Synthesis of d-labeled and unlabeled ethyl succinic anhydrides and application to quantitative analysis of peptides by isotope differential mass spectrometry Fulltext Access 5 Pages 2016
Novel fluorescent substrates for detection of trypsin activity and inhibitor screening by self-quenching Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of heteroaryl styryl sulfone derivatives as anticancer agents Fulltext Access 5 Pages 2016
Identification of lead small molecule inhibitors of glycogen synthase kinase-3 beta using a fragment-linking strategy Fulltext Access 5 Pages 2016
Design, synthesis and transfection efficiency of a novel redox-sensitive polycationic amphiphile Fulltext Access 5 Pages 2016
Parallel inhibition of amino acid efflux and growth of erythrocytic Plasmodium falciparum by mefloquine and non-piperidine analogs: Implication for the mechanism of antimalarial action Fulltext Access 5 Pages 2016
One pot Click chemistry: A three component reaction for the synthesis of 2-mercaptobenzimidazole linked coumarinyl triazoles as anti-tubercular agents Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of the codrug of Leonurine and Aspirin as cardioprotective agents Fulltext Access 5 Pages 2016
Potential therapeutic application of small molecule with sulfonamide for chondrogenic differentiation and articular cartilage repair Fulltext Access 5 Pages 2016
Dihydropyrimidinones and -thiones with improved activity against human polyomavirus family members Fulltext Access 5 Pages 2016
Synthesis of novel arylaminoquinazolinylurea derivatives and their antiproliferative activities against bladder cancer cell line Fulltext Access 5 Pages 2016
Design, synthesis, antibacterial activity and docking study of some new trimethoprim derivatives Fulltext Access 5 Pages 2016
Design, synthesis and structure-activity relationships of novel phenylalanine-based amino acids as kainate receptors ligands Fulltext Access 5 Pages 2016
Synthesis and cytotoxicity study of novel 3-(triazolyl)coumarins based fluorescent scaffolds Fulltext Access 5 Pages 2016
Structure-activity relationship of cyclic pentapeptide malformins as fibrinolysis enhancers Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of ricinoleic acid-based lipoamino acid derivatives Fulltext Access 5 Pages 2016
Synthesis, structure determination, and biological evaluation of phenylsulfonyl hydrazide derivatives as potential anti-inflammatory agents Fulltext Access 5 Pages 2016
Facile analysis of contents and compositions of the chondroitin sulfate/dermatan sulfate hybrid chain in shark and ray tissues Fulltext Access 5 Pages 2016
Formation of isomers of anionic hemiesters of sugars and carbonic acid in aqueous medium Fulltext Access 5 Pages 2016
(7-Diethylaminocoumarin-4-yl)methyl ester of suberoylanilide hydroxamic acid as a caged inhibitor for photocontrol of histone deacetylase activity Fulltext Access 5 Pages 2016
Synthesis, structure and antimicrobial evaluation of a new gossypol triazole conjugates functionalized with aliphatic chains and benzyloxy groups Fulltext Access 5 Pages 2016
Design, synthesis and biological evaluation of photoaffinity probes of antiangiogenic homoisoflavonoids Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of matrine derivatives as anti-hepatocellular cancer agents Fulltext Access 5 Pages 2016
Self-assembling tryptophan-based designer peptides as intracellular delivery vehicles Fulltext Access 5 Pages 2016
Synthesis and biological activity of diisothiocyanate-derived mercapturic acids Fulltext Access 5 Pages 2016
Synthesis and fluorescent study of 5-phenyl furocoumarin derivatives as vasodilatory agents Fulltext Access 5 Pages 2016
Synthesis of novel ethyl 1-ethyl-6-fluoro-7-(fatty amido)-1,4-dihydro-4-oxoquinoline-3-carboxylate derivatives and their biological evaluation Fulltext Access 5 Pages 2016
Synthesis of a new inhibitor of breast cancer resistance protein with significantly improved pharmacokinetic profiles Fulltext Access 5 Pages 2016
Design, synthesis and in vivo screening of some novel quinazoline analogs as anti-hyperlipidemic and hypoglycemic agents Fulltext Access 5 Pages 2016
Increase of rutin antioxidant activity by generating Maillard reaction products with lysine Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of aryloxyacetamide derivatives as neuroprotective agents Fulltext Access 5 Pages 2016
New ligands of the ghrelin receptor based on the 1,2,4-triazole scaffold by introduction of a second chiral center Fulltext Access 5 Pages 2016
Synthesis of 6-phosphofructose aspartic acid and some related Amadori compounds Fulltext Access 5 Pages 2016
A ring closing metathesis strategy for carbapyranosides of xylose and arabinose Fulltext Access 5 Pages 2016
A cell-based approach to characterize antimicrobial compounds through kinetic dose response Fulltext Access 5 Pages 2016
Doped ionic liquid crystals as effective weakly alignment media for polar solutes Fulltext Access 5 Pages 2016
Correlation of transverse relaxation time with structure of biological tissue Fulltext Access 5 Pages 2016
Accelerating flow propagator measurements for the investigation of reactive transport in porous media Fulltext Access 5 Pages 2016
Herbivore-induced volatile organic compounds emitted by maize: Electrophysiological responses in Spodoptera frugiperda females Fulltext Access 5 Pages 2016
Cytotoxic and antimalarial constituents from the roots of Toddalia asiatica Fulltext Access 5 Pages 2016
Rational design and synthesis of novel anti-prostate cancer agents bearing a 3,5-bis-trifluoromethylphenyl moiety Fulltext Access 5 Pages 2016
Synthesis and in vitro evaluation of water-soluble 1,4-diphenethylpiperazine analogs as novel inhibitors of the vesicular monoamine transporter-2 Fulltext Access 5 Pages 2016
Design, synthesis, and protein methyltransferase activity of a unique set of constrained amine containing compounds Fulltext Access 5 Pages 2016
Development of indole sulfonamides as cannabinoid receptor negative allosteric modulators Fulltext Access 5 Pages 2016
Suppression of store overload-induced calcium release by hydroxylated metabolites of carvedilol Fulltext Access 5 Pages 2016
Diversification of edaravone via palladium-catalyzed hydrazine cross-coupling: Applications against protein misfolding and oligomerization of beta-amyloid Fulltext Access 5 Pages 2016
Synthesis and biological evaluation of a novel artesunate–podophyllotoxin conjugate as anticancer agent Fulltext Access 5 Pages 2016
Synthesis, crystal structures, molecular docking, and in vitro biological activities of transition metals with 4-(2,3-dichlorophenyl)piperazine-1-carboxylic acid Fulltext Access 5 Pages 2016
Identification of new quinic acid derivatives as histone deacetylase inhibitors by fluorescence-based cellular assay Fulltext Access 5 Pages 2016
One-pot synthesis and antifungal activity against plant pathogens of quinazolinone derivatives containing an amide moiety Fulltext Access 5 Pages 2016
Synthesis and docking studies of pyrazine–thiazolidinone hybrid scaffold targeting dormant tuberculosis Fulltext Access 5 Pages 2016
Synthesis and activity of benzimidazole-1,3-dioxide inhibitors of separase Fulltext Access 5 Pages 2016
Synthesis of lignan conjugates via cyclopropanation: Antimicrobial and antioxidant studies Fulltext Access 5 Pages 2016
Synthesis and cytotoxic activities of semisynthetic zearalenone analogues Fulltext Access 5 Pages 2016
Design, synthesis, and evaluation of water-soluble morpholino-decorated paclitaxel prodrugs with remarkably decreased toxicity Fulltext Access 5 Pages 2016
An evolved oxazolidinone with selective potency against Mycobacterium tuberculosis and gram positive bacteria Fulltext Access 5 Pages 2016
Synthesis, characterization and anti-cancer activity of a peptide nucleolipid bioconjugate Fulltext Access 5 Pages 2016
Design and synthesis of novel hybrid sydnonimine and prodrug useful for glaucomatous optic neuropathy Fulltext Access 5 Pages 2016
The natural flavone fukugetin as a mixed-type inhibitor for human tissue kallikreins Fulltext Access 5 Pages 2016
Carbohydrate-based inducers of cellular stress for targeting cancer cells Fulltext Access 5 Pages 2016
Anti-inflammatory and antioxidant properties of a novel resveratrol–salicylate hybrid analog Fulltext Access 5 Pages 2016
Synthesis and anti-proliferative activity of fluoro-substituted chalcones Fulltext Access 5 Pages 2016
Development of curcumin–cyclodextrin/cellulose nanocrystals complexes: New anticancer drug delivery systems Fulltext Access 5 Pages 2016
Synthesis, anti-inflammatory, ulcerogenic and cyclooxygenase activities of indenopyrimidine derivatives Fulltext Access 5 Pages 2016
Synthesis, antimicrobial activity of Schiff base compounds of cinnamaldehyde and amino acids Fulltext Access 5 Pages 2016
The semi-synthesis of novel andrographolide analogues and anti-influenza virus activity evaluation of their derivatives Fulltext Access 5 Pages 2016
Carbamate substituted 2-amino-4,6-diphenylpyrimidines as adenosine receptor antagonists Fulltext Access 5 Pages 2016
Design and synthesis of sarolaner, a novel, once-a-month, oral isoxazoline for the control of fleas and ticks on dogs Fulltext Access 5 Pages 2016
Discovery of boronic acid-based fluorescent probes targeting amyloid-beta plaques in Alzheimer’s disease Fulltext Access 5 Pages 2016
Carbon nanodots as molecular scaffolds for development of antimicrobial agents Fulltext Access 5 Pages 2016
Biological evaluation and molecular docking studies of new curcuminoid derivatives: Synthesis and characterization Fulltext Access 5 Pages 2016
Optimization of isoxazoline amide benzoxaboroles for identification of a development candidate as an oral long acting animal ectoparasiticide Fulltext Access 5 Pages 2016
Antibacterial and antifungal activities of 2,3-pyrrolidinedione derivatives against oral pathogens Fulltext Access 5 Pages 2016
Sequential one-pot synthesis of bis(indolyl)glyoxylamides: Evaluation of antibacterial and anticancer activities Fulltext Access 5 Pages 2016
Quinazolinones–Phenylquinoxaline hybrids with unsaturation/saturation linkers as novel anti-proliferative agents Fulltext Access 5 Pages 2016
Solubility-driven lead optimisation: Recent examples and personal perspectives Fulltext Access 5 Pages 2016
Synthesis, biological evaluation and molecular docking of 2-phenyl-benzo[d]oxazole-7-carboxamide derivatives as potential Staphylococcus aureus Sortase A inhibitors Fulltext Access 5 Pages 2016
Cationic lioposomes with folic acid as targeting ligand for gene delivery Fulltext Access 5 Pages 2016
Antioxidant properties of thio-caffeine derivatives: Identification of the newly synthesized 8-[(pyrrolidin-1-ylcarbonothioyl)sulfanyl]caffeine as antioxidant and highly potent cytoprotective agent Fulltext Access 5 Pages 2016
Synthesis and evaluation of novel 1,2,3-triazole-based acetylcholinesterase inhibitors with neuroprotective activity Fulltext Access 5 Pages 2016
Pyridazinone substituted benzenesulfonamides as potent carbonic anhydrase inhibitors Fulltext Access 5 Pages 2016
Polycyclic amines as chloroquine resistance modulating agents in Plasmodium falciparum Fulltext Access 5 Pages 2016