Keywords: CPS; chemoprophylaxis with sporozoites; CQ; chloroquine; CQ-CPS; chloroquine chemoprophylaxis with sporozoites; DHA-PPQ; co-formulation of dihydroartemisinin and piperaquine-tetraphosphate; GMP; good manufacturing practice; PPQ; piperaquine-tetraphosphate
مقالات ISI (ترجمه نشده)
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Inhibition of CYP3A by Antimalarial Piperaquine and Its Metabolites in Human Liver Microsomes With IVIV Extrapolation
Keywords: piperaquine; CYP inhibition; drug-drug interaction;
Efficacy and safety of intermittent preventive treatment in schoolchildren with sulfadoxine/pyrimethamine (SP) and SP plus piperaquine in Democratic Republic of the Congo: a randomised controlled trial
Keywords: Intermittent preventive treatment; Malaria; Schoolchildren; Sulfadoxine/pyrimethamine; Piperaquine; Kinshasa;
LC-MS/MS quantitation of antimalarial drug piperaquine and metabolites in human plasma
Keywords: Piperaquine; Malaria; LC-MS/MS; Pharmacokinetics; Drug metabolism;
Efficacy of Synriamâ¢, a new antimalarial combination of OZ277 and piperaquine, against different developmental stages of Schistosoma mansoni
Keywords: Synriamâ¢; 1,2,4 Trioxolane; Piperaquine; Anti-schistosomal drug; Drug repositioning;
Refrigeration provides a simple means to synchronize in vitro cultures of Plasmodium falciparum
Keywords: DHA; dihydroartemisinin; PPQ; piperaquine; CQ; chloroquine; QN; quinine; Synchronization; Plasmodium falciparum; Refrigeration; Drug susceptibility;
Piperaquine and Lumefantrine resistance in Plasmodium berghei ANKA associated with increased expression of Ca2+/H+ antiporter and glutathione associated enzymes
Keywords: Malaria; Plasmodium berghei; Resistance; Piperaquine; Lumefantrine;
Orally Formulated Artemisinin in Healthy Fasting Vietnamese Male Subjects: A Randomized, Four-Sequence, Open-Label, Pharmacokinetic Crossover Study
Keywords: ACT; artemisinin; bioequivalence; malaria; pharmacokinetics; piperaquine;
Investigation of reproductive toxicity of piperaquine in mice
Keywords: Piperaquine; Pregnancy; Mouse; Toxicology; Biochemistry; Haematology; Pharmacokinetics; Malaria
Plasmodium berghei ANKA: Selection of resistance to piperaquine and lumefantrine in a mouse model
Keywords: Malaria; Plasmodium berghei; Drug resistance; Cross-resistance; Lumefantrine; Piperaquine;
The influence of food on the pharmacokinetics of piperaquine in healthy Vietnamese volunteers
Keywords: Malaria; Piperaquine; Food–drug interactions; Pharmacokinetics
Quality control of piperaquine in pharmaceutical formulations by capillary zone electrophoresis
Keywords: Piperaquine; Quality control; Capillary zone electrophoresis; Pharmaceutical formulations
Toxicology and pharmacokinetics of piperaquine in mice
Keywords: Piperaquine; Pharmacokinetics; Toxicology; Mouse
Development and validation of a liquid chromatographic-tandem mass spectrometric method for determination of piperaquine in plasma: Stable isotope labeled internal standard does not always compensate for matrix effects
Keywords: Antimalarial; Differential matrix effect; High throughput; Ion suppression; Liquid chromatography/tandem mass spectrometry (LC-MS/MS); Piperaquine; Stable isotope labeled (SIL) internal standard; Solid-phase extraction
In vitro and in vivo interaction of synthetic peroxide RBx11160 (OZ277) with piperaquine in Plasmodium models
Keywords: Malaria; Plasmodium falciparum; Plasmodium berghei; RBx11160 (OZ277); Peroxide; Piperaquine; In vitro and in vivo combinations; MMV, Medicines for Malaria Venture; Mean ΣFICs; Mean sums of fractional inhibitory concentrations; ACT, artemisinin-based combi
Activity of piperaquine and other 4-aminoquinoline antiplasmodial drugs against chloroquine-sensitive and resistant blood-stages of Plasmodium falciparum: Role of β-haematin inhibition and drug concentration in vacuolar water- and lipid-phases
Keywords: Plasmodium; 4-Aminoquinolines; Piperaquine; Lysosomotropism; Drug-resistance; Hydrophobicity
Identification of an isomer impurity in piperaquine drug substance
Keywords: Antimalarial; Impurity; Positional isomer; Liquid chromatography; MS; NMR; Piperaquine
Development and validation of an automated solid phase extraction and liquid chromatographic method for the determination of piperaquine in urine
Keywords: Piperaquine; Liquid chromatography; Solid-phase extraction; Validation; Method development; Urine;
Safety and efficacy of dihydroartemisinin/piperaquine (Artekin®) for the treatment of uncomplicated Plasmodium falciparum malaria in Rwandan children
Keywords: Malaria; Plasmodium falciparum; Piperaquine; Amodiaquine; Sulfadoxine/pyrimethamine; Rwanda
A new approach to evaluate regression models during validation of bioanalytical assays
Keywords: Bioanalytical assays; Calibration; Transformation; Weighting; Piperaquine; Linear regression; Liquid chromatography
High throughput assay for the determination of piperaquine in plasma
Keywords: Antimalarial; High throughput; Liquid chromatography; Piperaquine; Solid phase extraction; 96-Well;