One-pot α-glycosylation pathway via the generation in situ of α-glycopyranosyl imidates in N,N-dimethylformamide Fulltext Access 9 Pages 2005
The application of phenylmethanethiol and benzenethiol derivatives as odorless organosulfur reagents in the synthesis of thiosugars and thioglycosides Fulltext Access 9 Pages 2005
Synthesis and conformational studies on methyl 4-O-acetyl-3-azido-2,3,6-trideoxy-hex-5-enopyranosides of the l series Fulltext Access 9 Pages 2005
Modeling ring puckering in strained systems: application to 3,6-anhydroglycosides Fulltext Access 9 Pages 2005
Stereospecific synthesis of a new class of compounds: bis-homoconduritol-A, -D, and -F Fulltext Access 9 Pages 2005
Glucose reactions within the heating period and the effect of heating rate on the reactions in hot compressed water Fulltext Access 9 Pages 2005
Dynamic site heterogeneity in amorphous maltose and maltitol from spectral heterogeneity in erythrosin B phosphorescence Fulltext Access 9 Pages 2005
Crystal structure and solid-state 13C NMR analysis of N-p-nitrophenyl-α-d-ribopyranosylamine, N-p-nitrophenyl-α-d-xylopyranosylamine, and solid-state 13C NMR analysis of N-p-nitrophenyl-2,3,4-tri-O-acetyl-β-d-lyxopyranosylamine and N-p-nitrophenyl-2,3,4-t Fulltext Access 9 Pages 2005
Interactions between metal ions and carbohydrates. The coordination behavior of neutral erythritol to lanthanum and erbium ions Fulltext Access 9 Pages 2005
Reactions of d-glucose with phenolic amino acids: further insights into the competition between Maillard and Pictet–Spengler condensation pathways Fulltext Access 9 Pages 2005
Trifluoromethyl group as a pharmacophore: Effect of replacing a CF3 group on binding and agonist activity of a glucocorticoid receptor ligand Fulltext Access 9 Pages 2005
Extraction of leukemia specific glycan motifs in humans by computational glycomics Fulltext Access 9 Pages 2005
Insecticidal anthranilic diamides: A new class of potent ryanodine receptor activators Fulltext Access 9 Pages 2005
3,5-Bicyclic aryl piperidines: A novel class of α4β2 neuronal nicotinic receptor partial agonists for smoking cessation Fulltext Access 9 Pages 2005
Modeling Km values using electrotopological state: Substrates for cytochrome P450 3A4-mediated metabolism Fulltext Access 9 Pages 2005
Docking studies on monoamine oxidase-B inhibitors: Estimation of inhibition constants (Ki) of a series of experimentally tested compounds Fulltext Access 9 Pages 2005
Selective and orally bioavailable phenylglycine tissue factor/factor VIIa inhibitors Fulltext Access 9 Pages 2005
Structure–activity study of epi-gallocatechin gallate (EGCG) analogs as proteasome inhibitors Fulltext Access 9 Pages 2005
Inhibitory effects of 2-substituted-1-naphthol derivatives on cyclooxygenase I and II Fulltext Access 9 Pages 2005
Synthesis of imidazo[1,5,4-de]quinoxalin-9-ones, benzimidazole analogues of pyrroloiminoquinone marine natural products Fulltext Access 9 Pages 2005
Synthesis of a heptasaccharide fragment of the O-deacetylated GXM of C. neoformans serotype C Fulltext Access 9 Pages 2005
Annealing of normal and mutant wheat starches. LM, SEM, DSC, and SAXS studies Fulltext Access 9 Pages 2005
Crystallization and X-ray diffraction of spray-dried and freeze-dried amorphous lactose Fulltext Access 9 Pages 2005
Conformational study of erythritol and threitol in the gas state by density functional theory calculations Fulltext Access 9 Pages 2005
Synthesis and NMR characterization of hydroxyurea and mesylglycol glycoconjugates as drug candidates for targeted cancer chemotherapy Fulltext Access 9 Pages 2005
Rapid synthesis of partially O-methylated alditol acetate standards for GC-MS: some relative activities of hydroxyl groups of methyl glycopyranosides on Purdie methylation Fulltext Access 9 Pages 2005
An α-glucan elicitor from the cell wall of a biocontrol binucleate Rhizoctonia isolate Fulltext Access 9 Pages 2005
The production, purification and characterisation of two novel α-d-mannosidases from Aspergillus phoenicis Fulltext Access 9 Pages 2005
Convenient preparation of 3,5-anhydro- and 2,5-anhydropentofuranosides, and 5,6-anhydro-d-glucofuranose by use of the Mitsunobu reaction Fulltext Access 9 Pages 2005
Stereoselective synthesis, structural characterization, and properties of 1,2-O-isopropylidene-3-C-(5-phenyl-1,2,4-oxadiazol-3-yl)-β-d-psicopyranose Fulltext Access 9 Pages 2005
CP-MLR directed QSAR studies on the antimycobacterial activity of functionalized alkenols-topological descriptors in modeling the activity Fulltext Access 9 Pages 2005
Conformational sampling of the botulinum neurotoxin serotype a light chain: implications for inhibitor binding Fulltext Access 9 Pages 2005
Predicting stability of Arc repressor mutants with protein stochastic moments Fulltext Access 9 Pages 2005
Design, synthesis and photobiological properties of 3,4-cyclopentenepsoralens Fulltext Access 9 Pages 2005
Synthesis and in vitro evaluation of new benzovesamicol analogues as potential imaging probes for the vesicular acetylcholine transporter Fulltext Access 9 Pages 2005
Synthesis and in vivo biodistribution of BPA-Gd-DTPA complex as a potential MRI contrast carrier for neutron capture therapy Fulltext Access 9 Pages 2005
Antileishmanial activity, cytotoxicity and QSAR analysis of synthetic dihydrobenzofuran lignans and related benzofurans Fulltext Access 9 Pages 2005
Ab initio molecular dynamics simulations of β-d-glucose and β-d-xylose degradation mechanisms in acidic aqueous solution Fulltext Access 9 Pages 2005
Synthesis and cytotoxic activity of N-[(alkylamino)alkyl]carboxamide derivatives of 7-oxo-7H-benz[de]anthracene, 7-oxo-7H-naphtho[1,2,3-de]quinoline, and 7-oxo-7H-benzo[e]perimidine Fulltext Access 9 Pages 2005
Synthesis and biological evaluation of novel 6-nitro-5-substituted aminoquinolines as local anesthetic and anti-arrhythmic agents: molecular modeling study Fulltext Access 9 Pages 2005
3D-QSAR studies on c-Src kinase inhibitors and docking analyses of a potent dual kinase inhibitor of c-Src and c-Abl kinases Fulltext Access 9 Pages 2005
Synthesis and C-11 labeling of three potent norepinephrine transporter selective ligands ((R)-nisoxetine, lortalamine, and oxaprotiline) for comparative PET studies in baboons Fulltext Access 9 Pages 2005
Oligonucleotides containing 2′-O-[2-(2,3-dihydroxypropyl)amino-2-oxoethyl]uridine as suitable precursors of 2′-aldehyde oligonucleotides for chemoselective ligation Fulltext Access 9 Pages 2005
Design and synthesis of low molecular weight compounds with complement inhibition activity Fulltext Access 9 Pages 2005
Design, synthesis, and biological evaluation of novel naphthoquinone derivatives with CDC25 phosphatase inhibitory activity Fulltext Access 9 Pages 2005
Synthesis of novel 5-aryl-2-thio-1,3,4-oxadiazoles and the study of their structure–anti-mycobacterial activities Fulltext Access 9 Pages 2005
Synthesis and antileishmanial activities of 4,5-di-substituted acridines as compared to their 4-mono-substituted homologues Fulltext Access 9 Pages 2005
Influence of esterification and modification of A-ring in a group of lupane acids on their cytotoxicity Fulltext Access 9 Pages 2005
Semisynthesis and biological activity of aminoacyl triesters of squamocin, an annonaceous acetogenin Fulltext Access 9 Pages 2005
Synthesis, in vitro, and in vivo characterization of an integrin αvβ3-targeted molecular probe for optical imaging of tumor Fulltext Access 9 Pages 2005
Anti-cancer ProTides: tuning the activity of BVDU phosphoramidates related to thymectacin Fulltext Access 9 Pages 2005
Design, syntheses, and biological evaluations of squamostolide and its related analogs Fulltext Access 9 Pages 2005
Synthesis and evaluation of antioxidative properties of a series of organoselenium compounds Fulltext Access 9 Pages 2005
Synthesis, anti-inflammatory and analgesic activities evaluation of some mono, bi and tricyclic pyrimidine derivatives Fulltext Access 9 Pages 2005
Antiviral cyclic d,l-α-peptides: Targeting a general biochemical pathway in virus infections Fulltext Access 9 Pages 2005
Design and synthesis of labeled analogs of PhTX-56, a potent and selective AMPA receptor antagonist Fulltext Access 9 Pages 2005
8-O-Azeloyl-14-benzoylaconine: A new alkaloid from the roots of Aconitum karacolicum Rapcs and its antiproliferative activities Fulltext Access 9 Pages 2005
Synthesis, antiproliferative, and antiplatelet activities of oxime- and methyloxime-containing flavone and isoflavone derivatives Fulltext Access 9 Pages 2005
Chalcogenoxanthylium photosensitizers for the photodynamic purging of blood-borne viral and bacterial pathogens Fulltext Access 9 Pages 2005
Dicationic near-linear biphenyl benzimidazole derivatives as DNA-targeted antiprotozoal agents Fulltext Access 9 Pages 2005
Synthesis and in vitro anti-mycobacterial activity of 5-substituted pyrimidine nucleosides Fulltext Access 9 Pages 2005
Design and synthesis of glycosidase inhibitor 5-amino-1,2,3,4-cyclohexanetetrol derivatives from (−)-vibo-quercitol Fulltext Access 9 Pages 2005
Synthesis and biological evaluation of 2-aminothiazoles and their amide derivatives on human adenosine receptors. Lack of effect of 2-aminothiazoles as allosteric enhancers Fulltext Access 9 Pages 2005
Synthesis, conformational analysis, and biological activity of new analogues of thiazole-4-carboxamide adenine dinucleotide (TAD) as IMP dehydrogenase inhibitors Fulltext Access 9 Pages 2005
Synthesis and biological activity of fluoroquinolone-pyrrolo[2,1-c][1,4]benzodiazepine conjugates Fulltext Access 9 Pages 2005
Chiral cyclopalladated complexes derived from N,N-dimethyl-1-phenethylamine with bridging bis(diphenylphosphine)ferrocene ligand as inhibitors of the cathepsin B activity and as antitumoral agents Fulltext Access 9 Pages 2005
Synthesis, properties, and photodynamic inactivation of Escherichia coli using a cationic and a noncharged Zn(II) pyridyloxyphthalocyanine derivatives Fulltext Access 9 Pages 2005
[11C]Glycylsarcosine: synthesis and in vivo evaluation as a PET tracer of PepT2 transporter function in kidney of PepT2 null and wild-type mice Fulltext Access 9 Pages 2005
Synthesis and biological evaluation of 3,4-diphenyl-1,2,5-oxadiazole-2-oxides and 3,4-diphenyl-1,2,5-oxadiazoles as potential hybrid COX-2 inhibitor/nitric oxide donor agents Fulltext Access 9 Pages 2005
Design, synthesis, and biological evaluation of 10-methanesulfonyl-DDACTHF, 10-methanesulfonyl-5-DACTHF, and 10-methylthio-DDACTHF as potent inhibitors of GAR Tfase and the de novo purine biosynthetic pathway Fulltext Access 9 Pages 2005
Horseradish peroxidase-mediated aerobic and anaerobic oxidations of 3-alkylindoles Fulltext Access 9 Pages 2005
Mutation of surface cysteine 374 to alanine in monoamine oxidase A alters substrate turnover and inactivation by cyclopropylamines Fulltext Access 9 Pages 2005
Synthesis and antiprotozoan evaluation of new alkyl-linked bis(2-thioxo-[1,3,5]thiadiazinan-3-yl) carboxylic acids Fulltext Access 9 Pages 2005
Design, synthesis, and biological testing of thiosalicylamides as a novel class of calcium channel blockers Fulltext Access 9 Pages 2005
Synthesis of acridinyl-thiazolino derivatives and their evaluation for anti-inflammatory, analgesic and kinase inhibition activities Fulltext Access 9 Pages 2005
3D-QSAR study of bis-azaaromatic quaternary ammonium analogs at the blood-brain barrier choline transporter Fulltext Access 9 Pages 2005
Synthesis of a C-terminally biotinylated macrocyclic peptide mimetic exhibiting high Grb2 SH2 domain-binding affinity Fulltext Access 9 Pages 2005
Radical scavenging activity of dicaffeoyloxycyclohexanes: Contribution of an intramolecular interaction of two caffeoyl residues Fulltext Access 9 Pages 2005
A quantitative structure-activity relationship study on some series of anthranilic acid-based matrix metalloproteinase inhibitors Fulltext Access 9 Pages 2005
Hypocholesterolemic effects of phenolic-rich extracts of Chemlali olive cultivar in rats fed a cholesterol-rich diet Fulltext Access 9 Pages 2005
Bridge-linked bis-quaternary ammonium anti-microbial agents: relationship between cytotoxicity and anti-bacterial activity of 5,5′-[2,2′-(tetramethylenedicarbonyldioxy)-diethyl]bis(3-alkyl-4-methylthiazonium iodide)s Fulltext Access 9 Pages 2005
Porphyrin substituted phosphoramidites: new building blocks for porphyrin–oligonucleotide syntheses Fulltext Access 9 Pages 2005
Quantitative structure–activity relationship to predict differential inhibition of aldose reductase by flavonoid compounds Fulltext Access 9 Pages 2005