Synthesis and biological evaluation of conformationally constrained analogs of the antitumor agents XK469 and SH80. Part 5 Fulltext Access 6 Pages 2006
New rifabutin analogs: Synthesis and biological activity against Mycobacterium tuberculosis Fulltext Access 6 Pages 2006
Distachyasin: A new antioxidant metabolite from the leaves of Carex distachya Fulltext Access 6 Pages 2006
Inhibition of Tpl2 kinase and TNFα production with quinoline-3-carbonitriles for the treatment of rheumatoid arthritis Fulltext Access 6 Pages 2006
Identification of 2-arylbenzimidazoles as potent human histamine H4 receptor ligands Fulltext Access 6 Pages 2006
Synthesis and antihyperlipidemic activity of novel glycosyl fructose derivatives Fulltext Access 6 Pages 2006
Comparative protein modeling and surface analysis of Leishmania sirtuin: A potential target for antileishmanial drug discovery Fulltext Access 6 Pages 2006
Metal complexes with superoxide dismutase-like activity as candidates for anti-prion drug Fulltext Access 6 Pages 2006
Expression of N-terminal Cys-protein fragments using an intein refolding strategy Fulltext Access 6 Pages 2006
Synthesis of a library of polycationic lipid core dendrimers and their evaluation in the delivery of an oligonucleotide with hVEGF inhibition Fulltext Access 6 Pages 2006
Closing in on the AMPA receptor: Synthesis and evaluation of 2-acetyl-1-(4′-chlorophenyl)-6-methoxy-7-[11C]methoxy-1,2,3,4-tetrahydroisoquinoline as a potential PET tracer Fulltext Access 6 Pages 2006
Lycopladines B–D and lyconadin B, new alkaloids from Lycopodium complanatum Fulltext Access 6 Pages 2006
Reactive oxygen species scavenging activity of aminoderivatized chitosan with different degree of deacetylation Fulltext Access 6 Pages 2006
Novel imidazole-based combretastatin A-4 analogues: Evaluation of their in vitro antitumor activity and molecular modeling study of their binding to the colchicine site of tubulin Fulltext Access 6 Pages 2006
Synthesis of ethylenediamine linked β-cyclodextrin dimer and its analytical application for tranilast determination by spectrofluorimetry Fulltext Access 6 Pages 2006
Synthesis and antimicrobial activity of novel 2-thiazolylimino-5-arylidene-4-thiazolidinones Fulltext Access 6 Pages 2006
Design, synthesis, SAR, and biological evaluation of new 4-(phenylamino)thieno[2,3-b]pyridine derivatives Fulltext Access 6 Pages 2006
4′-Fluorinated carbocyclic nucleosides: Synthesis and inhibitory activity against S-adenosyl-l-homocysteine hydrolase Fulltext Access 6 Pages 2006
An easy preparation of ‘monolithic type’ hydrophilic solid phase: Capability for affinity resin to isolate target proteins Fulltext Access 6 Pages 2006
Secondary assembly of bile salts mediated by β-cyclodextrin–terbium(III) complex Fulltext Access 6 Pages 2006
Role of glutamine 148 of human 15-hydroxyprostaglandin dehydrogenase in catalytic oxidation of prostaglandin E2 Fulltext Access 6 Pages 2006
Design, synthesis and antibacterial activity of novel 1,3-thiazolidine pyrimidine nucleoside analogues Fulltext Access 6 Pages 2006
Synthesis of new chemical entities from paracetamol and NSAIDs with improved pharmacodynamic profile Fulltext Access 6 Pages 2006
Heteropoly acids as solid green Brønsted acids for a one-pot synthesis of β-acetamido ketones by Dakin–West reaction Fulltext Access 6 Pages 2006
Fungal metabolites of xanthohumol with potent antiproliferative activity on human cancer cell lines in vitro Fulltext Access 6 Pages 2006
Design and synthesis of heterocyclic malonyl-CoA decarboxylase inhibitors Fulltext Access 6 Pages 2006
Synthesis of the novel series of bispyridinium compounds bearing (E)-but-2-ene linker and evaluation of their reactivation activity against chlorpyrifos-inhibited acetylcholinesterase Fulltext Access 6 Pages 2006
Conversion of A3 adenosine receptor agonists into selective antagonists by modification of the 5′-ribofuran-uronamide moiety Fulltext Access 6 Pages 2006
Isolation and inhibitory activity against ERK Phosphorylation of hydroxyanthraquinones from rhubarb Fulltext Access 6 Pages 2006
Designing rapid onset selective serotonin re-uptake inhibitors. Part 1: Structure–activity relationships of substituted (1S,4S)-4-(3,4-dichlorophenyl)-N-methyl-1,2,3,4-tetrahydro-1-naphthaleneamine Fulltext Access 6 Pages 2006
Antioxidant activity and cytoprotective effect of κ-carrageenan oligosaccharides and their different derivatives Fulltext Access 6 Pages 2006
A topological function based on spectral moments for predicting affinity toward A3 adenosine receptors Fulltext Access 6 Pages 2006
The cytotoxicity of ortho alkyl substituted 4-X-phenols: A QSAR based on theoretical bond lengths and electron densities Fulltext Access 6 Pages 2006
Phenolics and antimicrobial activity of traditional stoned table olives ‘alcaparra’ Fulltext Access 6 Pages 2006
Oxadiazole derivatives as a novel class of antimitotic agents: Synthesis, inhibition of tubulin polymerization, and activity in tumor cell lines Fulltext Access 6 Pages 2006
Convenient synthesis of 3- and 6-deoxy-d-myo-inositol phosphate analogues from (+)-epi- and (−)-vibo-quercitols Fulltext Access 6 Pages 2006
Synthesis and SAR of arylaminoethyl amides as noncovalent inhibitors of cathepsin S: P3 cyclic ethers Fulltext Access 6 Pages 2006
Synthesis, radiolabeling, and in vivo evaluation of an 18F-labeled isatin analog for imaging caspase-3 activation in apoptosis Fulltext Access 6 Pages 2006
Synthesis and in vitro biological evaluation of aryl boronic acids as potential inhibitors of factor XIa Fulltext Access 6 Pages 2006
Development of 6-substituted indolylquinolinones as potent Chek1 kinase inhibitors Fulltext Access 6 Pages 2006
4′-Alkoxyl substitution enhancing the anti-mitotic effect of 5-(3′,4′,5′-substituted)anilino-4-hydroxy-8-nitroquinazolines as a novel class of anti-microtubule agents Fulltext Access 6 Pages 2006
A novel oxazine ring closure reaction affording (Z)-((E)-2-styrylbenzo[b]furo[3,2-d][1,3]oxazin-4-ylideno)acetaldehydes and their anti-osteoclastic bone resorption activity Fulltext Access 6 Pages 2006
The synthesis and SAR of 2-amino-pyrrolo[2,3-d]pyrimidines: A new class of Aurora-A kinase inhibitors Fulltext Access 6 Pages 2006
Synthesis of radiolabeled stilbene derivatives as new potential PET probes for aryl hydrocarbon receptor in cancers Fulltext Access 6 Pages 2006
Interspecies variation in yolk selenium concentrations among eggs of free-living birds: The effect of phylogeny Fulltext Access 6 Pages 2006
A multi-component reaction to 5-cyanouracils: Synthesis and mechanistic study Fulltext Access 6 Pages 2006
Controllable synthesis of polymerizable ester and amide prodrugs of acyclovir by enzyme in organic solvent Fulltext Access 6 Pages 2006
The synthesis and anti-proliferative effects of β-elemene derivatives with mTOR inhibition activity Fulltext Access 6 Pages 2006
Development of affinity chromatography using a bioactive peptide as a ligand Fulltext Access 6 Pages 2006
Anticonvulsant and toxicity evaluation of some 7-alkoxy-4,5-dihydro-[1,2,4]triazolo[4,3-a]quinoline-1(2H)-ones Fulltext Access 6 Pages 2006
Synthesis and antimalarial activities of novel 3,3,6,6-tetraalkyl-1,2,4,5-tetraoxanes Fulltext Access 6 Pages 2006
Effect of cooking and legume species upon calcium, iron and zinc uptake by Caco-2 cells Fulltext Access 6 Pages 2006
Rubidium content in autopsy liver tissue samples from Greenlandic Inuit and Danes measured by X-ray fluorescence spectrometry Fulltext Access 6 Pages 2006
Intracellular magnesium in elderly patients with heart failure: Effects of diabetes and renal dysfunction Fulltext Access 6 Pages 2006
Hypoglycemic activity of fermented mushroom of Coprinus comatus rich in vanadium Fulltext Access 6 Pages 2006
A new phenanthrene with a spirolactone from Dendrobium chrysanthum and its anti-inflammatory activities Fulltext Access 6 Pages 2006
Foreign accent syndrome: Best practice, theoretical issues and outstanding questions Fulltext Access 6 Pages 2006
Antibacterial performance of photocatalyst thin film fabricated by defection effect in visible light Fulltext Access 6 Pages 2006
Magnetoelectroporation: improved labeling of neural stem cells and leukocytes for cellular magnetic resonance imaging using a single FDA-approved agent Fulltext Access 6 Pages 2006
Sortie de CEC difficile : tableaux cliniques et modalités thérapeutiques Fulltext Access 6 Pages 2006
Kinetic modeling and simulation of the gluco regulatory system to detect endocrine system failure Fulltext Access 6 Pages 2006
Facile synthesis of non-steroidal anti-inflammatory active bisbenzamide-containing compounds Fulltext Access 6 Pages 2006
Microwave-assisted, one-pot syntheses and fungicidal activity of polyfluorinated 2-benzylthiobenzothiazoles Fulltext Access 6 Pages 2006
Screening a natural product-based combinatorial library using FTICR mass spectrometry Fulltext Access 6 Pages 2006
The acetates of p-nitrophenyl α-l-arabinofuranoside—Regioselective preparation by action of lipases Fulltext Access 6 Pages 2006
Fluorescently tagged iminoalditol glycosidase inhibitors as novel biological probes and diagnostics Fulltext Access 6 Pages 2006
Human serum albumin interaction with formononetin studied using fluorescence anisotropy, FT-IR spectroscopy, and molecular modeling methods Fulltext Access 6 Pages 2006
The 3D-QSAR analysis of 4(3H)-quinazolinone derivatives with dithiocarbamate side chains on thymidylate synthase Fulltext Access 6 Pages 2006
Microwave enhanced solid support synthesis of fluorine containing benzopyrano-triazolo-thiadiazepines as potent anti-fungal agents Fulltext Access 6 Pages 2006
Effects of 9,10-dihydroxy-4,4-dimethyl-5,8-dihydro-1(4H)-anthracenone derivatives on tumor cell respiration Fulltext Access 6 Pages 2006
Design, synthesis, and antitumor evaluation of novel acenaphtho[1,2-b]pyrrole-carboxylic acid esters with amino chain substitution Fulltext Access 6 Pages 2006
Antimalarial potential of xestoquinone, a protein kinase inhibitor isolated from a Vanuatu marine sponge Xestospongia sp. Fulltext Access 6 Pages 2006
Effects of structural modification on the DNA binding properties and photo-induced cleavage reactivity of propargylic sulfones conjugated with an anthraquinone structure Fulltext Access 6 Pages 2006
Synthesis, cytotoxicity, and anti-inflammatory evaluation of 2-(furan-2-yl)-4-(phenoxy)quinoline derivatives. Part 4 Fulltext Access 6 Pages 2006
Natural products as starting materials for development of second-generation SERCA inhibitors targeted towards prostate cancer cells Fulltext Access 6 Pages 2006
Synthesis and antifungal activity of substituted-10-methyl-1,2,3,4-tetrahydropyrazino[1,2-a]indoles Fulltext Access 6 Pages 2006
Design, synthesis, and biological evaluation of 1,3-diarylprop-2-en-1-ones : A novel class of cyclooxygenase-2 inhibitors Fulltext Access 6 Pages 2006
Design and synthesis of quinolinones as methionyl-tRNA synthetase inhibitors Fulltext Access 6 Pages 2006
Synthesis, pulse radiolysis, and in vitro radioprotection studies of melatoninolipoamide, a novel conjugate of melatonin and α-lipoic acid Fulltext Access 6 Pages 2006
Ribokinase from E. coli: Expression, purification, and substrate specificity Fulltext Access 6 Pages 2006
Design of multifunctional peptides expressing both antimicrobial activity and shiga toxin neutralization activity Fulltext Access 6 Pages 2006