Keywords: مهارکننده پپتید; Antibiotic resistance; Penicillinase; Enzyme inhibitor; Peptide inhibitor; Phage display; Surface plasmon resonance
مقالات ISI مهارکننده پپتید (ترجمه نشده)
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در صورتی که به ترجمه آماده هر یک از مقالات زیر نیاز داشته باشید، می توانید سفارش دهید تا مترجمان با تجربه این مجموعه در اسرع وقت آن را برای شما ترجمه نمایند.
Keywords: مهارکننده پپتید; Design; Diabetes mellitus type 2; Insulin receptor; Peptide inhibitor; Modification
Development of a potent peptide inhibitor of estrogen receptor α
Keywords: مهارکننده پپتید; Peptide inhibitor; TD strategy; N-terminus helix-nucleating strategy; Estrogen receptor α; Cell penetrating peptide;
Ac-LVFFARK-NH2 conjugation to β-cyclodextrin exhibits significantly enhanced performance on inhibiting amyloid β-protein fibrillogenesis and cytotoxicity
Keywords: مهارکننده پپتید; Amyloid β-protein; Peptide inhibitor; β-Cyclodextrin; Conjugation; Inhibition;
The inhibitory effects of biomimetically designed peptides on α-synuclein aggregation
Keywords: مهارکننده پپتید; Peptide inhibitor; Amyloid fibril formation; α-Synuclein; Parkinson's disease;
Development of peptide inhibitors of HIV transmission
Keywords: مهارکننده پپتید; HIV; HIV treatment; Drug development; Peptide therapeutic; Peptide inhibitor; HIV; human immunodeficiency virus; AIDS; acquired immunodeficiency syndrome; CDC; Centers for Disease Control and Prevention; FY; fiscal year; R&D; research and development; FDA
Engineering a peptide inhibitor towards the KCNQ1/KCNE1 potassium channel (IKs)
Keywords: مهارکننده پپتید; KCNQ1/KCNE1; Peptide inhibitor; Molecular design; MT2 peptide; MT2-2 peptide;
A new Kunitz-type plasmin inhibitor from scorpion venom
Keywords: مهارکننده پپتید; Plasmin; BmKTT-2; Peptide inhibitor; Kunitz-type; Scorpion venom
Effects of Lys to Glu mutations in GsMTx4 on membrane binding, peptide orientation, and self-association propensity, as analyzed by molecular dynamics simulations
Keywords: مهارکننده پپتید; Peptide inhibitor; Mechanotransduction; Multiscale simulations; Membrane-active peptide;
Inhibition of embryo implantation in mice through vaginal administration of a proprotein convertase 6 inhibitor
Keywords: مهارکننده پپتید; Proprotein convertase; Embryo implantation; Peptide inhibitor; Vaginal drug delivery; Contraceptive
Class specific peptide inhibitors for secretory phospholipases A2
Keywords: مهارکننده پپتید; AMP; antimicrobial peptides; bv; bee venom; C28-O-PHPM; 1-octosanyl-2-(pyren-1-yl)hexanoyl-sn-glycero-3-phospho-monomethyl ester; cPLA2; cytosolic PLA2; CSSP; continuum secondary structure predictor; EM; electron microscopy; FFA; free fatty acid; Hsp70; h
A novel retro-inverso peptide is a preferential JNK substrate-competitive inhibitor
Keywords: مهارکننده پپتید; c-Jun N-terminal kinase; Peptide inhibitor; Activity assays; Binding assays; Substrate selectivity;
A multivalent peptide as an activator of hypoxia inducible factor-1α
Keywords: مهارکننده پپتید; Hypoxia-inducible factor; Peptide inhibitor; VBC; Multivalent peptide inhibitor; VEGF
Tripeptide inhibitors of dengue and West Nile virus NS2B-NS3 protease
Keywords: مهارکننده پپتید; Dengue virus; West Nile virus; NS2B-NS3 protease; Peptide inhibitor;
Inhibition of isoflurane-induced increase of cell-surface redistribution and activity of glutamate transporter type 3 by serine 465 sequence-specific peptides
Keywords: مهارکننده پپتید; Glutamate transporter; Isoflurane; Neuron; Peptide inhibitor; Protein kinase C; Trafficking;
Neurite outgrowth from PC12 cells is enhanced by an inhibitor of mechanical channels
Keywords: مهارکننده پپتید; Neurite outgrowth; Mechanical channels; GsMTx4; Peptide inhibitor; NGF; PC12
Venom neutralization by purified bioactive molecules: Synthetic peptide derivatives of the endogenous PLA2 inhibitory protein PIP (a mini-review)
Keywords: مهارکننده پپتید; Antivenom; Snake venom; Neutralization; Secretory phospholipase A2; Metalloproteinase; Peptide inhibitor
Inhibition of HSP27 phosphorylation by a cell-permeant MAPKAP Kinase 2 inhibitor
Keywords: مهارکننده پپتید; Heat shock protein 27; HSP27 phosphorylation; MAPKAP Kinase 2; Keloid fibroblast; TGF-β1; CTGF; Collagen type I; Peptide inhibitor
A novel non-phosphorylated potential antitumoral peptide inhibits STAT3 biological activity
Keywords: مهارکننده پپتید; STAT3; Peptide inhibitor; Immunofluorescence; Cellular effects; Ahx; 6-amino hexanoic acid; Antp; Antennapedia sequence; BOP; (benzotriazol-1-yloxy)tris(dimethylamino)phosphonium hexafluorophosphate; DIPEA; diisopropylethylamine; GPK; GMP-protein dependan
Substrate specificity and screening of the integral membrane protease Pla
Keywords: مهارکننده پپتید; Yersinia pestis; Plasminogen activator; Protease substrate; Peptide inhibitor; Positional scan; Parallel synthesis;
Inhibition of IL-1β transcription by peptides derived from the hCMV IE2 transactivator
Keywords: مهارکننده پپتید; hCMV; human cytomegalovirus; DBD; DNA-binding domain; IL1B; gene encoding IL-1β; TLR; Toll-like receptor; bZIP; basic leucine zipper domain; Interleukin 1β; Cytomegalovirus; IE2; Transcription factors; Peptide inhibitor;
Effect of transcription peptide inhibitors on HIV-1 replication
Keywords: مهارکننده پپتید; HIV; Cyclin-dependent kinase; Tat; Peptide inhibitor; Transcription; Cell cycle; Computer modeling; PBMC; Small animal model; Stem cells
Neutralization of the haemorrhagic activities of viperine snake venoms and venom metalloproteinases using synthetic peptide inhibitors and chelators
Keywords: مهارکننده پپتید; Snake venom; Echis; Haemorrhagic activity; Metalloproteinase; Peptide inhibitor; Chelator
Development of a peptide inhibitor-based cantilever sensor assay for cyclic adenosine monophosphate-dependent protein kinase
Keywords: مهارکننده پپتید; Peptide inhibitor; Heat-stable protein kinase inhibitor; Cyclic adenosine monophosphate-dependent protein kinase; Nanomechanical cantilever; Surface plasmon resonance; Capillary electrophoresis; Fluorescence polarization
The N-terminal octapeptide acts as a dimerization inhibitor of SARS coronavirus 3C-like proteinase
Keywords: مهارکننده پپتید; SARS coronavirus; 3C-like proteinase; Mutational study; N-terminal peptide; Dimerization inhibitor; Peptide inhibitor; Zhang–Poorman plot
The domain on the mouse Duffy protein for Plasmodium yoelii binding and invasion to mouse erythrocytes
Keywords: مهارکننده پپتید; Malaria; Duffy/DARC binding domain; Decoy receptor; Peptide inhibitor
A novel approach to identifying β-secretase inhibitors: Bis-statine peptide mimetics discovered using structure and spot synthesis
Keywords: مهارکننده پپتید; Aspartic protease; Peptide inhibitor; Peptide spot synthesis; Crystallography; Bis-statine
Inhibition of severe acute respiratory syndrome-associated coronavirus (SARS-CoV) infectivity by peptides analogous to the viral spike protein
Keywords: مهارکننده پپتید; Severe acute respiratory syndrome-associated coronavirus; Class I viral fusion protein; Peptide inhibitor; Murine hepatitis virus; Six-helix bundle; Anti-viral
Inhibition of HIV-1 virus replication using small soluble Tat peptides
Keywords: مهارکننده پپتید; HIV; Cyclin-dependent kinase; Tat; Peptide inhibitor; Transcription; Cell cycle; Computer modeling; PBMC
Exploiting structural principles to design cyclin-dependent kinase inhibitors
Keywords: مهارکننده پپتید; CDK; cyclin-dependent kinase; PKA; cAMP-dependent protein kinase; CMGC-I; CDK-like protein kinases; CML; Chronic myelogenous leukaemia; PfPK5; Plasmodium falciparum Protein Kinase 5; Cyclin-dependent kinase inhibitor; CDK; Drug design; Protein dynamic; Pr
Peptide inhibitors of botulinum neurotoxin by mRNA display
Keywords: مهارکننده پپتید; Toxin; Botulinum; mRNA display; Peptide inhibitor; Protease; Medium-throughput assay; Synthetic cDNA; Expression and purification; Biotin; Ubiquitin; Transcription; Translation;
A peptide inhibitor of exportin1 blocks shuttling of the adenoviral E1B 55 kDa protein but not export of viral late mRNAs
Keywords: مهارکننده پپتید; Adenoviral E1B 55 kDa protein; mRNA export; Exportin1; Peptide Inhibitor;
Peptide inhibitors of protein kinases-discovery, characterisation and use
Keywords: مهارکننده پپتید; AKAP; A-Kinase Anchoring Protein; EGF-R; Epidermal Growth Factor-Receptor; GSK; Glycogen Synthase Kinase; IC50; concentration of compound to achieve 50% inhibition; JIP; JNK Interacting Protein; JNK; c-Jun N-terminal Kinase; Ki; inhibition constant; MLCK;