysiology
Selective PPARγ modulators with improved pharmacological profiles
Keywords: آگونیست های جزئی; PPAR; Selective modulator; Partial agonists
Buprenorphine: Considerations for Pain Management
Keywords: آگونیست های جزئی; Buprenorphine; pharmacology; pharmacodynamics; pharmacokinetics; pain management; partial agonists; formulations; opioids;